Drug Gene Type Source flurbiprofen AKR1C1 Text_Mining(decreases(activity)) CTD flurbiprofen AKR1C2 Text_Mining(decreases(activity)) CTD flurbiprofen AKR1C3 Text_Mining(decreases(activity)) CTD flurbiprofen AKR1C3 Text_Mining(increases(chemical synthesis)) CTD flurbiprofen AKR1C3 Text_Mining(increases(metabolic processing)) CTD flurbiprofen ALB Text_Mining(affects(binding)) CTD flurbiprofen APP Text_Mining(decreases(reaction)) CTD flurbiprofen APP Text_Mining(decreases(secretion)) CTD flurbiprofen APP Text_Mining(affects(cotreatment)) CTD flurbiprofen APP Text_Mining(increases(secretion)) CTD flurbiprofen APP Text_Mining(increases(reaction)) CTD flurbiprofen CCNB1 Text_Mining(decreases(expression)) CTD flurbiprofen CYP2C9 Text_Mining(decreases(reaction)) CTD flurbiprofen CYP2C9 Text_Mining(increases(hydroxylation)) CTD flurbiprofen CYP2C9 Text_Mining(affects(hydroxylation)) CTD flurbiprofen CYP2C9 Text_Mining(increases(reaction)) CTD flurbiprofen CYP2C9 Text_Mining(affects(hydrolysis)) CTD flurbiprofen CYP2C9 Text_Mining(affects(metabolic processing)) CTD flurbiprofen CYP2C9 Text_Mining(increases(hydrolysis)) CTD flurbiprofen CYP2C9 Text_Mining(increases(metabolic processing)) CTD flurbiprofen CYP2C9 Text_Mining(affects(reaction)) CTD flurbiprofen CYP2C9 Text_Mining(affects(binding)) CTD flurbiprofen EIF4E Text_Mining(increases(phosphorylation)) CTD flurbiprofen EIF4E Text_Mining(increases(reaction)) CTD flurbiprofen ELAVL1 Text_Mining(increases(expression)) CTD flurbiprofen ELAVL1 Text_Mining(increases(reaction)) CTD flurbiprofen ELAVL1 Text_Mining(affects(binding)) CTD flurbiprofen FOS Text_Mining(decreases(reaction)) CTD flurbiprofen FOS Text_Mining(increases(expression)) CTD flurbiprofen GDF15 Text_Mining(decreases(reaction)) CTD flurbiprofen GDF15 Text_Mining(increases(expression)) CTD flurbiprofen GDF15 Text_Mining(increases(reaction)) CTD flurbiprofen HPGD Text_Mining(decreases(degradation)) CTD flurbiprofen HPGD Text_Mining(increases(activity)) CTD flurbiprofen HPGD Text_Mining(increases(expression)) CTD flurbiprofen HPGD Text_Mining(decreases(expression)) CTD flurbiprofen IFNG Text_Mining(affects(cotreatment)) CTD flurbiprofen IFNG Text_Mining(decreases(reaction)) CTD flurbiprofen IFNG Text_Mining(increases(secretion)) CTD flurbiprofen IL1B Text_Mining(decreases(reaction)) CTD flurbiprofen IL1B Text_Mining(increases(expression)) CTD flurbiprofen IL1B Text_Mining(increases(chemical synthesis)) CTD flurbiprofen IL1B Text_Mining(increases(reaction)) CTD flurbiprofen MAPK1 Text_Mining(decreases(activity)) CTD flurbiprofen MAPK1 Text_Mining(decreases(phosphorylation)) CTD flurbiprofen MAPK11 Text_Mining(increases(expression)) CTD flurbiprofen MAPK11 Text_Mining(increases(reaction)) CTD flurbiprofen MAPK14 Text_Mining(increases(expression)) CTD flurbiprofen MAPK14 Text_Mining(increases(reaction)) CTD flurbiprofen MAPK14 Text_Mining(increases(phosphorylation)) CTD flurbiprofen MAPK3 Text_Mining(decreases(activity)) CTD flurbiprofen MAPK3 Text_Mining(decreases(phosphorylation)) CTD flurbiprofen MAPKAPK2 Text_Mining(increases(activity)) CTD flurbiprofen MAPKAPK2 Text_Mining(increases(phosphorylation)) CTD