Drug Gene Type Source clozapine ABCB1 Text_Mining(decreases(activity)) CTD clozapine ABCB11 Text_Mining(decreases(activity)) CTD clozapine ABCG1 Text_Mining(increases(expression)) CTD clozapine ABCG2 Text_Mining(decreases(reaction)) CTD clozapine ABCG2 Text_Mining(increases(transport)) CTD clozapine ABLIM2 Text_Mining(increases(expression)) CTD clozapine ACAT2 Text_Mining(increases(expression)) CTD clozapine ADIPOQ Text_Mining(decreases(expression)) CTD clozapine AGT Text_Mining(decreases(reaction)) CTD clozapine AGT Text_Mining(increases(reaction)) CTD clozapine AGT Text_Mining(increases(secretion)) CTD clozapine AKT1 Text_Mining(increases(expression)) CTD clozapine AKT1 Text_Mining(increases(phosphorylation)) CTD clozapine ALPP Text_Mining(decreases(reaction)) CTD clozapine ALPP Text_Mining(increases(expression)) CTD clozapine AP1S1 Text_Mining(decreases(expression)) CTD clozapine ASAH1 Text_Mining(increases(expression)) CTD clozapine ASNS Text_Mining(increases(expression)) CTD clozapine BAX Text_Mining(increases(expression)) CTD clozapine BAX Text_Mining(decreases(reaction)) CTD clozapine BIK Text_Mining(increases(expression)) CTD clozapine BIK Text_Mining(decreases(reaction)) CTD clozapine C10ORF10 Text_Mining(increases(expression)) CTD clozapine CASP3 Text_Mining(increases(activity)) CTD clozapine CASP3 Text_Mining(increases(reaction)) CTD clozapine CASP7 Text_Mining(increases(activity)) CTD clozapine CASP7 Text_Mining(increases(reaction)) CTD clozapine CCL1 Text_Mining(decreases(expression)) CTD clozapine CHRM1 Text_Mining(affects(binding)) CTD clozapine CLOCK Text_Mining(affects(response to substance)) CTD clozapine COMT Text_Mining(increases(response to substance)) CTD clozapine COMT Text_Mining(affects(response to substance)) CTD clozapine CRH Text_Mining(decreases(expression)) CTD clozapine CRP Text_Mining(increases(expression)) CTD clozapine CSF3 Text_Mining(decreases(reaction)) CTD clozapine CSF3 Text_Mining(increases(expression)) CTD clozapine CXCL1 Text_Mining(decreases(expression)) CTD clozapine CXCL5 Text_Mining(decreases(expression)) CTD clozapine CYP1A2 Text_Mining(decreases(activity)) CTD clozapine CYP1A2 Text_Mining(increases(abundance)) CTD clozapine CYP1A2 Text_Mining(decreases(reaction)) CTD clozapine CYP1A2 Text_Mining(increases(activity)) CTD clozapine CYP1A2 Text_Mining(affects(metabolic processing)) CTD clozapine CYP1A2 Text_Mining(affects(response to substance)) CTD clozapine CYP1A2 Text_Mining(decreases(metabolic processing)) CTD clozapine CYP1A2 Text_Mining(decreases(response to substance)) CTD clozapine CYP1A2 Text_Mining(increases(metabolic processing)) CTD clozapine CYP1A2 Text_Mining(affects(cotreatment)) CTD clozapine CYP1A2 Text_Mining(affects(reaction)) CTD clozapine CYP1A2 Text_Mining(increases(reaction)) CTD clozapine CYP2C19 Text_Mining(affects(cotreatment)) CTD clozapine CYP2C19 Text_Mining(affects(response to substance)) CTD clozapine CYP2C9 Text_Mining(decreases(activity)) CTD clozapine CYP2C9 Text_Mining(increases(response to substance)) CTD clozapine CYP2C9 