Drug Gene Type Source lovastatin ABCA1 Text_Mining(increases(expression)) CTD lovastatin ABCB1 Text_Mining(increases(transport)) CTD lovastatin ABCB1 Text_Mining(decreases(reaction)) CTD lovastatin ABCB1 Text_Mining(decreases(activity)) CTD lovastatin ABCB11 Text_Mining(decreases(reaction)) CTD lovastatin ABCB11 Text_Mining(increases(transport)) CTD lovastatin ABCB11 Text_Mining(decreases(activity)) CTD lovastatin ABCC2 Text_Mining(affects(binding)) CTD lovastatin ABCC2 Text_Mining(increases(uptake)) CTD lovastatin ABCC2 Text_Mining(decreases(reaction)) CTD lovastatin ABCC2 Text_Mining(increases(transport)) CTD lovastatin ABCC2 Text_Mining(decreases(activity)) CTD lovastatin ACTA2 Text_Mining(decreases(reaction)) CTD lovastatin ACTA2 Text_Mining(increases(expression)) CTD lovastatin ACTA2 Text_Mining(decreases(expression)) CTD lovastatin AKAP7 Text_Mining(decreases(response to substance)) CTD lovastatin AKT1 Text_Mining(decreases(reaction)) CTD lovastatin AKT1 Text_Mining(increases(phosphorylation)) CTD lovastatin AKT1 Text_Mining(decreases(phosphorylation)) CTD lovastatin ANK2 Text_Mining(decreases(response to substance)) CTD lovastatin APOA1 Text_Mining(affects(cotreatment)) CTD lovastatin APOA1 Text_Mining(increases(expression)) CTD lovastatin APOB Text_Mining(decreases(secretion)) CTD lovastatin APOB Text_Mining(affects(cotreatment)) CTD lovastatin APOB Text_Mining(decreases(expression)) CTD lovastatin BAX Text_Mining(increases(expression)) CTD lovastatin BCL2 Text_Mining(decreases(expression)) CTD lovastatin BCL2 Text_Mining(decreases(reaction)) CTD lovastatin BCL2L11 Text_Mining(decreases(reaction)) CTD lovastatin BCL2L11 Text_Mining(increases(expression)) CTD lovastatin BIRC5 Text_Mining(decreases(expression)) CTD lovastatin BIRC5 Text_Mining(decreases(reaction)) CTD lovastatin CASP2 Text_Mining(increases(activity)) CTD lovastatin CASP3 Text_Mining(decreases(reaction)) CTD lovastatin CASP3 Text_Mining(increases(activity)) CTD lovastatin CASP3 Text_Mining(increases(cleavage)) CTD lovastatin CASP6 Text_Mining(increases(activity)) CTD lovastatin CASP8 Text_Mining(increases(activity)) CTD lovastatin CASP9 Text_Mining(increases(activity)) CTD lovastatin CCND1 Text_Mining(decreases(expression)) CTD lovastatin CCND3 Text_Mining(decreases(expression)) CTD lovastatin CD44 Text_Mining(decreases(expression)) CTD lovastatin CDC42 Text_Mining(increases(expression)) CTD lovastatin CDK2 Text_Mining(decreases(activity)) CTD lovastatin CDKN1A Text_Mining(increases(expression)) CTD lovastatin CDKN1B Text_Mining(increases(expression)) CTD lovastatin CENPF Text_Mining(increases(expression)) CTD lovastatin CENPF Text_Mining(increases(reaction)) CTD lovastatin CENPF Text_Mining(decreases(reaction)) CTD lovastatin CHEK1 Text_Mining(decreases(reaction)) CTD lovastatin CHEK1 Text_Mining(increases(phosphorylation)) CTD lovastatin CTNNB1 Text_Mining(affects(localization)) CTD lovastatin CTNNB1 Text_Mining(increases(expression)) CTD lovastatin CYP2C8 Text_Mining(decreases(activity)) CTD lovastatin CYP3A4 Text_Mining(increases(activity)) CTD lovastatin CYP3A4 Text_Mining(increases(expression)) CTD lovastatin EAF2 Text_Mining(decreases(response to substance)) CTD lovastatin EGF