Drug Gene Type Source NSC94017 ABCC4 Text_Mining(increases(transport)) CTD NSC94017 ADCYAP1 Text_Mining(affects(binding)) CTD NSC94017 ADCYAP1 Text_Mining(increases(abundance)) CTD NSC94017 ADIPOQ Text_Mining(increases(abundance)) CTD NSC94017 ADRB1 Text_Mining(affects(binding)) CTD NSC94017 ADRB1 Text_Mining(decreases(abundance)) CTD NSC94017 ADRB1 Text_Mining(decreases(activity)) CTD NSC94017 ADRB1 Text_Mining(affects(cotreatment)) CTD NSC94017 ADRB1 Text_Mining(increases(abundance)) CTD NSC94017 ADRB1 Text_Mining(affects(abundance)) CTD NSC94017 ADRB1 Text_Mining(affects(reaction)) CTD NSC94017 ADRB1 Text_Mining(decreases(reaction)) CTD NSC94017 ADRB1 Text_Mining(increases(reaction)) CTD NSC94017 ADRB1 Text_Mining(increases(activity)) CTD NSC94017 ADRB2 Text_Mining(affects(binding)) CTD NSC94017 ADRB2 Text_Mining(increases(abundance)) CTD NSC94017 ADRB2 Text_Mining(affects(abundance)) CTD NSC94017 ADRB2 Text_Mining(increases(chemical synthesis)) CTD NSC94017 ADRB2 Text_Mining(increases(activity)) CTD NSC94017 ADRB2 Text_Mining(decreases(abundance)) CTD NSC94017 ADRB2 Text_Mining(decreases(activity)) CTD NSC94017 ADRB2 Text_Mining(decreases(reaction)) CTD NSC94017 ADRB2 Text_Mining(affects(cotreatment)) CTD NSC94017 ADRB2 Text_Mining(increases(reaction)) CTD NSC94017 ADRB3 Text_Mining(affects(binding)) CTD NSC94017 ADRB3 Text_Mining(decreases(reaction)) CTD NSC94017 ADRB3 Text_Mining(increases(abundance)) CTD NSC94017 ADRB3 Text_Mining(increases(activity)) CTD NSC94017 ADRB3 Text_Mining(affects(abundance)) CTD NSC94017 ADRB3 Text_Mining(decreases(abundance)) CTD NSC94017 ADRB3 Text_Mining(decreases(activity)) CTD NSC94017 ALPP Text_Mining(increases(abundance)) CTD NSC94017 ALPP Text_Mining(increases(expression)) CTD NSC94017 AVP Text_Mining(affects(binding)) CTD NSC94017 AVP Text_Mining(increases(abundance)) CTD NSC94017 AVP Text_Mining(increases(activity)) CTD NSC94017 AVPR2 Text_Mining(affects(binding)) CTD NSC94017 AVPR2 Text_Mining(increases(abundance)) CTD NSC94017 AVPR2 Text_Mining(increases(activity)) CTD NSC94017 BRAF Text_Mining(increases(activity)) CTD NSC94017 CALCA Text_Mining(increases(abundance)) CTD NSC94017 CALCA Text_Mining(decreases(reaction)) CTD NSC94017 CARM1 Text_Mining(increases(activity)) CTD NSC94017 CARM1 Text_Mining(increases(reaction)) CTD NSC94017 CARM1 Text_Mining(increases(expression)) CTD NSC94017 CARM1 Text_Mining(affects(binding)) CTD NSC94017 CARM1 Text_Mining(increases(phosphorylation)) CTD NSC94017 CCND1 Text_Mining(increases(abundance)) CTD NSC94017 CCND1 Text_Mining(increases(expression)) CTD NSC94017 CDKN1B Text_Mining(increases(abundance)) CTD NSC94017 CDKN1B Text_Mining(increases(expression)) CTD NSC94017 CFTR Text_Mining(increases(reaction)) CTD NSC94017 CFTR Text_Mining(increases(transport)) CTD NSC94017 CFTR Text_Mining(increases(activity)) CTD NSC94017 CGA Text_Mining(affects(secretion)) CTD NSC94017 CGA Text_Mining(increases(secretion)) CTD NSC94017 CGA Text_Mining(affects(cotreatment)) CTD NSC94017 CGA Text_Mining(increases(abundance)) CTD NSC94017 CGA Text_Mining(increases(reaction)) CTD NSC94017 CGB Text_Mining(decreases(reaction)) CTD NSC94017 CGB Text_Mining(increases(secretion)) CTD