Drug Gene Type Source desipramine ALPP Text_Mining(decreases(reaction)) CTD desipramine ALPP Text_Mining(increases(expression)) CTD desipramine CASP3 Text_Mining(increases(activity)) CTD desipramine CASP3 Text_Mining(increases(reaction)) CTD desipramine CCL5 Text_Mining(decreases(reaction)) CTD desipramine CCL5 Text_Mining(increases(expression)) CTD desipramine CYP2A6 Text_Mining(decreases(activity)) CTD desipramine CYP2C19 Text_Mining(decreases(activity)) CTD desipramine CYP2C9 Text_Mining(decreases(activity)) CTD desipramine CYP2D6 Text_Mining(affects(metabolic processing)) CTD desipramine CYP2E1 Text_Mining(decreases(activity)) CTD desipramine CYP3A4 Text_Mining(increases(response to substance)) CTD desipramine CYP3A4 Text_Mining(decreases(activity)) CTD desipramine HTR1A Text_Mining(decreases(expression)) CTD desipramine HTR1A Text_Mining(decreases(reaction)) CTD desipramine IFNA1 Text_Mining(decreases(expression)) CTD desipramine IFNA1 Text_Mining(decreases(reaction)) CTD desipramine MAPK8 Text_Mining(increases(phosphorylation)) CTD desipramine MAPK8 Text_Mining(increases(reaction)) CTD desipramine MAPK8 Text_Mining(increases(activity)) CTD desipramine KCNH2 Text_Mining(decreases(activity)) CTD desipramine MAPK1 Text_Mining(increases(activity)) CTD desipramine MAPK14 Text_Mining(increases(activity)) CTD desipramine MAPK3 Text_Mining(increases(activity)) CTD desipramine NFE2L2 Text_Mining(affects(response to substance)) CTD desipramine NR3C1 Text_Mining(decreases(expression)) CTD desipramine NR3C1 Text_Mining(decreases(reaction)) CTD desipramine SLC22A2 Text_Mining(decreases(reaction)) CTD desipramine SLC22A2 Text_Mining(increases(uptake)) CTD desipramine SLC6A2 Text_Mining(decreases(reaction)) CTD desipramine SLC6A2 Text_Mining(increases(activity)) CTD desipramine SLC6A2 Text_Mining(increases(reaction)) CTD desipramine SMPD1 Text_Mining(decreases(activity)) CTD desipramine TAAR1 Text_Mining(decreases(reaction)) CTD desipramine TAAR1 Text_Mining(increases(activity)) CTD desipramine TAAR1 Text_Mining(increases(reaction)) CTD desipramine TNF Text_Mining(decreases(reaction)) CTD desipramine TNF Text_Mining(increases(expression)) CTD desipramine TNF Text_Mining(decreases(activity)) CTD desipramine ARSA Potency=21.3313(uM) D4 PubChem desipramine CYP1A2 None=None(uM) D4 PubChem desipramine CYP2D6 Potency=3.9811(uM) D4 PubChem desipramine CYP2D6 Potency=25.1189(uM) D4 PubChem desipramine CYP2D6 None=None(uM) D4 PubChem desipramine CYP2D6 Potency=3981.1(nM) D4 ChEMBL desipramine CYP2D6 AC50=3981.07(nM) D4 ChEMBL desipramine CYP2D6 AC50=25118.9(nM) D4 ChEMBL desipramine CYP2D6 Potency=25118.9(nM) D4 ChEMBL desipramine CYP3A4 Potency=19.9526(uM) D4 PubChem desipramine CYP3A4 None=None(uM) D4 PubChem desipramine CYP3A4 AC50=19952.6(nM) D4 ChEMBL desipramine CYP3A4 Potency=19952.6(nM) D4 ChEMBL desipramine SLC6A2 Activity=None(Unspecified) D4 ChEMBL desipramine THPO Potency=12.5893(uM) D4 PubChem desipramine THPO Potency=12589.3(nM) D4 ChEMBL