Drug Gene Type Source benzbromarone ABCB11 Text_Mining(decreases(reaction)) CTD benzbromarone ABCB11 Text_Mining(increases(transport)) CTD benzbromarone ABCB11 Text_Mining(decreases(activity)) CTD benzbromarone ABCC1 Text_Mining(affects(activity)) CTD benzbromarone ABCC1 Text_Mining(decreases(reaction)) CTD benzbromarone ABCC1 Text_Mining(increases(export)) CTD benzbromarone ABCC1 Text_Mining(increases(secretion)) CTD benzbromarone ABCC2 Text_Mining(decreases(activity)) CTD benzbromarone ABCC6 Text_Mining(affects(transport)) CTD benzbromarone ABCC6 Text_Mining(decreases(reaction)) CTD benzbromarone ABCC6 Text_Mining(decreases(activity)) CTD benzbromarone ADIPOQ Text_Mining(increases(expression)) CTD benzbromarone AKR1C1 Text_Mining(decreases(activity)) CTD benzbromarone AKR1C2 Text_Mining(decreases(activity)) CTD benzbromarone AKR1C3 Text_Mining(decreases(activity)) CTD benzbromarone AKR1C4 Text_Mining(decreases(activity)) CTD benzbromarone CRP Text_Mining(decreases(reaction)) CTD benzbromarone CRP Text_Mining(increases(expression)) CTD benzbromarone CRP Text_Mining(decreases(expression)) CTD benzbromarone CYP2C19 Text_Mining(affects(binding)) CTD benzbromarone CYP2C19 Text_Mining(decreases(activity)) CTD benzbromarone CYP2C9 Text_Mining(affects(binding)) CTD benzbromarone CYP2C9 Text_Mining(decreases(activity)) CTD benzbromarone CYP2C9 Text_Mining(affects(metabolic processing)) CTD benzbromarone CYP2C9 Text_Mining(decreases(reaction)) CTD benzbromarone CYP2C9 Text_Mining(affects(hydroxylation)) CTD benzbromarone CYP2C9 Text_Mining(increases(reaction)) CTD benzbromarone EYA2 Text_Mining(decreases(activity)) CTD benzbromarone EYA3 Text_Mining(decreases(activity)) CTD benzbromarone IL1A Text_Mining(affects(cotreatment)) CTD benzbromarone IL1A Text_Mining(increases(response to substance)) CTD benzbromarone IL1B Text_Mining(decreases(reaction)) CTD benzbromarone IL1B Text_Mining(increases(expression)) CTD benzbromarone IL6 Text_Mining(affects(cotreatment)) CTD benzbromarone IL6 Text_Mining(increases(response to substance)) CTD benzbromarone IYD Text_Mining(decreases(activity)) CTD benzbromarone LPL Text_Mining(increases(expression)) CTD benzbromarone SLC22A12 Text_Mining(affects(activity)) CTD benzbromarone SLC22A12 Text_Mining(decreases(reaction)) CTD benzbromarone SLC22A12 Text_Mining(increases(uptake)) CTD benzbromarone SLC22A12 Text_Mining(decreases(activity)) CTD benzbromarone SLC22A12 Text_Mining(affects(response to substance)) CTD benzbromarone SLC22A6 Text_Mining(affects(transport)) CTD benzbromarone SLC22A6 Text_Mining(decreases(reaction)) CTD benzbromarone SLC2A9 Text_Mining(decreases(reaction)) CTD benzbromarone SLC2A9 Text_Mining(increases(transport)) CTD benzbromarone TNF Text_Mining(increases(expression)) CTD benzbromarone TNF Text_Mining(affects(cotreatment)) CTD benzbromarone TNF Text_Mining(increases(response to substance)) CTD