NSC94017 CGB Text_Mining(increases(abundance)) CTD NSC94017 CGB Text_Mining(increases(reaction)) CTD NSC94017 CGB Text_Mining(increases(activity)) CTD NSC94017 CGB Text_Mining(affects(cotreatment)) CTD NSC94017 CNR1 Text_Mining(affects(binding)) CTD NSC94017 CNR1 Text_Mining(increases(abundance)) CTD NSC94017 CNR1 Text_Mining(increases(activity)) CTD NSC94017 CNR1 Text_Mining(decreases(reaction)) CTD NSC94017 CNR2 Text_Mining(affects(binding)) CTD NSC94017 CNR2 Text_Mining(decreases(reaction)) CTD NSC94017 CNR2 Text_Mining(increases(abundance)) CTD NSC94017 CNR2 Text_Mining(increases(activity)) CTD NSC94017 CREBBP Text_Mining(increases(activity)) CTD NSC94017 CREBBP Text_Mining(increases(reaction)) CTD NSC94017 CRH Text_Mining(affects(binding)) CTD NSC94017 CRH Text_Mining(increases(abundance)) CTD NSC94017 CRH Text_Mining(increases(activity)) CTD NSC94017 CRH Text_Mining(increases(reaction)) CTD NSC94017 CRHR1 Text_Mining(affects(binding)) CTD NSC94017 CRHR1 Text_Mining(increases(abundance)) CTD NSC94017 CRHR1 Text_Mining(increases(activity)) CTD NSC94017 CRHR1 Text_Mining(increases(reaction)) CTD NSC94017 CSF3 Text_Mining(increases(expression)) CTD NSC94017 CXCL8 Text_Mining(increases(abundance)) CTD NSC94017 CXCL8 Text_Mining(increases(expression)) CTD NSC94017 CYP11B1 Text_Mining(increases(expression)) CTD NSC94017 CYP11B1 Text_Mining(decreases(reaction)) CTD NSC94017 CYP17A1 Text_Mining(affects(cotreatment)) CTD NSC94017 CYP17A1 Text_Mining(decreases(activity)) CTD NSC94017 CYP17A1 Text_Mining(increases(activity)) CTD NSC94017 DISC1 Text_Mining(affects(binding)) CTD NSC94017 DISC1 Text_Mining(decreases(reaction)) CTD NSC94017 DKK1 Text_Mining(affects(response to substance)) CTD NSC94017 DRD1 Text_Mining(increases(chemical synthesis)) CTD NSC94017 DRD1 Text_Mining(increases(reaction)) CTD NSC94017 DRD2 Text_Mining(affects(binding)) CTD NSC94017 DRD2 Text_Mining(decreases(reaction)) CTD NSC94017 DRD2 Text_Mining(increases(abundance)) CTD NSC94017 DRD2 Text_Mining(increases(activity)) CTD NSC94017 ESR1 Text_Mining(increases(activity)) CTD NSC94017 ESR1 Text_Mining(increases(reaction)) CTD NSC94017 ESR1 Text_Mining(affects(binding)) CTD NSC94017 ESR1 Text_Mining(increases(phosphorylation)) CTD NSC94017 ESR1 Text_Mining(increases(abundance)) CTD NSC94017 ESR1 Text_Mining(decreases(reaction)) CTD NSC94017 ESR2 Text_Mining(increases(abundance)) CTD NSC94017 ESR2 Text_Mining(increases(activity)) CTD NSC94017 ESR2 Text_Mining(increases(reaction)) CTD NSC94017 F2RL1 Text_Mining(increases(reaction)) CTD NSC94017 F2RL1 Text_Mining(increases(transport)) CTD NSC94017 FOS Text_Mining(affects(cotreatment)) CTD NSC94017 FOS Text_Mining(increases(expression)) CTD NSC94017 FSHB Text_Mining(affects(cotreatment)) CTD NSC94017 FSHB Text_Mining(increases(chemical synthesis)) CTD NSC94017 GDNF Text_Mining(affects(cotreatment)) CTD NSC94017 GDNF Text_Mining(decreases(reaction)) CTD NSC94017 GDNF Text_Mining(increases(response to substance)) CTD NSC94017 GDNF Text_Mining(decreases(response to substance)) CTD NSC94017 GHRH Text_Mining(affects(binding)) CTD NSC94017 GHRH Text_Mining(increases(abundance)) CTD NSC94017 GHRH