Text_Mining(decreases(reaction)) CTD lovastatin EGF Text_Mining(increases(phosphorylation)) CTD lovastatin EGF Text_Mining(increases(reaction)) CTD lovastatin EGFR Text_Mining(decreases(reaction)) CTD lovastatin EGFR Text_Mining(increases(phosphorylation)) CTD lovastatin EGFR Text_Mining(increases(reaction)) CTD lovastatin FAS Text_Mining(decreases(reaction)) CTD lovastatin FAS Text_Mining(increases(expression)) CTD lovastatin FASLG Text_Mining(decreases(reaction)) CTD lovastatin FASLG Text_Mining(increases(expression)) CTD lovastatin FASN Text_Mining(increases(expression)) CTD lovastatin FDFT1 Text_Mining(increases(activity)) CTD lovastatin GAP43 Text_Mining(increases(expression)) CTD lovastatin GSK3B Text_Mining(decreases(phosphorylation)) CTD lovastatin H2AFX Text_Mining(decreases(reaction)) CTD lovastatin H2AFX Text_Mining(increases(phosphorylation)) CTD lovastatin HMGCR Text_Mining(decreases(reaction)) CTD lovastatin HMGCR Text_Mining(increases(abundance)) CTD lovastatin HMGCR Text_Mining(decreases(activity)) CTD lovastatin HMGCR Text_Mining(decreases(abundance)) CTD lovastatin HMGCR Text_Mining(increases(expression)) CTD lovastatin HMOX1 Text_Mining(increases(expression)) CTD lovastatin HRAS Text_Mining(decreases(localization)) CTD lovastatin HRAS Text_Mining(decreases(prenylation)) CTD lovastatin INSIG1 Text_Mining(increases(expression)) CTD lovastatin KCNH2 Text_Mining(affects(activity)) CTD lovastatin KRAS Text_Mining(decreases(prenylation)) CTD lovastatin LDLR Text_Mining(increases(activity)) CTD lovastatin LDLR Text_Mining(increases(expression)) CTD lovastatin LDLR Text_Mining(increases(reaction)) CTD lovastatin LEF1 Text_Mining(affects(localization)) CTD lovastatin LMNB1 Text_Mining(affects(localization)) CTD lovastatin LMNB1 Text_Mining(decreases(farnesylation)) CTD lovastatin LMNB1 Text_Mining(increases(degradation)) CTD lovastatin LPA Text_Mining(affects(cotreatment)) CTD lovastatin LPA Text_Mining(decreases(expression)) CTD lovastatin LPIN2 Text_Mining(decreases(response to substance)) CTD lovastatin MAPK1 Text_Mining(decreases(reaction)) CTD lovastatin MAPK1 Text_Mining(increases(phosphorylation)) CTD lovastatin MAPK1 Text_Mining(decreases(activity)) CTD lovastatin MAPK3 Text_Mining(decreases(reaction)) CTD lovastatin MAPK3 Text_Mining(increases(phosphorylation)) CTD lovastatin MAPK3 Text_Mining(decreases(activity)) CTD lovastatin MMP2 Text_Mining(decreases(expression)) CTD lovastatin MMP9 Text_Mining(decreases(expression)) CTD lovastatin NR1I2 Text_Mining(increases(activity)) CTD lovastatin NR1I2 Text_Mining(increases(expression)) CTD lovastatin NRAS Text_Mining(decreases(prenylation)) CTD lovastatin PARVB Text_Mining(decreases(response to substance)) CTD lovastatin PON3 Text_Mining(increases(hydrolysis)) CTD lovastatin PPARG Text_Mining(affects(reaction)) CTD lovastatin PPARG Text_Mining(increases(expression)) CTD lovastatin PTEN Text_Mining(decreases(reaction)) CTD lovastatin PTEN Text_Mining(increases(expression)) CTD lovastatin PTEN Text_Mining(affects(reaction)) CTD lovastatin PTGS2 Text_Mining(decreases(expression)) CTD lovastatin RAC1 Text_Mining(affects(localization)) CTD lovastatin RAC1 Text_Mining(decreases(reaction)) CTD lovastatin RAC1 Text_Mining(decreases(activity)) CTD