Text_Mining(affects(cotreatment)) CTD clozapine CYP2C9 Text_Mining(affects(response to substance)) CTD clozapine CYP2D6 Text_Mining(affects(cotreatment)) CTD clozapine CYP2D6 Text_Mining(affects(response to substance)) CTD clozapine CYP2D6 Text_Mining(affects(metabolic processing)) CTD clozapine CYP3A4 Text_Mining(increases(expression)) CTD clozapine CYP3A4 Text_Mining(increases(reaction)) CTD clozapine CYP3A4 Text_Mining(affects(cotreatment)) CTD clozapine CYP3A4 Text_Mining(affects(response to substance)) CTD clozapine CYP3A4 Text_Mining(affects(metabolic processing)) CTD clozapine CYP3A4 Text_Mining(decreases(reaction)) CTD clozapine DHCR7 Text_Mining(increases(expression)) CTD clozapine DISC1 Text_Mining(decreases(response to substance)) CTD clozapine DISC1 Text_Mining(affects(response to substance)) CTD clozapine DRD1 Text_Mining(affects(binding)) CTD clozapine DRD1 Text_Mining(affects(response to substance)) CTD clozapine DRD2 Text_Mining(affects(binding)) CTD clozapine DRD2 Text_Mining(affects(cotreatment)) CTD clozapine DRD2 Text_Mining(increases(secretion)) CTD clozapine DRD2 Text_Mining(affects(response to substance)) CTD clozapine DRD2 Text_Mining(increases(response to substance)) CTD clozapine DRD3 Text_Mining(decreases(response to substance)) CTD clozapine DRD3 Text_Mining(affects(response to substance)) CTD clozapine DRD4 Text_Mining(affects(binding)) CTD clozapine DRD4 Text_Mining(affects(response to substance)) CTD clozapine DTNBP1 Text_Mining(increases(response to substance)) CTD clozapine DTNBP1 Text_Mining(affects(response to substance)) CTD clozapine FABP1 Text_Mining(increases(expression)) CTD clozapine FASLG Text_Mining(affects(cotreatment)) CTD clozapine FASLG Text_Mining(increases(expression)) CTD clozapine FASN Text_Mining(increases(expression)) CTD clozapine FCGR3B Text_Mining(affects(cotreatment)) CTD clozapine FCGR3B Text_Mining(decreases(expression)) CTD clozapine FDPS Text_Mining(increases(expression)) CTD clozapine FGFBP2 Text_Mining(increases(expression)) CTD clozapine FNDC4 Text_Mining(increases(expression)) CTD clozapine GAD1 Text_Mining(increases(expression)) CTD clozapine GDPD3 Text_Mining(increases(expression)) CTD clozapine GNB3 Text_Mining(decreases(response to substance)) CTD clozapine GNB3 Text_Mining(increases(response to substance)) CTD clozapine GNB3 Text_Mining(affects(response to substance)) CTD clozapine GSK3B Text_Mining(increases(phosphorylation)) CTD clozapine GSTA1 Text_Mining(decreases(activity)) CTD clozapine GSTA1 Text_Mining(increases(glutathionylation)) CTD clozapine GSTM1 Text_Mining(decreases(activity)) CTD clozapine GSTM1 Text_Mining(increases(glutathionylation)) CTD clozapine GSTP1 Text_Mining(affects(binding)) CTD clozapine GSTP1 Text_Mining(decreases(activity)) CTD clozapine GSTP1 Text_Mining(affects(metabolic processing)) CTD clozapine GSTP1 Text_Mining(increases(glutathionylation)) CTD clozapine HMGCR Text_Mining(increases(activity)) CTD clozapine HMGCR Text_Mining(increases(abundance)) CTD clozapine HMGCR Text_Mining(increases(expression)) CTD