flurbiprofen MAPKAPK2 Text_Mining(increases(expression)) CTD flurbiprofen MAPKAPK2 Text_Mining(increases(reaction)) CTD flurbiprofen MAPKAPK3 Text_Mining(increases(expression)) CTD flurbiprofen MAPKAPK3 Text_Mining(increases(reaction)) CTD flurbiprofen MMP9 Text_Mining(decreases(expression)) CTD flurbiprofen MMP9 Text_Mining(increases(expression)) CTD flurbiprofen MMP9 Text_Mining(decreases(degradation)) CTD flurbiprofen NGFR Text_Mining(decreases(reaction)) CTD flurbiprofen NGFR Text_Mining(increases(expression)) CTD flurbiprofen NGFR Text_Mining(increases(reaction)) CTD flurbiprofen NGFR Text_Mining(affects(binding)) CTD flurbiprofen NGFR Text_Mining(increases(stability)) CTD flurbiprofen NQO1 Text_Mining(increases(activity)) CTD flurbiprofen PLA2G4A Text_Mining(decreases(reaction)) CTD flurbiprofen PLA2G4A Text_Mining(increases(expression)) CTD flurbiprofen PTGS1 Text_Mining(decreases(activity)) CTD flurbiprofen PTGS2 Text_Mining(decreases(reaction)) CTD flurbiprofen PTGS2 Text_Mining(increases(expression)) CTD flurbiprofen PTGS2 Text_Mining(increases(chemical synthesis)) CTD flurbiprofen PTGS2 Text_Mining(increases(reaction)) CTD flurbiprofen PTGS2 Text_Mining(decreases(activity)) CTD flurbiprofen PTGS2 Text_Mining(increases(activity)) CTD flurbiprofen RXRA Text_Mining(affects(binding)) CTD flurbiprofen RXRA Text_Mining(decreases(reaction)) CTD flurbiprofen RXRA Text_Mining(decreases(secretion)) CTD flurbiprofen RXRA Text_Mining(increases(reaction)) CTD flurbiprofen SELL Text_Mining(decreases(expression)) CTD flurbiprofen TIMP1 Text_Mining(increases(expression)) CTD flurbiprofen TIMP1 Text_Mining(decreases(expression)) CTD flurbiprofen TIMP1 Text_Mining(decreases(degradation)) CTD flurbiprofen TNF Text_Mining(affects(cotreatment)) CTD flurbiprofen TNF Text_Mining(decreases(reaction)) CTD flurbiprofen TNF Text_Mining(increases(secretion)) CTD flurbiprofen TP53 Text_Mining(increases(abundance)) CTD flurbiprofen TP53 Text_Mining(increases(phosphorylation)) CTD flurbiprofen TP53 Text_Mining(increases(expression)) CTD flurbiprofen TP53 Text_Mining(decreases(response to substance)) CTD flurbiprofen TP53 Text_Mining(increases(response to substance)) CTD flurbiprofen UGT1A1 Text_Mining(increases(glucuronidation)) CTD flurbiprofen UGT1A10 Text_Mining(increases(glucuronidation)) CTD flurbiprofen UGT1A3 Text_Mining(increases(glucuronidation)) CTD flurbiprofen UGT1A4 Text_Mining(increases(glucuronidation)) CTD flurbiprofen UGT1A6 Text_Mining(increases(glucuronidation)) CTD flurbiprofen UGT1A7 Text_Mining(increases(glucuronidation)) CTD flurbiprofen UGT1A8 Text_Mining(increases(glucuronidation)) CTD flurbiprofen UGT1A9 Text_Mining(increases(glucuronidation)) CTD flurbiprofen UGT2B4 Text_Mining(increases(glucuronidation)) CTD flurbiprofen UGT2B7 Text_Mining(increases(glucuronidation)) CTD flurbiprofen ESR1 Potency-Replicate_1=4.522(uM) D4 PubChem flurbiprofen PPARG Ratio Potency (uM)=None(uM) D4 PubChem flurbiprofen PPARG None=None(uM) D4 PubChem flurbiprofen PRKACB None=None(uM) D4 PubChem flurbiprofen PRKAR2B None=None(uM) D4 PubChem flurbiprofen PTGS2 Inhibition=None(Unspecified) D4 ChEMBL