Drug Gene Type Source Calcimycin ALOX5 Text_Mining(decreases(reaction)) CTD Calcimycin ALOX5 Text_Mining(increases(activity)) CTD Calcimycin ALOX5 Text_Mining(increases(localization)) CTD Calcimycin ALOX5 Text_Mining(decreases(activity)) CTD Calcimycin ALOX5 Text_Mining(increases(abundance)) CTD Calcimycin CASP1 Text_Mining(affects(cotreatment)) CTD Calcimycin CASP1 Text_Mining(increases(activity)) CTD Calcimycin CASP1 Text_Mining(decreases(reaction)) CTD Calcimycin CASP1 Text_Mining(increases(cleavage)) CTD Calcimycin CASP3 Text_Mining(decreases(reaction)) CTD Calcimycin CASP3 Text_Mining(increases(activity)) CTD Calcimycin CASP7 Text_Mining(increases(activity)) CTD Calcimycin CCL11 Text_Mining(affects(abundance)) CTD Calcimycin CCL11 Text_Mining(affects(chemical synthesis)) CTD Calcimycin CCL11 Text_Mining(increases(reaction)) CTD Calcimycin CCL5 Text_Mining(affects(abundance)) CTD Calcimycin CCL5 Text_Mining(affects(chemical synthesis)) CTD Calcimycin CCL5 Text_Mining(increases(reaction)) CTD Calcimycin CD40 Text_Mining(affects(cotreatment)) CTD Calcimycin CD40 Text_Mining(decreases(reaction)) CTD Calcimycin CD40 Text_Mining(increases(expression)) CTD Calcimycin CD69 Text_Mining(affects(cotreatment)) CTD Calcimycin CD69 Text_Mining(decreases(reaction)) CTD Calcimycin CD69 Text_Mining(increases(expression)) CTD Calcimycin CDH1 Text_Mining(increases(cleavage)) CTD Calcimycin CDH1 Text_Mining(increases(reaction)) CTD Calcimycin CXCL8 Text_Mining(affects(cotreatment)) CTD Calcimycin CXCL8 Text_Mining(decreases(reaction)) CTD Calcimycin CXCL8 Text_Mining(increases(expression)) CTD Calcimycin CXCL8 Text_Mining(increases(reaction)) CTD Calcimycin CXCL8 Text_Mining(increases(secretion)) CTD Calcimycin DDIT3 Text_Mining(increases(activity)) CTD Calcimycin DDIT3 Text_Mining(increases(expression)) CTD Calcimycin DDIT3 Text_Mining(increases(reaction)) CTD Calcimycin DDIT3 Text_Mining(decreases(reaction)) CTD Calcimycin EIF2A Text_Mining(increases(phosphorylation)) CTD Calcimycin EIF2A Text_Mining(decreases(reaction)) CTD Calcimycin ERN1 Text_Mining(increases(expression)) CTD Calcimycin GPX4 Text_Mining(decreases(expression)) CTD Calcimycin HDC Text_Mining(increases(expression)) CTD Calcimycin HMOX1 Text_Mining(decreases(reaction)) CTD Calcimycin HMOX1 Text_Mining(increases(expression)) CTD Calcimycin HSPA5 Text_Mining(increases(expression)) CTD Calcimycin HSPA5 Text_Mining(decreases(reaction)) CTD Calcimycin IFNG Text_Mining(affects(cotreatment)) CTD Calcimycin IFNG Text_Mining(increases(expression)) CTD Calcimycin IFNG Text_Mining(decreases(reaction)) CTD Calcimycin IL13 Text_Mining(affects(cotreatment)) CTD Calcimycin IL13 Text_Mining(increases(expression)) CTD Calcimycin IL13 Text_Mining(decreases(reaction)) CTD Calcimycin IL18R1 Text_Mining(affects(cotreatment)) CTD Calcimycin IL18R1 Text_Mining(increases(expression)) CTD Calcimycin IL1B Text_Mining(affects(cotreatment)) CTD Calcimycin IL1B Text_Mining(decreases(reaction)) CTD Calcimycin IL1B Text_Mining(increases(expression)) CTD Calcimycin IL1B Text_Mining(increases(secretion)) CTD Calcimycin IL1B Text_Mining(increases(activity)) CTD Calcimycin IL1B Text_Mining(increases(reaction)) CTD Calcimycin IL2 Text_Mining(affects(cotreatment)) CTD Calcimycin IL2 Text_Mining(decreases(reaction)) CTD Calcimycin IL2 Text_Mining(increases(expression)) CTD Calcimycin IL2 Text_Mining(increases(secretion)) CTD Calcimycin IL4 Text_Mining(affects(cotreatment)) CTD Calcimycin IL4 Text_Mining(increases(expression)) CTD