clozapine HMGCS1 Text_Mining(increases(expression)) CTD clozapine HMOX1 Text_Mining(increases(expression)) CTD clozapine HPN Text_Mining(increases(expression)) CTD clozapine HRH1 Text_Mining(affects(binding)) CTD clozapine HTR1A Text_Mining(affects(activity)) CTD clozapine HTR1A Text_Mining(affects(binding)) CTD clozapine HTR2A Text_Mining(affects(binding)) CTD clozapine HTR2A Text_Mining(decreases(activity)) CTD clozapine HTR2A Text_Mining(decreases(reaction)) CTD clozapine HTR2A Text_Mining(increases(response to substance)) CTD clozapine HTR2A Text_Mining(affects(response to substance)) CTD clozapine HTR2C Text_Mining(affects(binding)) CTD clozapine HTR2C Text_Mining(affects(response to substance)) CTD clozapine HTR3A Text_Mining(affects(binding)) CTD clozapine HTR3A Text_Mining(decreases(activity)) CTD clozapine HTR3A Text_Mining(affects(response to substance)) CTD clozapine HTR6 Text_Mining(affects(binding)) CTD clozapine HTR7 Text_Mining(affects(binding)) CTD clozapine HTR7 Text_Mining(decreases(activity)) CTD clozapine HTR7 Text_Mining(decreases(reaction)) CTD clozapine HTR7 Text_Mining(increases(abundance)) CTD clozapine IFNG Text_Mining(affects(expression)) CTD clozapine IFNG Text_Mining(decreases(expression)) CTD clozapine IGF1 Text_Mining(decreases(expression)) CTD clozapine IL2RA Text_Mining(increases(secretion)) CTD clozapine IL5 Text_Mining(affects(expression)) CTD clozapine INHBE Text_Mining(increases(expression)) CTD clozapine INS Text_Mining(affects(secretion)) CTD clozapine INS Text_Mining(increases(expression)) CTD clozapine KCNH2 Text_Mining(decreases(reaction)) CTD clozapine KCNH2 Text_Mining(increases(transport)) CTD clozapine KMT2A Text_Mining(increases(expression)) CTD clozapine LDLR Text_Mining(increases(expression)) CTD clozapine LEAP2 Text_Mining(increases(expression)) CTD clozapine LEP Text_Mining(affects(response to substance)) CTD clozapine LSS Text_Mining(increases(expression)) CTD clozapine MBP Text_Mining(increases(expression)) CTD clozapine MC1R Text_Mining(increases(expression)) CTD clozapine MMP10 Text_Mining(decreases(expression)) CTD clozapine MMP7 Text_Mining(decreases(expression)) CTD clozapine MTHFR Text_Mining(affects(response to substance)) CTD clozapine NFE2L2 Text_Mining(affects(response to substance)) CTD clozapine NQO2 Text_Mining(affects(response to substance)) CTD clozapine NR0B2 Text_Mining(increases(expression)) CTD clozapine NR1I2 Text_Mining(increases(expression)) CTD clozapine NR1I2 Text_Mining(increases(reaction)) CTD clozapine NR1I2 Text_Mining(decreases(reaction)) CTD clozapine NRG1 Text_Mining(increases(expression)) CTD clozapine NUPR1 Text_Mining(increases(expression)) CTD clozapine OVGP1 Text_Mining(increases(expression)) CTD clozapine OXT Text_Mining(affects(response to substance)) CTD clozapine PRL Text_Mining(affects(cotreatment)) CTD clozapine PRL Text_Mining(increases(secretion)) CTD clozapine PRL Text_Mining(increases(expression)) CTD clozapine PROC Text_Mining(increases(expression)) CTD clozapine SC5D Text_Mining(increases(expression)) CTD