Drug Gene Type Source buspirone CYP2D6 Text_Mining(increases(oxidation)) CTD buspirone CYP3A4 Text_Mining(increases(metabolic processing)) CTD buspirone CYP3A4 Text_Mining(increases(oxidation)) CTD buspirone CYP3A4 Text_Mining(decreases(reaction)) CTD buspirone CYP3A5 Text_Mining(increases(oxidation)) CTD buspirone HTR1A Text_Mining(affects(activity)) CTD buspirone HTR1A Text_Mining(affects(binding)) CTD buspirone POMC Text_Mining(increases(expression)) CTD buspirone POMC Text_Mining(decreases(reaction)) CTD buspirone PRL Text_Mining(increases(expression)) CTD buspirone PRL Text_Mining(increases(secretion)) CTD buspirone PRL Text_Mining(decreases(reaction)) CTD buspirone SLC22A2 Text_Mining(decreases(reaction)) CTD buspirone SLC22A2 Text_Mining(increases(uptake)) CTD buspirone ALDH1A1 Potency=4.4668(uM) D4 PubChem buspirone ALDH1A1 Potency=4466.8(nM) D4 ChEMBL buspirone EHMT2 Potency=12.5893(uM) D4 PubChem buspirone EHMT2 Potency=12589.3(nM) D4 ChEMBL buspirone ESR1 Potency-Replicate_1=30.6379(uM) D4 PubChem buspirone ESR1 ER Potency (uM)=38.5708(uM) D4 PubChem buspirone HTR1A None=None(uM) D4 PubChem buspirone NFE2L2 Potency-Replicate_1=27.306(uM) D4 PubChem buspirone NFE2L2 Ratio Potency (uM)=30.6379(uM) D4 PubChem