lovastatin RAC1 Text_Mining(increases(expression)) CTD lovastatin RAF1 Text_Mining(decreases(reaction)) CTD lovastatin RAF1 Text_Mining(increases(phosphorylation)) CTD lovastatin RAF1 Text_Mining(decreases(activity)) CTD lovastatin RAP1A Text_Mining(increases(expression)) CTD lovastatin RB1 Text_Mining(decreases(phosphorylation)) CTD lovastatin RHOA Text_Mining(affects(localization)) CTD lovastatin RHOA Text_Mining(decreases(reaction)) CTD lovastatin RHOA Text_Mining(decreases(prenylation)) CTD lovastatin RHOB Text_Mining(decreases(prenylation)) CTD lovastatin RHOB Text_Mining(increases(expression)) CTD lovastatin SLCO1B1 Text_Mining(decreases(reaction)) CTD lovastatin SLCO1B1 Text_Mining(increases(transport)) CTD lovastatin SLCO1B1 Text_Mining(decreases(activity)) CTD lovastatin SREBF2 Text_Mining(increases(localization)) CTD lovastatin STEAP2 Text_Mining(decreases(response to substance)) CTD lovastatin TG Text_Mining(increases(secretion)) CTD lovastatin TGFB1 Text_Mining(decreases(reaction)) CTD lovastatin TGFB1 Text_Mining(increases(abundance)) CTD lovastatin TGFB1 Text_Mining(increases(expression)) CTD lovastatin TH Text_Mining(increases(expression)) CTD lovastatin TH Text_Mining(decreases(reaction)) CTD lovastatin TNFSF10 Text_Mining(increases(response to substance)) CTD lovastatin TP53 Text_Mining(decreases(reaction)) CTD lovastatin TP53 Text_Mining(increases(expression)) CTD lovastatin TP53 Text_Mining(increases(phosphorylation)) CTD lovastatin ABCB1 None=None(uM) D4 PubChem lovastatin AKT1 Activity=None(Unspecified) D4 ChEMBL lovastatin AR Ratio Potency (uM)=5.26203(uM) D4 PubChem lovastatin CYP19A1 Potency-Replicate_1=11.8832(uM) D4 PubChem lovastatin CYP19A1 Potency-Replicate_1=27.1672(uM) D4 PubChem lovastatin CYP19A1 Potency-Replicate_1=34.859(uM) D4 PubChem lovastatin CYP19A1 None=None(uM) D4 PubChem lovastatin CYP1A2 Inhibition=None(Unspecified) D4 ChEMBL lovastatin CYP2C19 Inhibition=None(Unspecified) D4 ChEMBL lovastatin CYP2C9 Inhibition=None(Unspecified) D4 ChEMBL lovastatin CYP2D6 Inhibition=None(Unspecified) D4 ChEMBL lovastatin CYP3A4 Potency=10.0(uM) D4 PubChem lovastatin CYP3A4 Inhibition=None(Unspecified) D4 ChEMBL lovastatin CYP3A4 Potency=10000.0(nM) D4 ChEMBL lovastatin EHMT2 Potency=15.8489(uM) D4 PubChem lovastatin EHMT2 Potency=15848.9(nM) D4 ChEMBL lovastatin GAPDH None=None(uM) D4 PubChem lovastatin IDH1 Potency=7.3078(uM) D4 PubChem lovastatin IDH1 Potency=18.3564(uM) D4 PubChem lovastatin MDM2 None=None(uM) D4 PubChem lovastatin MDM4 None=None(uM) D4 PubChem lovastatin NFE2L2 Ratio Potency (uM)=30.4821(uM) D4 PubChem lovastatin NR0B1 None=None(uM) D4 PubChem lovastatin NR1I2 Potency-Replicate_1=31.6228(uM) D4 PubChem lovastatin NR3C1 Potency-Replicate_1=21.3138(uM) D4 PubChem lovastatin NR3C1 None=None(uM) D4 PubChem lovastatin SMARCA2 None=None(uM) D4 PubChem lovastatin SMN1; SMN2 Potency=15848.9(nM) D4 ChEMBL lovastatin SMN2 Potency=15.8489(uM) D4 PubChem lovastatin STK33 None=None(uM) D4 PubChem lovastatin TDP1 Potency=11.8856(uM) D4 PubChem lovastatin TDP1 Potency=13.3359(uM) D4 PubChem lovastatin TDP1 Potency=20.5962(uM) D4 PubChem lovastatin TDP1 Potency=25.929(uM) D4 PubChem lovastatin VDR Potency=50.1187(uM) D4 PubChem