Drug Gene Type Source medazepam AKR1C1 Text_Mining(decreases(activity)) CTD medazepam AKR1C2 Text_Mining(decreases(activity)) CTD medazepam AKR1C3 Text_Mining(decreases(activity)) CTD medazepam AKR1C4 Text_Mining(decreases(activity)) CTD medazepam CYP3A4 Text_Mining(increases(expression)) CTD medazepam NR1I2 Text_Mining(affects(binding)) CTD medazepam NR1I2 Text_Mining(increases(activity)) CTD