Drug Gene Type Source busulfan ANP32B Text_Mining(affects(cotreatment)) CTD busulfan ANP32B Text_Mining(increases(cleavage)) CTD busulfan APEX1 Text_Mining(increases(response to substance)) CTD busulfan AR Text_Mining(decreases(reaction)) CTD busulfan AR Text_Mining(increases(activity)) CTD busulfan ARHGDIA Text_Mining(affects(reaction)) CTD busulfan ARHGDIA Text_Mining(increases(activity)) CTD busulfan ARHGDIA Text_Mining(affects(response to substance)) CTD busulfan ATM Text_Mining(affects(cotreatment)) CTD busulfan ATM Text_Mining(increases(phosphorylation)) CTD busulfan CASP3 Text_Mining(affects(reaction)) CTD busulfan CASP3 Text_Mining(increases(activity)) CTD busulfan CASP3 Text_Mining(affects(cotreatment)) CTD busulfan CASP3 Text_Mining(increases(cleavage)) CTD busulfan CASP8 Text_Mining(increases(activity)) CTD busulfan CASP8 Text_Mining(affects(cotreatment)) CTD busulfan CASP8 Text_Mining(decreases(reaction)) CTD busulfan CASP9 Text_Mining(affects(cotreatment)) CTD busulfan CASP9 Text_Mining(increases(cleavage)) CTD busulfan CASP9 Text_Mining(decreases(reaction)) CTD busulfan CASP9 Text_Mining(increases(activity)) CTD busulfan CDC25B Text_Mining(affects(cotreatment)) CTD busulfan CDC25B Text_Mining(increases(phosphorylation)) CTD busulfan CDKN1A Text_Mining(increases(expression)) CTD busulfan CDKN1A Text_Mining(affects(cotreatment)) CTD busulfan CHEK1 Text_Mining(affects(cotreatment)) CTD busulfan CHEK1 Text_Mining(increases(phosphorylation)) CTD busulfan CHEK2 Text_Mining(affects(cotreatment)) CTD busulfan CHEK2 Text_Mining(increases(phosphorylation)) CTD busulfan GSTA1 Text_Mining(affects(abundance)) CTD busulfan GSTA1 Text_Mining(affects(metabolic processing)) CTD busulfan GSTA1 Text_Mining(affects(response to substance)) CTD busulfan GSTA1 Text_Mining(affects(cotreatment)) CTD busulfan GSTA1 Text_Mining(decreases(response to substance)) CTD busulfan GSTM1 Text_Mining(affects(abundance)) CTD busulfan GSTM1 Text_Mining(affects(response to substance)) CTD busulfan GSTM1 Text_Mining(affects(cotreatment)) CTD busulfan GSTM1 Text_Mining(affects(metabolic processing)) CTD busulfan GSTP1 Text_Mining(affects(abundance)) CTD busulfan GSTP1 Text_Mining(affects(metabolic processing)) CTD busulfan GSTT1 Text_Mining(affects(cotreatment)) CTD busulfan GSTT1 Text_Mining(affects(metabolic processing)) CTD busulfan H2AFX Text_Mining(increases(phosphorylation)) CTD busulfan H2AFX Text_Mining(affects(cotreatment)) CTD busulfan H2AFX Text_Mining(increases(expression)) CTD busulfan INHBA Text_Mining(decreases(reaction)) CTD busulfan INHBA Text_Mining(increases(expression)) CTD busulfan MAPK1 Text_Mining(increases(activity)) CTD busulfan MAPK3 Text_Mining(increases(activity)) CTD busulfan MGST2 Text_Mining(decreases(response to substance)) CTD busulfan MYC Text_Mining(affects(cotreatment)) CTD busulfan MYC Text_Mining(decreases(expression)) CTD busulfan NPM1 Text_Mining(affects(cotreatment)) CTD busulfan NPM1 Text_Mining(increases(response to substance)) CTD busulfan PARP1 Text_Mining(increases(cleavage)) CTD busulfan PARP1 Text_Mining(affects(cotreatment)) CTD busulfan PARP1 Text_Mining(decreases(reaction)) CTD busulfan PTGS2 Text_Mining(increases(expression)) CTD busulfan SERPINC1 Text_Mining(affects(expression)) CTD busulfan SERPINE1 Text_Mining(decreases(reaction)) CTD busulfan SERPINE1 Text_Mining(increases(expression)) CTD busulfan SMC1A Text_Mining(affects(cotreatment)) CTD busulfan SMC1A Text_Mining(increases(phosphorylation)) CTD busulfan SMC3 Text_Mining(affects(cotreatment)) CTD busulfan SMC3 Text_Mining(increases(phosphorylation)) CTD busulfan TF Text_Mining(decreases(reaction)) CTD busulfan TF Text_Mining(increases(expression)) CTD busulfan TFPI Text_Mining(decreases(expression)) CTD busulfan TGFB1 Text_Mining(increases(expression)) CTD busulfan THBS1 Text_Mining(increases(expression)) CTD busulfan TNF Text_Mining(increases(expression)) CTD busulfan TP53 Text_Mining(affects(activity)) CTD busulfan TP53 Text_Mining(affects(phosphorylation)) CTD busulfan XIAP Text_Mining(affects(cotreatment)) CTD busulfan XIAP Text_Mining(decreases(expression)) CTD busulfan CYP1A2 Inhibition=None(Unspecified) D4 ChEMBL busulfan CYP2C19 Inhibition=None(Unspecified) D4 ChEMBL busulfan CYP2C9 Inhibition=None(Unspecified) D4 ChEMBL busulfan CYP2D6 Inhibition=None(Unspecified) D4 ChEMBL busulfan CYP3A4 Inhibition=None(Unspecified) D4 ChEMBL busulfan ESR1 Potency-Replicate_1=11.8832(uM) D4 PubChem