Drug Gene Type Source chlorambucil ABCB1 Text_Mining(increases(expression)) CTD chlorambucil ABCC1 Text_Mining(affects(export)) CTD chlorambucil ABCC1 Text_Mining(decreases(response to substance)) CTD chlorambucil ABCC1 Text_Mining(increases(response to substance)) CTD chlorambucil ABCC1 Text_Mining(increases(reaction)) CTD chlorambucil ABCC2 Text_Mining(affects(export)) CTD chlorambucil ABCC2 Text_Mining(decreases(response to substance)) CTD chlorambucil ABCC2 Text_Mining(increases(reaction)) CTD chlorambucil BAX Text_Mining(increases(expression)) CTD chlorambucil BBC3 Text_Mining(increases(expression)) CTD chlorambucil BCL2 Text_Mining(decreases(expression)) CTD chlorambucil BCL2 Text_Mining(decreases(reaction)) CTD chlorambucil BIRC2 Text_Mining(decreases(response to substance)) CTD chlorambucil BIRC5 Text_Mining(affects(expression)) CTD chlorambucil CASP3 Text_Mining(increases(activity)) CTD chlorambucil CASP8 Text_Mining(increases(activity)) CTD chlorambucil CDA Text_Mining(decreases(response to substance)) CTD chlorambucil CDK1 Text_Mining(decreases(activity)) CTD chlorambucil CDK1 Text_Mining(increases(phosphorylation)) CTD chlorambucil CDKN1A Text_Mining(increases(expression)) CTD chlorambucil DHFR Text_Mining(decreases(response to substance)) CTD chlorambucil FANCC Text_Mining(increases(response to substance)) CTD chlorambucil FANCG Text_Mining(increases(response to substance)) CTD chlorambucil FAS Text_Mining(increases(expression)) CTD chlorambucil GCLC Text_Mining(affects(cotreatment)) CTD chlorambucil GCLC Text_Mining(decreases(response to substance)) CTD chlorambucil GCLM Text_Mining(affects(cotreatment)) CTD chlorambucil GCLM Text_Mining(decreases(response to substance)) CTD chlorambucil GSTA1 Text_Mining(decreases(response to substance)) CTD chlorambucil GSTA1 Text_Mining(increases(reaction)) CTD chlorambucil GSTA1 Text_Mining(decreases(activity)) CTD chlorambucil GSTA1 Text_Mining(affects(cotreatment)) CTD chlorambucil GSTA1 Text_Mining(affects(metabolic processing)) CTD chlorambucil GSTM1 Text_Mining(decreases(response to substance)) CTD chlorambucil GSTP1 Text_Mining(affects(binding)) CTD chlorambucil GSTP1 Text_Mining(affects(response to substance)) CTD chlorambucil GSTP1 Text_Mining(decreases(response to substance)) CTD chlorambucil GSTP1 Text_Mining(increases(reaction)) CTD chlorambucil GSTP1 Text_Mining(increases(metabolic processing)) CTD chlorambucil H2AFX Text_Mining(increases(phosphorylation)) CTD chlorambucil HIST1H4C Text_Mining(decreases(expression)) CTD chlorambucil IL4 Text_Mining(decreases(expression)) CTD chlorambucil IL4 Text_Mining(decreases(reaction)) CTD chlorambucil IL4 Text_Mining(affects(cotreatment)) CTD chlorambucil IL4 Text_Mining(increases(expression)) CTD chlorambucil KEAP1 Text_Mining(decreases(reaction)) CTD chlorambucil KEAP1 Text_Mining(decreases(response to substance)) CTD chlorambucil KEAP1 Text_Mining(increases(activity)) CTD chlorambucil MDM2 Text_Mining(increases(expression)) CTD chlorambucil MYC Text_Mining(affects(expression)) CTD chlorambucil MYC Text_Mining(increases(expression)) CTD chlorambucil MYC Text_Mining(affects(cotreatment)) CTD chlorambucil MYC Text_Mining(decreases(reaction)) CTD chlorambucil NFE2L2 Text_Mining(decreases(reaction)) CTD chlorambucil NFE2L2 Text_Mining(decreases(response to substance)) CTD chlorambucil NFE2L2 Text_Mining(increases(activity)) CTD chlorambucil NFE2L2 Text_Mining(increases(response to substance)) CTD chlorambucil RAD51 Text_Mining(increases(expression)) CTD chlorambucil SFN Text_Mining(increases(expression)) CTD chlorambucil TNFRSF10A Text_Mining(affects(expression)) CTD chlorambucil TNFRSF10B Text_Mining(affects(expression)) CTD chlorambucil TNFRSF10B Text_Mining(increases(expression)) CTD chlorambucil TP53 Text_Mining(increases(expression)) CTD chlorambucil TP53 Text_Mining(affects(cotreatment)) CTD chlorambucil TP53 Text_Mining(decreases(reaction)) CTD chlorambucil BAZ2B Potency=56.2341(uM) D4 PubChem chlorambucil BAZ2B Potency=56234.1(nM) D4 ChEMBL chlorambucil GFER AC50_uM=0.005(uM) D4 PubChem chlorambucil GFER None=None(uM) D4 PubChem chlorambucil GFER AC50=5.0(nM) D4 ChEMBL chlorambucil NFE2L2 Ratio Potency (uM)=66.2759(uM) D4 PubChem chlorambucil NFKB1 Potency=8.9125(uM) D4 PubChem chlorambucil NFKB1 Potency=8912.5(nM) D4 ChEMBL chlorambucil STK33 None=None(uM) D4 PubChem chlorambucil TDP1 Potency=0.4611(uM) D4 PubChem chlorambucil TDP1 Potency=0.5623(uM) D4 PubChem chlorambucil TDP1 Potency=0.6513(uM) D4 PubChem chlorambucil TDP1 Potency=0.8913(uM) D4 PubChem chlorambucil TDP1 Potency=14.581(uM) D4 PubChem