Drug Gene Type Source amitriptyline AP1S1 Text_Mining(decreases(expression)) CTD amitriptyline ASAH1 Text_Mining(increases(expression)) CTD amitriptyline ASNS Text_Mining(increases(expression)) CTD amitriptyline C10ORF10 Text_Mining(increases(expression)) CTD amitriptyline CAT Text_Mining(decreases(expression)) CTD amitriptyline CYP1A2 Text_Mining(increases(metabolic processing)) CTD amitriptyline CYP1A2 Text_Mining(affects(cotreatment)) CTD amitriptyline CYP1A2 Text_Mining(affects(response to substance)) CTD amitriptyline CYP2C19 Text_Mining(affects(cotreatment)) CTD amitriptyline CYP2C19 Text_Mining(affects(response to substance)) CTD amitriptyline CYP2C9 Text_Mining(affects(cotreatment)) CTD amitriptyline CYP2C9 Text_Mining(affects(response to substance)) CTD amitriptyline CYP2D6 Text_Mining(decreases(activity)) CTD amitriptyline CYP2D6 Text_Mining(increases(metabolic processing)) CTD amitriptyline CYP2D6 Text_Mining(affects(cotreatment)) CTD amitriptyline CYP2D6 Text_Mining(affects(response to substance)) CTD amitriptyline CYP3A4 Text_Mining(increases(metabolic processing)) CTD amitriptyline CYP3A4 Text_Mining(affects(cotreatment)) CTD amitriptyline CYP3A4 Text_Mining(affects(response to substance)) CTD amitriptyline CYP3A5 Text_Mining(increases(metabolic processing)) CTD amitriptyline FABP1 Text_Mining(increases(expression)) CTD amitriptyline FNDC4 Text_Mining(increases(expression)) CTD amitriptyline GDPD3 Text_Mining(increases(expression)) CTD amitriptyline GSTP1 Text_Mining(decreases(activity)) CTD amitriptyline HMGCS1 Text_Mining(increases(expression)) CTD amitriptyline HPN Text_Mining(increases(expression)) CTD amitriptyline HTR2C Text_Mining(affects(binding)) CTD amitriptyline INHBE Text_Mining(increases(expression)) CTD amitriptyline KCNH2 Text_Mining(decreases(reaction)) CTD amitriptyline KCNH2 Text_Mining(increases(transport)) CTD amitriptyline LSS Text_Mining(increases(expression)) CTD amitriptyline NR0B2 Text_Mining(increases(expression)) CTD amitriptyline NUPR1 Text_Mining(increases(expression)) CTD amitriptyline PHYH Text_Mining(increases(expression)) CTD amitriptyline SCD Text_Mining(increases(expression)) CTD amitriptyline SERPINA3 Text_Mining(increases(expression)) CTD amitriptyline SLC22A2 Text_Mining(decreases(reaction)) CTD amitriptyline SLC22A2 Text_Mining(increases(uptake)) CTD amitriptyline SLC22A6 Text_Mining(decreases(reaction)) CTD amitriptyline SLC22A6 Text_Mining(increases(uptake)) CTD amitriptyline SLC2A3 Text_Mining(decreases(expression)) CTD amitriptyline SREBF1 Text_Mining(increases(activity)) CTD amitriptyline SREBF1 Text_Mining(increases(cleavage)) CTD amitriptyline SREBF2 Text_Mining(increases(activity)) CTD amitriptyline SREBF2 Text_Mining(increases(cleavage)) CTD amitriptyline TAGLN Text_Mining(decreases(expression)) CTD amitriptyline TRH Text_Mining(decreases(expression)) CTD amitriptyline TRH Text_Mining(decreases(reaction)) CTD amitriptyline TSHB Text_Mining(decreases(expression)) CTD amitriptyline TSHB Text_Mining(decreases(reaction)) CTD amitriptyline WIPI1 Text_Mining(increases(expression)) CTD amitriptyline CYP1A2 None=None(uM) D4 PubChem amitriptyline CYP1A2 Inhibition=None(Unspecified) D4 ChEMBL amitriptyline CYP2C9 Inhibition=None(Unspecified) D4 ChEMBL amitriptyline CYP2D6 Potency=7.9433(uM) D4 PubChem amitriptyline CYP2D6 None=None(uM) D4 PubChem amitriptyline CYP2D6 AC50=7943.28(nM) D4 ChEMBL amitriptyline CYP2D6 Inhibition=None(Unspecified) D4 ChEMBL amitriptyline CYP2D6 Potency=7943.3(nM) D4 ChEMBL amitriptyline CYP3A4 Inhibition=None(Unspecified) D4 ChEMBL amitriptyline DRD1 Potency=1.122(uM) D4 PubChem amitriptyline DRD1 Potency=1122.0(nM) D4 ChEMBL amitriptyline HTR6 None=None(uM) D4 PubChem