Drug Gene Type Source colchicine ABCB1 Text_Mining(affects(transport)) CTD colchicine ABCB1 Text_Mining(decreases(response to substance)) CTD colchicine ABCB1 Text_Mining(increases(export)) CTD colchicine ABCB1 Text_Mining(decreases(reaction)) CTD colchicine ABCB1 Text_Mining(increases(activity)) CTD colchicine ABCB1 Text_Mining(increases(expression)) CTD colchicine ABCB1 Text_Mining(affects(cotreatment)) CTD colchicine ABCC1 Text_Mining(decreases(response to substance)) CTD colchicine AHR Text_Mining(decreases(activity)) CTD colchicine ALB Text_Mining(affects(expression)) CTD colchicine ATXN1 Text_Mining(decreases(expression)) CTD colchicine AURKB Text_Mining(increases(expression)) CTD colchicine BAX Text_Mining(increases(expression)) CTD colchicine BCL2 Text_Mining(decreases(expression)) CTD colchicine BLM Text_Mining(decreases(expression)) CTD colchicine BTG1 Text_Mining(decreases(expression)) CTD colchicine BTG2 Text_Mining(decreases(expression)) CTD colchicine BTG3 Text_Mining(decreases(expression)) CTD colchicine C12ORF5 Text_Mining(decreases(expression)) CTD colchicine C7ORF26 Text_Mining(decreases(expression)) CTD colchicine CASP3 Text_Mining(increases(activity)) CTD colchicine CASP9 Text_Mining(increases(activity)) CTD colchicine CCDC51 Text_Mining(decreases(expression)) CTD colchicine CCNB1 Text_Mining(increases(expression)) CTD colchicine CCNE2 Text_Mining(decreases(expression)) CTD colchicine CD59 Text_Mining(increases(mutagenesis)) CTD colchicine CDC25A Text_Mining(decreases(expression)) CTD colchicine CDC6 Text_Mining(decreases(expression)) CTD colchicine CDH1 Text_Mining(affects(activity)) CTD colchicine CDKN1A Text_Mining(decreases(expression)) CTD colchicine CELF2 Text_Mining(decreases(reaction)) CTD colchicine CELF2 Text_Mining(increases(expression)) CTD colchicine CHAF1A Text_Mining(decreases(expression)) CTD colchicine CHAF1B Text_Mining(decreases(expression)) CTD colchicine CLN8 Text_Mining(decreases(expression)) CTD colchicine COA7 Text_Mining(decreases(expression)) CTD colchicine CPT2 Text_Mining(decreases(expression)) CTD colchicine CSF2 Text_Mining(decreases(reaction)) CTD colchicine CSF2 Text_Mining(increases(secretion)) CTD colchicine CYP1A1 Text_Mining(decreases(reaction)) CTD colchicine CYP1A1 Text_Mining(increases(activity)) CTD colchicine CYP1A1 Text_Mining(increases(expression)) CTD colchicine CYP3A4 Text_Mining(affects(metabolic processing)) CTD colchicine DDIT4 Text_Mining(decreases(expression)) CTD colchicine DUSP14 Text_Mining(decreases(expression)) CTD colchicine E2F1 Text_Mining(decreases(expression)) CTD colchicine ENC1 Text_Mining(decreases(expression)) CTD colchicine F2 Text_Mining(affects(activity)) CTD colchicine FDXR Text_Mining(decreases(expression)) CTD colchicine FOXJ2 Text_Mining(decreases(expression)) CTD colchicine FTSJ2 Text_Mining(decreases(expression)) CTD colchicine FZD1 Text_Mining(decreases(expression)) CTD colchicine GCH1 Text_Mining(decreases(expression)) CTD colchicine GDF15 Text_Mining(decreases(expression)) CTD colchicine GRPEL1 Text_Mining(decreases(expression)) CTD colchicine ID3 Text_Mining(decreases(expression)) CTD colchicine IKBKB Text_Mining(affects(binding)) CTD colchicine IKBKB Text_Mining(decreases(localization)) CTD colchicine IKBKB Text_Mining(increases(phosphorylation)) CTD colchicine IL1A Text_Mining(decreases(reaction)) CTD colchicine IL1A Text_Mining(increases(expression)) CTD colchicine IL2 Text_Mining(decreases(expression)) CTD colchicine ISG20L2 Text_Mining(decreases(expression)) CTD colchicine JUN Text_Mining(increases(phosphorylation)) CTD colchicine JUN Text_Mining(affects(reaction)) CTD colchicine KIF20A Text_Mining(decreases(expression)) CTD colchicine KLF6 Text_Mining(increases(expression)) CTD colchicine KRT18 Text_Mining(decreases(expression)) CTD