Drug Gene Type Source loperamide CES2 Text_Mining(decreases(activity)) CTD loperamide CES2 Text_Mining(increases(response to substance)) CTD loperamide IL2 Text_Mining(decreases(expression)) CTD loperamide IL4 Text_Mining(increases(expression)) CTD loperamide MAPK1 Text_Mining(increases(phosphorylation)) CTD loperamide MAPK3 Text_Mining(increases(phosphorylation)) CTD loperamide NFKBIA Text_Mining(increases(expression)) CTD loperamide NR1I2 Text_Mining(affects(cotreatment)) CTD loperamide NR1I2 Text_Mining(increases(activity)) CTD loperamide NR1I3 Text_Mining(affects(binding)) CTD loperamide NR1I3 Text_Mining(decreases(activity)) CTD loperamide NR1I3 Text_Mining(affects(cotreatment)) CTD loperamide PLD2 Text_Mining(increases(activity)) CTD loperamide SLC22A2 Text_Mining(decreases(reaction)) CTD loperamide SLC22A2 Text_Mining(increases(uptake)) CTD loperamide AR Potency-Replicate_1=26.6032(uM) D4 PubChem loperamide CYP19A1 Potency-Replicate_1=26.6032(uM) D4 PubChem loperamide CYP2D6 Potency=0.0158(uM) D4 PubChem loperamide CYP2D6 Potency=10.0(uM) D4 PubChem loperamide CYP2D6 Potency=25.1189(uM) D4 PubChem loperamide CYP2D6 None=None(uM) D4 PubChem loperamide CYP2D6 AC50=15.85(nM) D4 ChEMBL loperamide CYP2D6 AC50=10000.0(nM) D4 ChEMBL loperamide CYP2D6 Potency=25118.9(nM) D4 ChEMBL loperamide CYP2D6 Potency=15.8(nM) D4 ChEMBL loperamide CYP2D6 AC50=25118.9(nM) D4 ChEMBL loperamide CYP2D6 Potency=10000.0(nM) D4 ChEMBL loperamide CYP3A4 Potency=5.0119(uM) D4 PubChem loperamide CYP3A4 Potency=5011.9(nM) D4 ChEMBL loperamide MTOR Potency=13.0918(uM) D4 PubChem loperamide MTOR Potency=18.4927(uM) D4 PubChem loperamide MTOR Potency=13091.8(nM) D4 ChEMBL loperamide MTOR Potency=18492.7(nM) D4 ChEMBL loperamide PDE4B None=None(uM) D4 PubChem loperamide STK33 None=None(uM) D4 PubChem loperamide TDP1 Potency=6.6838(uM) D4 PubChem loperamide TDP1 Potency=8.4144(uM) D4 PubChem loperamide TDP1 Potency=9.7264(uM) D4 PubChem loperamide TDP1 Potency=23.715(uM) D4 PubChem loperamide TEK Activity=None(Unspecified) D4 ChEMBL loperamide TP53 Potency=31.6228(uM) D4 PubChem loperamide TP53 Potency=31622.8(nM) D4 ChEMBL loperamide TSHR Potency=1.2589(uM) D4 PubChem loperamide TSHR Potency=1258.9(nM) D4 ChEMBL