clozapine SCD Text_Mining(increases(expression)) CTD clozapine SERPINA3 Text_Mining(increases(expression)) CTD clozapine SLC22A2 Text_Mining(decreases(reaction)) CTD clozapine SLC22A2 Text_Mining(increases(uptake)) CTD clozapine SLC2A3 Text_Mining(decreases(expression)) CTD clozapine SLC6A3 Text_Mining(affects(response to substance)) CTD clozapine SLC6A4 Text_Mining(decreases(response to substance)) CTD clozapine SLC6A4 Text_Mining(decreases(uptake)) CTD clozapine SLC6A4 Text_Mining(affects(response to substance)) CTD clozapine SNAP25 Text_Mining(affects(response to substance)) CTD clozapine SPP1 Text_Mining(decreases(expression)) CTD clozapine SREBF1 Text_Mining(increases(expression)) CTD clozapine SREBF2 Text_Mining(decreases(activity)) CTD clozapine SREBF2 Text_Mining(decreases(reaction)) CTD clozapine SREBF2 Text_Mining(increases(activity)) CTD clozapine SREBF2 Text_Mining(increases(cleavage)) CTD clozapine SREBF2 Text_Mining(increases(expression)) CTD clozapine TAGLN Text_Mining(decreases(expression)) CTD clozapine TNF Text_Mining(affects(response to substance)) CTD clozapine TNFSF15 Text_Mining(decreases(expression)) CTD clozapine TP53 Text_Mining(increases(expression)) CTD clozapine TP53 Text_Mining(decreases(reaction)) CTD clozapine UGT1A1 Text_Mining(increases(expression)) CTD clozapine UGT1A4 Text_Mining(increases(glucuronidation)) CTD clozapine WIPI1 Text_Mining(increases(expression)) CTD clozapine AR AR Potency (uM)=28.7255(uM) D4 PubChem clozapine CBX1 Potency=79.4328(uM) D4 PubChem clozapine CBX1 Potency=79432.8(nM) D4 ChEMBL clozapine CHRM1 None=None(uM) D4 PubChem clozapine CHRM4 None=None(uM) D4 PubChem clozapine CHRM5 None=None(uM) D4 PubChem clozapine CYP1A2 None=None(uM) D4 PubChem clozapine CYP1A2 Inhibition=None(Unspecified) D4 ChEMBL clozapine CYP2C19 Inhibition=None(Unspecified) D4 ChEMBL clozapine CYP2C9 Inhibition=None(Unspecified) D4 ChEMBL clozapine CYP3A4 Inhibition=None(Unspecified) D4 ChEMBL clozapine DRD1 Potency=0.631(uM) D4 PubChem clozapine DRD1 None=None(uM) D4 PubChem clozapine DRD1 Potency=631.0(nM) D4 ChEMBL clozapine DRD2 None=None(uM) D4 PubChem clozapine DRD2 Activity=None(Unspecified) D4 ChEMBL clozapine DRD3 None=None(uM) D4 PubChem clozapine HTR1A None=None(uM) D4 PubChem clozapine HTR1B None=None(uM) D4 PubChem clozapine HTR1D None=None(uM) D4 PubChem clozapine HTR1E None=None(uM) D4 PubChem clozapine HTR1F None=None(uM) D4 PubChem clozapine HTR2A None=None(uM) D4 PubChem clozapine HTR2B None=None(uM) D4 PubChem clozapine HTR2C None=None(uM) D4 PubChem clozapine HTR5A None=None(uM) D4 PubChem clozapine HTR6 None=None(uM) D4 PubChem clozapine HTR7 None=None(uM) D4 PubChem clozapine HTR7 Inhibition=None(Unspecified) D4 ChEMBL clozapine MAPT None=None(uM) D4 PubChem clozapine NR3C1 None=None(uM) D4 PubChem clozapine POLI Potency=79.4328(uM) D4 PubChem clozapine PPARG None=None(uM) D4 PubChem clozapine RGS4 None=None(uM) D4 PubChem clozapine TDP1 Potency=16.3601(uM) D4 PubChem clozapine TDP1 Potency=18.8375(uM) D4 PubChem clozapine TDP1 Potency=23.715(uM) D4 PubChem