Drug Gene Type Source chlorpromazine ABCB1 Text_Mining(increases(expression)) CTD chlorpromazine ABCB1 Text_Mining(decreases(activity)) CTD chlorpromazine ABCC3 Text_Mining(increases(expression)) CTD chlorpromazine ABCG2 Text_Mining(decreases(reaction)) CTD chlorpromazine ABCG2 Text_Mining(increases(transport)) CTD chlorpromazine ACHE Text_Mining(decreases(activity)) CTD chlorpromazine ACHE Text_Mining(increases(reaction)) CTD chlorpromazine AFP Text_Mining(decreases(expression)) CTD chlorpromazine ALPP Text_Mining(decreases(reaction)) CTD chlorpromazine ALPP Text_Mining(increases(expression)) CTD chlorpromazine AP1S1 Text_Mining(decreases(expression)) CTD chlorpromazine AREG Text_Mining(decreases(expression)) CTD chlorpromazine ASAH1 Text_Mining(increases(expression)) CTD chlorpromazine ASNS Text_Mining(increases(expression)) CTD chlorpromazine AVP Text_Mining(increases(expression)) CTD chlorpromazine BAG4 Text_Mining(decreases(expression)) CTD chlorpromazine BDNF Text_Mining(affects(response to substance)) CTD chlorpromazine BHLHE40 Text_Mining(increases(expression)) CTD chlorpromazine BIRC5 Text_Mining(decreases(expression)) CTD chlorpromazine BTG2 Text_Mining(increases(expression)) CTD chlorpromazine BTG3 Text_Mining(increases(expression)) CTD chlorpromazine C10ORF10 Text_Mining(increases(expression)) CTD chlorpromazine CCNB2 Text_Mining(decreases(expression)) CTD chlorpromazine CCND3 Text_Mining(decreases(expression)) CTD chlorpromazine CCNF Text_Mining(decreases(expression)) CTD chlorpromazine CD86 Text_Mining(increases(expression)) CTD chlorpromazine CDK5 Text_Mining(decreases(expression)) CTD chlorpromazine CDK7 Text_Mining(increases(expression)) CTD chlorpromazine CDKN2C Text_Mining(decreases(expression)) CTD chlorpromazine CHTF18 Text_Mining(decreases(expression)) CTD chlorpromazine CKS2 Text_Mining(decreases(expression)) CTD chlorpromazine CRH Text_Mining(decreases(expression)) CTD chlorpromazine CYP1A1 Text_Mining(decreases(reaction)) CTD chlorpromazine CYP1A1 Text_Mining(increases(activity)) CTD chlorpromazine CYP1A2 Text_Mining(decreases(reaction)) CTD chlorpromazine CYP1A2 Text_Mining(increases(activity)) CTD chlorpromazine CYP1A2 Text_Mining(affects(cotreatment)) CTD chlorpromazine CYP1A2 Text_Mining(affects(response to substance)) CTD chlorpromazine CYP1A2 Text_Mining(decreases(methylation)) CTD chlorpromazine CYP1A2 Text_Mining(increases(metabolic processing)) CTD chlorpromazine CYP1A2 Text_Mining(increases(oxidation)) CTD chlorpromazine CYP2A6 Text_Mining(decreases(activity)) CTD chlorpromazine CYP2B6 Text_Mining(increases(activity)) CTD chlorpromazine CYP2B6 Text_Mining(increases(expression)) CTD chlorpromazine CYP2C19 Text_Mining(decreases(activity)) CTD chlorpromazine CYP2C19 Text_Mining(affects(cotreatment)) CTD chlorpromazine CYP2C19 Text_Mining(affects(response to substance)) CTD chlorpromazine CYP2C19 Text_Mining(affects(methylation)) CTD chlorpromazine CYP2C9 Text_Mining(decreases(activity)) CTD chlorpromazine CYP2C9 Text_Mining(affects(cotreatment)) CTD chlorpromazine CYP2C9 Text_Mining(affects(response to substance)) CTD chlorpromazine CYP2D6 Text_Mining(affects(cotreatment)) CTD chlorpromazine CYP2D6 Text_Mining(affects(response to substance)) CTD chlorpromazine CYP2D6 Text_Mining(increases(activity)) CTD chlorpromazine CYP2D6 Text_Mining(increases(metabolic processing)) CTD chlorpromazine CYP2E1 Text_Mining(decreases(activity)) CTD chlorpromazine