Text_Mining(increases(activity)) CTD NSC94017 GNAS Text_Mining(increases(abundance)) CTD NSC94017 GNAS Text_Mining(increases(activity)) CTD NSC94017 GNAS Text_Mining(increases(reaction)) CTD NSC94017 GPBAR1 Text_Mining(affects(binding)) CTD NSC94017 GPBAR1 Text_Mining(increases(abundance)) CTD NSC94017 GPBAR1 Text_Mining(increases(activity)) CTD NSC94017 HCAR2 Text_Mining(decreases(reaction)) CTD NSC94017 HCAR2 Text_Mining(increases(abundance)) CTD NSC94017 HCAR2 Text_Mining(increases(activity)) CTD NSC94017 HCAR2 Text_Mining(decreases(abundance)) CTD NSC94017 HCAR2 Text_Mining(affects(binding)) CTD NSC94017 HCAR3 Text_Mining(decreases(abundance)) CTD NSC94017 HRH1 Text_Mining(decreases(abundance)) CTD NSC94017 HRH1 Text_Mining(decreases(reaction)) CTD NSC94017 HRH1 Text_Mining(increases(reaction)) CTD NSC94017 HRH2 Text_Mining(affects(binding)) CTD NSC94017 HRH2 Text_Mining(decreases(abundance)) CTD NSC94017 HRH2 Text_Mining(decreases(activity)) CTD NSC94017 HRH2 Text_Mining(decreases(reaction)) CTD NSC94017 HRH2 Text_Mining(increases(abundance)) CTD NSC94017 HRH2 Text_Mining(increases(activity)) CTD NSC94017 HRH2 Text_Mining(decreases(expression)) CTD NSC94017 HRH2 Text_Mining(increases(reaction)) CTD NSC94017 HSD3B2 Text_Mining(increases(expression)) CTD NSC94017 HTR1A Text_Mining(decreases(reaction)) CTD NSC94017 HTR1A Text_Mining(increases(abundance)) CTD NSC94017 HTR1A Text_Mining(affects(binding)) CTD NSC94017 HTR1A Text_Mining(increases(activity)) CTD NSC94017 HTR1B Text_Mining(affects(reaction)) CTD NSC94017 HTR1B Text_Mining(decreases(reaction)) CTD NSC94017 HTR1B Text_Mining(increases(abundance)) CTD NSC94017 HTR7 Text_Mining(affects(binding)) CTD NSC94017 HTR7 Text_Mining(decreases(activity)) CTD NSC94017 HTR7 Text_Mining(decreases(reaction)) CTD NSC94017 HTR7 Text_Mining(increases(abundance)) CTD NSC94017 HTR7 Text_Mining(increases(activity)) CTD NSC94017 HTR7 Text_Mining(decreases(abundance)) CTD NSC94017 IL12A Text_Mining(decreases(expression)) CTD NSC94017 IL12A Text_Mining(increases(activity)) CTD NSC94017 IL12A Text_Mining(increases(reaction)) CTD NSC94017 IL12B Text_Mining(decreases(expression)) CTD NSC94017 IL12B Text_Mining(increases(activity)) CTD NSC94017 IL12B Text_Mining(increases(reaction)) CTD NSC94017 IL1B Text_Mining(increases(abundance)) CTD NSC94017 IL1B Text_Mining(increases(reaction)) CTD NSC94017 IL1B Text_Mining(decreases(reaction)) CTD NSC94017 INHBA Text_Mining(increases(secretion)) CTD NSC94017 JUN Text_Mining(affects(cotreatment)) CTD NSC94017 JUN Text_Mining(increases(expression)) CTD NSC94017 LEP Text_Mining(increases(abundance)) CTD NSC94017 LHB Text_Mining(affects(secretion)) CTD NSC94017 LHB Text_Mining(increases(secretion)) CTD NSC94017 LHB Text_Mining(affects(cotreatment)) CTD NSC94017 LHB Text_Mining(increases(abundance)) CTD NSC94017 LHCGR Text_Mining(increases(abundance)) CTD NSC94017 LHCGR Text_Mining(increases(activity)) CTD NSC94017 LHCGR Text_Mining(increases(reaction)) CTD NSC94017 LHCGR Text_Mining(decreases(reaction)) CTD NSC94017 LIPE Text_Mining(increases(activity)) CTD NSC94017 MC2R Text_Mining(affects(cotreatment)) CTD NSC94017 MC2R Text_Mining(decreases(expression)) CTD