colchicine LHX2 Text_Mining(decreases(expression)) CTD colchicine LRRC47 Text_Mining(decreases(expression)) CTD colchicine MAPK8 Text_Mining(increases(phosphorylation)) CTD colchicine MAPK8 Text_Mining(affects(reaction)) CTD colchicine MAPK9 Text_Mining(increases(phosphorylation)) CTD colchicine MAPK9 Text_Mining(affects(reaction)) CTD colchicine MAPT Text_Mining(decreases(expression)) CTD colchicine MCM10 Text_Mining(decreases(expression)) CTD colchicine MGMT Text_Mining(affects(cotreatment)) CTD colchicine MGMT Text_Mining(decreases(response to substance)) CTD colchicine MSH6 Text_Mining(decreases(expression)) CTD colchicine MYT1 Text_Mining(increases(phosphorylation)) CTD colchicine NFATC4 Text_Mining(decreases(localization)) CTD colchicine NFKBIA Text_Mining(affects(binding)) CTD colchicine NFKBIA Text_Mining(decreases(localization)) CTD colchicine NFKBIA Text_Mining(increases(phosphorylation)) CTD colchicine NR3C1 Text_Mining(decreases(activity)) CTD colchicine NR3C1 Text_Mining(decreases(localization)) CTD colchicine NR3C1 Text_Mining(increases(activity)) CTD colchicine NR3C1 Text_Mining(increases(degradation)) CTD colchicine ORAI3 Text_Mining(decreases(expression)) CTD colchicine PALB2 Text_Mining(decreases(expression)) CTD colchicine PELO Text_Mining(decreases(expression)) CTD colchicine PHLDA3 Text_Mining(decreases(expression)) CTD colchicine PIDD1 Text_Mining(decreases(expression)) CTD colchicine PLEKHF1 Text_Mining(decreases(expression)) CTD colchicine PLXNB2 Text_Mining(decreases(expression)) CTD colchicine PPM1D Text_Mining(decreases(expression)) CTD colchicine PRKAB1 Text_Mining(decreases(expression)) CTD colchicine PSMC3IP Text_Mining(decreases(expression)) CTD colchicine PTK2B Text_Mining(decreases(reaction)) CTD colchicine PTK2B Text_Mining(increases(phosphorylation)) CTD colchicine PTP4A1 Text_Mining(decreases(expression)) CTD colchicine PUS3 Text_Mining(decreases(expression)) CTD colchicine RAD51C Text_Mining(decreases(expression)) CTD colchicine RALBP1 Text_Mining(affects(transport)) CTD colchicine RALBP1 Text_Mining(decreases(reaction)) CTD colchicine RAP2B Text_Mining(decreases(expression)) CTD colchicine RBM34 Text_Mining(decreases(expression)) CTD colchicine RFC1 Text_Mining(decreases(expression)) CTD colchicine RGS16 Text_Mining(decreases(expression)) CTD colchicine RNF113A Text_Mining(decreases(expression)) CTD colchicine RNF19B Text_Mining(decreases(expression)) CTD colchicine SAC3D1 Text_Mining(decreases(expression)) CTD colchicine SDC1 Text_Mining(decreases(expression)) CTD colchicine SDHAF1 Text_Mining(decreases(expression)) CTD colchicine SESN1 Text_Mining(decreases(expression)) CTD colchicine SGK1 Text_Mining(decreases(expression)) CTD colchicine SLBP Text_Mining(decreases(expression)) CTD colchicine SLC1A5 Text_Mining(decreases(expression)) CTD colchicine TAT Text_Mining(decreases(expression)) CTD colchicine TAT Text_Mining(decreases(reaction)) CTD colchicine TIPIN Text_Mining(decreases(expression)) CTD colchicine TMEM185B Text_Mining(decreases(expression)) CTD colchicine TNF Text_Mining(decreases(reaction)) CTD colchicine TNF Text_Mining(increases(expression)) CTD colchicine TNF Text_Mining(decreases(expression)) CTD colchicine TNFRSF10B Text_Mining(decreases(expression)) CTD colchicine TNFSF9 Text_Mining(decreases(expression)) CTD colchicine TOP3A Text_Mining(decreases(expression)) CTD colchicine TOR1A Text_Mining(decreases(expression)) CTD colchicine TP53 Text_Mining(affects(reaction)) CTD colchicine TP53 Text_Mining(increases(phosphorylation)) CTD colchicine TRIAP1 Text_Mining(decreases(expression)) CTD colchicine TRIM22 Text_Mining(decreases(expression)) CTD colchicine TRIM26 Text_Mining(decreases(expression)) CTD colchicine TRIM32 Text_Mining(decreases(expression)) CTD