benzbromarone ABCB1 None=None(uM) D4 PubChem benzbromarone ABCC2 Inhibition=None(Unspecified) D4 ChEMBL benzbromarone ABHD5 None=None(uM) D4 PubChem benzbromarone ATG4B None=None(uM) D4 PubChem benzbromarone CRHBP None=None(uM) D4 PubChem benzbromarone CRHR2 None=None(uM) D4 PubChem benzbromarone CYP1A2 None=None(uM) D4 PubChem benzbromarone CYP1A2 AC50=12589.2(nM) D4 ChEMBL benzbromarone CYP2C9 Potency=0.0079(uM) D4 PubChem benzbromarone CYP2C9 Potency=0.0398(uM) D4 PubChem benzbromarone CYP2C9 None=None(uM) D4 PubChem benzbromarone CYP2C9 AC50=7.94(nM) D4 ChEMBL benzbromarone CYP2C9 Potency=39.8(nM) D4 ChEMBL benzbromarone CYP2C9 Potency=7.9(nM) D4 ChEMBL benzbromarone ESR1 Potency-Replicate_1=10.6822(uM) D4 PubChem benzbromarone ESR1 Ratio Potency (uM)=14.5209(uM) D4 PubChem benzbromarone GFER None=None(uM) D4 PubChem benzbromarone GMNN Potency=1.8356(uM) D4 PubChem benzbromarone GMNN Potency=2.9855(uM) D4 PubChem benzbromarone GMNN Potency=7.3078(uM) D4 PubChem benzbromarone HCRTR1 None=None(uM) D4 PubChem benzbromarone HIF1A Potency=3.9811(uM) D4 PubChem benzbromarone HIF1A Potency=3981.1(nM) D4 ChEMBL benzbromarone HPGD Potency=17.7828(uM) D4 PubChem benzbromarone HPGD Potency=17782.8(nM) D4 ChEMBL benzbromarone HSD17B10 Potency=12589.3(nM) D4 ChEMBL benzbromarone HSPB1 Ratio Potency (uM)=None(uM) D4 PubChem benzbromarone KCNE1 None=None(uM) D4 PubChem benzbromarone KCNJ1 None=None(uM) D4 PubChem benzbromarone KCNQ1 None=None(uM) D4 PubChem benzbromarone MCL1 None=None(uM) D4 PubChem benzbromarone NCOR2 IC50=4.811(uM) D4 PubChem benzbromarone NCOR2 None=None(uM) D4 PubChem benzbromarone NCOR2 IC50=4811.0(nM) D4 ChEMBL benzbromarone NOD1 EC50=None(uM) D4 PubChem benzbromarone NOD2 EC50=None(uM) D4 PubChem benzbromarone NR2E3 None=None(uM) D4 PubChem benzbromarone NR3C1 Potency-Replicate_1=15.089(uM) D4 PubChem benzbromarone PLA2G1B None=None(uM) D4 PubChem benzbromarone PLIN1 None=None(uM) D4 PubChem benzbromarone PLIN5 None=None(uM) D4 PubChem benzbromarone PLK1 Potency=8.4368(uM) D4 PubChem benzbromarone POLB Potency=50.1187(uM) D4 PubChem benzbromarone POLB Potency=50118.7(nM) D4 ChEMBL benzbromarone PPARG Ratio Potency (uM)=2.68325(uM) D4 PubChem benzbromarone PPARG Potency-Replicate_1=3.0107(uM) D4 PubChem benzbromarone PPARG IC50=4.811(uM) D4 PubChem benzbromarone PPARG None=None(uM) D4 PubChem benzbromarone PPARG IC50=4811.0(nM) D4 ChEMBL benzbromarone PTGER2 None=None(uM) D4 PubChem benzbromarone S1PR1 None=None(uM) D4 PubChem benzbromarone SLC12A5 None=None(uM) D4 PubChem benzbromarone TNF None=None(uM) D4 PubChem benzbromarone TNNC1 None=None(uM) D4 PubChem benzbromarone TNNI3 None=None(uM) D4 PubChem benzbromarone TNNT2 None=None(uM) D4 PubChem benzbromarone TSHR None=None(uM) D4 PubChem benzbromarone USP1 Potency=31.6228(uM) D4 PubChem benzbromarone VDR Potency=28.1838(uM) D4 PubChem benzbromarone VDR Potency=50.1187(uM) D4 PubChem