CYP3A4 Text_Mining(decreases(activity)) CTD chlorpromazine CYP3A4 Text_Mining(increases(activity)) CTD chlorpromazine CYP3A4 Text_Mining(increases(expression)) CTD chlorpromazine CYP3A4 Text_Mining(affects(cotreatment)) CTD chlorpromazine CYP3A4 Text_Mining(affects(response to substance)) CTD chlorpromazine CYP3A4 Text_Mining(affects(methylation)) CTD chlorpromazine CYP3A4 Text_Mining(affects(oxidation)) CTD chlorpromazine DAO Text_Mining(decreases(activity)) CTD chlorpromazine DRD1 Text_Mining(decreases(activity)) CTD chlorpromazine DRD2 Text_Mining(decreases(activity)) CTD chlorpromazine DRD2 Text_Mining(decreases(response to substance)) CTD chlorpromazine DUSP1 Text_Mining(increases(expression)) CTD chlorpromazine DUSP9 Text_Mining(decreases(expression)) CTD chlorpromazine E2F1 Text_Mining(decreases(expression)) CTD chlorpromazine F2 Text_Mining(decreases(expression)) CTD chlorpromazine FABP1 Text_Mining(increases(expression)) CTD chlorpromazine FAS Text_Mining(increases(expression)) CTD chlorpromazine FGFR1 Text_Mining(decreases(expression)) CTD chlorpromazine FKBP5 Text_Mining(decreases(expression)) CTD chlorpromazine FKBP5 Text_Mining(decreases(reaction)) CTD chlorpromazine FNDC4 Text_Mining(increases(expression)) CTD chlorpromazine FOSL1 Text_Mining(increases(expression)) CTD chlorpromazine G6PD Text_Mining(decreases(expression)) CTD chlorpromazine GDPD3 Text_Mining(increases(expression)) CTD chlorpromazine HMGCR Text_Mining(increases(expression)) CTD chlorpromazine HMGCS1 Text_Mining(increases(expression)) CTD chlorpromazine HMOX1 Text_Mining(increases(expression)) CTD chlorpromazine HPN Text_Mining(increases(expression)) CTD chlorpromazine IGFBP1 Text_Mining(increases(expression)) CTD chlorpromazine IKBKG Text_Mining(increases(expression)) CTD chlorpromazine IL1A Text_Mining(affects(cotreatment)) CTD chlorpromazine IL1A Text_Mining(increases(response to substance)) CTD chlorpromazine IL2 Text_Mining(decreases(reaction)) CTD chlorpromazine IL2 Text_Mining(increases(phosphorylation)) CTD chlorpromazine IL6 Text_Mining(affects(cotreatment)) CTD chlorpromazine IL6 Text_Mining(increases(response to substance)) CTD chlorpromazine INHBE Text_Mining(increases(expression)) CTD chlorpromazine KCNH2 Text_Mining(decreases(reaction)) CTD chlorpromazine KCNH2 Text_Mining(increases(transport)) CTD chlorpromazine KCNH2 Text_Mining(decreases(activity)) CTD chlorpromazine LDLR Text_Mining(increases(expression)) CTD chlorpromazine LSS Text_Mining(increases(expression)) CTD chlorpromazine MAPK1 Text_Mining(decreases(reaction)) CTD chlorpromazine MAPK1 Text_Mining(increases(phosphorylation)) CTD chlorpromazine MAPK14 Text_Mining(decreases(expression)) CTD chlorpromazine MAPK3 Text_Mining(decreases(expression)) CTD chlorpromazine MAPK3 Text_Mining(decreases(reaction)) CTD chlorpromazine MAPK3 Text_Mining(increases(phosphorylation)) CTD chlorpromazine MCM3 Text_Mining(decreases(expression)) CTD chlorpromazine MCM5 Text_Mining(decreases(expression)) CTD chlorpromazine MKI67 Text_Mining(decreases(expression)) CTD chlorpromazine MSH2 Text_Mining(decreases(expression)) CTD chlorpromazine MYBL2 Text_Mining(decreases(expression)) CTD chlorpromazine NR0B2 Text_Mining(increases(expression)) CTD chlorpromazine NR1I2 Text_Mining(increases(expression)) CTD chlorpromazine NR1I2 Text_Mining(increases(activity)) CTD chlorpromazine NR1I3 Text_Mining(increases(activity)) CTD chlorpromazine NR1I3 