colchicine TRIM38 Text_Mining(decreases(expression)) CTD colchicine UTP3 Text_Mining(decreases(expression)) CTD colchicine VCAM1 Text_Mining(decreases(reaction)) CTD colchicine VCAM1 Text_Mining(increases(expression)) CTD colchicine XPC Text_Mining(decreases(expression)) CTD colchicine ZBED1 Text_Mining(decreases(expression)) CTD colchicine ZBTB24 Text_Mining(decreases(expression)) CTD colchicine ZFP36L1 Text_Mining(decreases(expression)) CTD colchicine ZNF200 Text_Mining(decreases(expression)) CTD colchicine ZNF202 Text_Mining(decreases(expression)) CTD colchicine ZNF232 Text_Mining(decreases(expression)) CTD colchicine ZNF337 Text_Mining(decreases(expression)) CTD colchicine ZNF45 Text_Mining(decreases(expression)) CTD colchicine ZNF544 Text_Mining(decreases(expression)) CTD colchicine AR Ratio Potency (uM)=0.00837973(uM) D4 PubChem colchicine AR Ratio Potency (uM)=0.0171721(uM) D4 PubChem colchicine AR Potency-Replicate_1=0.0601(uM) D4 PubChem colchicine AR Ratio Potency (uM)=0.0674001(uM) D4 PubChem colchicine ATAD5 Potency=0.4609(uM) D4 PubChem colchicine ATAD5 Potency=460.9(nM) D4 ChEMBL colchicine CREBBP Potency=5011.9(nM) D4 ChEMBL colchicine CXCL8 Potency=0.0473(uM) D4 PubChem colchicine CXCL8 Potency=0.0531(uM) D4 PubChem colchicine CYP1A2 Inhibition=None(Unspecified) D4 ChEMBL colchicine CYP2C19 Potency=12.5893(uM) D4 PubChem colchicine CYP2C19 None=None(uM) D4 PubChem colchicine CYP2C19 Inhibition=None(Unspecified) D4 ChEMBL colchicine CYP2C19 AC50=12589.2(nM) D4 ChEMBL colchicine CYP2C19 Potency=12589.3(nM) D4 ChEMBL colchicine CYP2C9 Potency=3.1623(uM) D4 PubChem colchicine CYP2C9 None=None(uM) D4 PubChem colchicine CYP2C9 Inhibition=None(Unspecified) D4 ChEMBL colchicine CYP2C9 AC50=3162.28(nM) D4 ChEMBL colchicine CYP2C9 Potency=3162.3(nM) D4 ChEMBL colchicine CYP2D6 Potency=0.7943(uM) D4 PubChem colchicine CYP2D6 None=None(uM) D4 PubChem colchicine CYP2D6 Inhibition=None(Unspecified) D4 ChEMBL colchicine CYP2D6 Potency=794.3(nM) D4 ChEMBL colchicine CYP2D6 AC50=794.33(nM) D4 ChEMBL colchicine CYP3A4 Inhibition=None(Unspecified) D4 ChEMBL colchicine ESR1 Ratio Potency (uM)=0.0128773(uM) D4 PubChem colchicine ESR1 Potency-Replicate_1=0.0153(uM) D4 PubChem colchicine ESR1 Potency-Replicate_1=0.0427(uM) D4 PubChem colchicine ESR1 ER Potency (uM)=0.0685896(uM) D4 PubChem colchicine ESR1 Potency-Replicate_1=0.0863(uM) D4 PubChem colchicine ESR1 ER Potency (uM)=0.0943918(uM) D4 PubChem colchicine ESR1 ER Potency (uM)=0.0957043(uM) D4 PubChem colchicine ESR1 Potency-Replicate_1=0.1188(uM) D4 PubChem colchicine GMNN Potency=0.0046(uM) D4 PubChem colchicine GMNN Potency=0.0337(uM) D4 PubChem colchicine GMNN Potency=0.0398(uM) D4 PubChem colchicine GMNN Potency=0.0422(uM) D4 PubChem colchicine GMNN Potency=0.0531(uM) D4 PubChem colchicine GMNN Potency=0.058(uM) D4 PubChem colchicine GMNN Potency=39.8(nM) D4 ChEMBL colchicine GMNN Potency=33.7(nM) D4 ChEMBL colchicine GMNN Potency=58.0(nM) D4 ChEMBL colchicine KLF5 None=None(uM) D4 PubChem colchicine MDM2 None=None(uM) D4 PubChem colchicine MDM4 None=None(uM) D4 PubChem colchicine NFE2L2 Ratio Potency (uM)=0.029847(uM) D4 PubChem colchicine NFE2L2 Ratio Potency (uM)=0.0364132(uM) D4 PubChem colchicine NFE2L2 Ratio Potency (uM)=0.0381006(uM) D4 PubChem colchicine NFE2L2 Potency=0.075(uM) D4 PubChem colchicine NR0B1 None=None(uM) D4 PubChem colchicine NR1H4 None=None(uM) D4 PubChem colchicine PAX8 AC50_uM=0.26(uM) D4 PubChem colchicine PAX8 None=None(uM) D4 PubChem colchicine STK33 None=None(uM) D4 PubChem colchicine TDP1 Potency=0.0164(uM) D4 PubChem colchicine TDP1 Potency=0.0473(uM) D4 PubChem colchicine TDP1 Potency=0.0668(uM) D4 PubChem colchicine TDP1 Potency=0.1884(uM) D4 PubChem colchicine TDP1 Potency=0.2661(uM) D4 PubChem colchicine VDR None=None(uM) D4 PubChem