NSC94017 NDUFB11 Text_Mining(increases(phosphorylation)) CTD NSC94017 NDUFB11 Text_Mining(decreases(reaction)) CTD NSC94017 OPRM1 Text_Mining(affects(binding)) CTD NSC94017 OPRM1 Text_Mining(decreases(activity)) CTD NSC94017 OPRM1 Text_Mining(increases(expression)) CTD NSC94017 OPRM1 Text_Mining(affects(cotreatment)) CTD NSC94017 PDE10A Text_Mining(decreases(reaction)) CTD NSC94017 PDE10A Text_Mining(increases(hydrolysis)) CTD NSC94017 PDE11A Text_Mining(increases(hydrolysis)) CTD NSC94017 PDE4B Text_Mining(decreases(activity)) CTD NSC94017 PDE4B Text_Mining(increases(abundance)) CTD NSC94017 PDE4B Text_Mining(affects(binding)) CTD NSC94017 PDE4B Text_Mining(decreases(reaction)) CTD NSC94017 PDE7A Text_Mining(decreases(reaction)) CTD NSC94017 PDE7A Text_Mining(increases(hydrolysis)) CTD NSC94017 PDE7B Text_Mining(decreases(reaction)) CTD NSC94017 PDE7B Text_Mining(increases(hydrolysis)) CTD NSC94017 PDE8A Text_Mining(decreases(reaction)) CTD NSC94017 PDE8A Text_Mining(increases(metabolic processing)) CTD NSC94017 PDE8B Text_Mining(decreases(reaction)) CTD NSC94017 PDE8B Text_Mining(increases(metabolic processing)) CTD NSC94017 PDE8B Text_Mining(increases(hydrolysis)) CTD NSC94017 PDE9A Text_Mining(increases(hydrolysis)) CTD NSC94017 PRL Text_Mining(increases(secretion)) CTD NSC94017 PROK1 Text_Mining(affects(response to substance)) CTD NSC94017 PTGIR Text_Mining(increases(abundance)) CTD NSC94017 PTGIR Text_Mining(increases(activity)) CTD NSC94017 PTGIR Text_Mining(increases(reaction)) CTD NSC94017 PTHLH Text_Mining(increases(abundance)) CTD NSC94017 RAP1B Text_Mining(affects(binding)) CTD NSC94017 RAP1B Text_Mining(increases(abundance)) CTD NSC94017 SLC22A8 Text_Mining(affects(transport)) CTD NSC94017 SLC2A5 Text_Mining(affects(expression)) CTD NSC94017 SLC2A5 Text_Mining(increases(abundance)) CTD NSC94017 SLC2A5 Text_Mining(increases(stability)) CTD NSC94017 SOD2 Text_Mining(affects(reaction)) CTD NSC94017 SOD2 Text_Mining(increases(abundance)) CTD NSC94017 SOD2 Text_Mining(increases(expression)) CTD NSC94017 TFF1 Text_Mining(increases(expression)) CTD NSC94017 TFF1 Text_Mining(increases(reaction)) CTD NSC94017 TFF1 Text_Mining(affects(binding)) CTD NSC94017 TNF Text_Mining(decreases(reaction)) CTD NSC94017 TNF Text_Mining(increases(expression)) CTD NSC94017 TNF Text_Mining(decreases(expression)) CTD NSC94017 TSHB Text_Mining(decreases(reaction)) CTD NSC94017 TSHB Text_Mining(increases(abundance)) CTD NSC94017 TSHB Text_Mining(increases(activity)) CTD NSC94017 TSHR Text_Mining(decreases(reaction)) CTD NSC94017 TSHR Text_Mining(increases(abundance)) CTD NSC94017 TSHR Text_Mining(increases(activity)) CTD NSC94017 VIP Text_Mining(affects(binding)) CTD NSC94017 VIP Text_Mining(increases(abundance)) CTD NSC94017 VIPR2 Text_Mining(affects(binding)) CTD NSC94017 VIPR2 Text_Mining(increases(abundance)) CTD NSC94017 WNT5A Text_Mining(affects(reaction)) CTD NSC94017 WNT5A Text_Mining(increases(abundance)) CTD NSC94017 WNT5A Text_Mining(increases(expression)) CTD NSC94017 DRD1 Potency=0.3663(uM) D4 PubChem NSC94017 EHMT2 Potency=2.8184(uM) D4 PubChem NSC94017 EHMT2 Potency=2818.4(nM) D4 ChEMBL NSC94017 PTGER2 None=None(uM) D4 PubChem