Text_Mining(increases(expression)) CTD chlorpromazine NUPR1 Text_Mining(increases(expression)) CTD chlorpromazine ORC1 Text_Mining(decreases(expression)) CTD chlorpromazine ORM1 Text_Mining(affects(binding)) CTD chlorpromazine ORM1 Text_Mining(decreases(reaction)) CTD chlorpromazine ORM2 Text_Mining(affects(binding)) CTD chlorpromazine ORM2 Text_Mining(decreases(reaction)) CTD chlorpromazine PDIA2 Text_Mining(increases(expression)) CTD chlorpromazine PHYH Text_Mining(increases(expression)) CTD chlorpromazine PIM1 Text_Mining(increases(expression)) CTD chlorpromazine POLA1 Text_Mining(decreases(expression)) CTD chlorpromazine POLD4 Text_Mining(increases(expression)) CTD chlorpromazine PRL Text_Mining(increases(expression)) CTD chlorpromazine SC5D Text_Mining(increases(expression)) CTD chlorpromazine SERPINA3 Text_Mining(increases(expression)) CTD chlorpromazine SLC22A2 Text_Mining(decreases(reaction)) CTD chlorpromazine SLC22A2 Text_Mining(increases(uptake)) CTD chlorpromazine SLC2A3 Text_Mining(decreases(expression)) CTD chlorpromazine SLC31A1 Text_Mining(affects(localization)) CTD chlorpromazine SLC31A1 Text_Mining(decreases(reaction)) CTD chlorpromazine SREBF2 Text_Mining(increases(activity)) CTD chlorpromazine SREBF2 Text_Mining(increases(cleavage)) CTD chlorpromazine STS Text_Mining(decreases(reaction)) CTD chlorpromazine STS Text_Mining(increases(activity)) CTD chlorpromazine TAGLN Text_Mining(decreases(expression)) CTD chlorpromazine TF Text_Mining(affects(localization)) CTD chlorpromazine TFDP1 Text_Mining(decreases(expression)) CTD chlorpromazine TNF Text_Mining(decreases(expression)) CTD chlorpromazine TNF Text_Mining(decreases(activity)) CTD chlorpromazine TNF Text_Mining(affects(cotreatment)) CTD chlorpromazine TNF Text_Mining(increases(response to substance)) CTD chlorpromazine TNFRSF14 Text_Mining(increases(expression)) CTD chlorpromazine UNG Text_Mining(decreases(expression)) CTD chlorpromazine VEGFA Text_Mining(increases(expression)) CTD chlorpromazine WIPI1 Text_Mining(increases(expression)) CTD chlorpromazine XRCC4 Text_Mining(decreases(expression)) CTD chlorpromazine CYP1A2 None=None(uM) D4 PubChem chlorpromazine CYP1A2 AC50=3981.07(nM) D4 ChEMBL chlorpromazine CYP1A2 AC50=1000.0(nM) D4 ChEMBL chlorpromazine CYP2C9 Inhibition=None(Unspecified) D4 ChEMBL chlorpromazine CYP2D6 Potency=0.1585(uM) D4 PubChem chlorpromazine CYP2D6 Potency=0.3981(uM) D4 PubChem chlorpromazine CYP2D6 None=None(uM) D4 PubChem chlorpromazine CYP2D6 AC50=398.11(nM) D4 ChEMBL chlorpromazine CYP2D6 Potency=158.5(nM) D4 ChEMBL chlorpromazine CYP2D6 Potency=398.1(nM) D4 ChEMBL chlorpromazine CYP2D6 AC50=158.49(nM) D4 ChEMBL chlorpromazine CYP3A4 Inhibition=None(Unspecified) D4 ChEMBL chlorpromazine HTR1A None=None(uM) D4 PubChem chlorpromazine HTR2A None=None(uM) D4 PubChem chlorpromazine HTR2C None=None(uM) D4 PubChem chlorpromazine HTR6 None=None(uM) D4 PubChem chlorpromazine HTR7 None=None(uM) D4 PubChem chlorpromazine IDH1 Potency=15.8489(uM) D4 PubChem chlorpromazine MAPT None=None(uM) D4 PubChem chlorpromazine NR1H4 Potency-Replicate_1=26.6011(uM) D4 PubChem chlorpromazine TDP1 Potency=10.0(uM) D4 PubChem chlorpromazine TDP1 Potency=11.2202(uM) D4 PubChem chlorpromazine TDP1 Potency=23.715(uM) D4 PubChem chlorpromazine THPO Potency=12.5893(uM) D4 PubChem chlorpromazine THPO Potency=12589.3(nM) D4 ChEMBL chlorpromazine TP53 Potency=10.0(uM) D4 PubChem chlorpromazine TP53 Potency=10000.0(nM) D4 ChEMBL