Drug Gene Type Source maprotiline BECN1 Text_Mining(increases(expression)) CTD maprotiline KCNH2 Text_Mining(decreases(reaction)) CTD maprotiline KCNH2 Text_Mining(increases(transport)) CTD maprotiline SLC22A2 Text_Mining(decreases(reaction)) CTD maprotiline SLC22A2 Text_Mining(increases(uptake)) CTD maprotiline AR AR Potency (uM)=33.4915(uM) D4 PubChem maprotiline ATXN2 Potency=15.8489(uM) D4 PubChem maprotiline ATXN2 Potency=31.6228(uM) D4 PubChem maprotiline CHRM1 None=None(uM) D4 PubChem maprotiline CHRM4 None=None(uM) D4 PubChem maprotiline CHRM5 None=None(uM) D4 PubChem maprotiline CYP1A2 Inhibition=None(Unspecified) D4 ChEMBL maprotiline CYP2C9 Inhibition=None(Unspecified) D4 ChEMBL maprotiline CYP2D6 Potency=3.9811(uM) D4 PubChem maprotiline CYP2D6 Potency=12.5893(uM) D4 PubChem maprotiline CYP2D6 None=None(uM) D4 PubChem maprotiline CYP2D6 AC50=3981.07(nM) D4 ChEMBL maprotiline CYP2D6 Inhibition=None(Unspecified) D4 ChEMBL maprotiline CYP2D6 Potency=3981.1(nM) D4 ChEMBL maprotiline CYP2D6 AC50=12589.2(nM) D4 ChEMBL maprotiline CYP2D6 Potency=12589.3(nM) D4 ChEMBL maprotiline CYP3A4 Potency=2.5119(uM) D4 PubChem maprotiline CYP3A4 Potency=3.1623(uM) D4 PubChem maprotiline CYP3A4 None=None(uM) D4 PubChem maprotiline CYP3A4 AC50=3162.28(nM) D4 ChEMBL maprotiline CYP3A4 AC50=2511.89(nM) D4 ChEMBL maprotiline CYP3A4 Potency=3162.3(nM) D4 ChEMBL maprotiline CYP3A4 Potency=2511.9(nM) D4 ChEMBL maprotiline DRD1 Potency=2.2387(uM) D4 PubChem maprotiline DRD1 Potency=11.2202(uM) D4 PubChem maprotiline DRD1 Potency=11220.2(nM) D4 ChEMBL maprotiline DRD1 Potency=2238.7(nM) D4 ChEMBL maprotiline DRD3 None=None(uM) D4 PubChem maprotiline MAPT None=None(uM) D4 PubChem maprotiline MTOR Potency=0.5212(uM) D4 PubChem maprotiline MTOR Potency=521.2(nM) D4 ChEMBL maprotiline PPARG Potency-Replicate_1=13.3322(uM) D4 PubChem maprotiline PPARG None=None(uM) D4 PubChem maprotiline TDP1 Potency=9.4411(uM) D4 PubChem maprotiline TDP1 Potency=11.8856(uM) D4 PubChem maprotiline TDP1 Potency=16.3601(uM) D4 PubChem maprotiline TDP1 Potency=21.136(uM) D4 PubChem maprotiline TP53 Potency=31.6228(uM) D4 PubChem maprotiline TP53 Potency=31622.8(nM) D4 ChEMBL maprotiline TSHR Potency=39.8107(uM) D4 PubChem maprotiline TSHR Potency=39810.7(nM) D4 ChEMBL maprotiline WHSC1 None=None(uM) D4 PubChem