Calcimycin IL4 Text_Mining(decreases(reaction)) CTD Calcimycin IL4 Text_Mining(affects(response to substance)) CTD Calcimycin IL4 Text_Mining(increases(metabolic processing)) CTD Calcimycin IL4 Text_Mining(increases(reaction)) CTD Calcimycin IL5 Text_Mining(affects(cotreatment)) CTD Calcimycin IL5 Text_Mining(increases(expression)) CTD Calcimycin IL5 Text_Mining(decreases(reaction)) CTD Calcimycin IL5 Text_Mining(affects(abundance)) CTD Calcimycin IL5 Text_Mining(affects(chemical synthesis)) CTD Calcimycin IL5 Text_Mining(increases(reaction)) CTD Calcimycin IL6 Text_Mining(affects(cotreatment)) CTD Calcimycin IL6 Text_Mining(decreases(reaction)) CTD Calcimycin IL6 Text_Mining(increases(expression)) CTD Calcimycin IL6 Text_Mining(increases(reaction)) CTD Calcimycin IL6 Text_Mining(increases(secretion)) CTD Calcimycin ITGAM Text_Mining(increases(expression)) CTD Calcimycin ITGAM Text_Mining(decreases(reaction)) CTD Calcimycin ITGB2 Text_Mining(increases(expression)) CTD Calcimycin MAPK1 Text_Mining(affects(cotreatment)) CTD Calcimycin MAPK1 Text_Mining(decreases(reaction)) CTD Calcimycin MAPK1 Text_Mining(increases(phosphorylation)) CTD Calcimycin MAPK1 Text_Mining(increases(activity)) CTD Calcimycin MAPK3 Text_Mining(affects(cotreatment)) CTD Calcimycin MAPK3 Text_Mining(decreases(reaction)) CTD Calcimycin MAPK3 Text_Mining(increases(phosphorylation)) CTD Calcimycin MAPK3 Text_Mining(increases(activity)) CTD Calcimycin MPO Text_Mining(increases(secretion)) CTD Calcimycin MPO Text_Mining(decreases(reaction)) CTD Calcimycin MSR1 Text_Mining(affects(cotreatment)) CTD Calcimycin MSR1 Text_Mining(increases(expression)) CTD Calcimycin MSR1 Text_Mining(increases(reaction)) CTD Calcimycin NFATC1 Text_Mining(affects(cotreatment)) CTD Calcimycin NFATC1 Text_Mining(increases(expression)) CTD Calcimycin NFATC1 Text_Mining(increases(reaction)) CTD Calcimycin NFATC1 Text_Mining(affects(localization)) CTD Calcimycin NFATC1 Text_Mining(decreases(expression)) CTD Calcimycin NFATC1 Text_Mining(decreases(reaction)) CTD Calcimycin NFATC2 Text_Mining(increases(activity)) CTD Calcimycin NFATC2 Text_Mining(decreases(reaction)) CTD Calcimycin NFATC2 Text_Mining(affects(cotreatment)) CTD Calcimycin NFATC2 Text_Mining(increases(expression)) CTD Calcimycin NFATC2 Text_Mining(increases(reaction)) CTD Calcimycin NFATC2 Text_Mining(decreases(phosphorylation)) CTD Calcimycin NFATC3 Text_Mining(affects(cotreatment)) CTD Calcimycin NFATC3 Text_Mining(increases(expression)) CTD Calcimycin NFATC3 Text_Mining(increases(reaction)) CTD Calcimycin NFATC4 Text_Mining(affects(cotreatment)) CTD Calcimycin NFATC4 Text_Mining(increases(expression)) CTD Calcimycin NFATC4 Text_Mining(increases(reaction)) CTD Calcimycin NFKBIA Text_Mining(affects(cotreatment)) CTD Calcimycin NFKBIA Text_Mining(increases(degradation)) CTD Calcimycin NFKBIA Text_Mining(decreases(reaction)) CTD Calcimycin NGF Text_Mining(affects(cotreatment)) CTD Calcimycin NGF Text_Mining(decreases(reaction)) CTD Calcimycin NGF Text_Mining(increases(expression)) CTD Calcimycin NGF Text_Mining(decreases(expression)) CTD Calcimycin NOS3 Text_Mining(decreases(expression)) CTD Calcimycin NOS3 Text_Mining(decreases(reaction)) CTD Calcimycin NOS3 Text_Mining(increases(expression)) CTD Calcimycin PRKCD Text_Mining(affects(cotreatment)) CTD Calcimycin PRKCD Text_Mining(decreases(reaction)) CTD Calcimycin PRKCD Text_Mining(increases(phosphorylation)) CTD Calcimycin PTGS2 Text_Mining(affects(cotreatment)) CTD Calcimycin PTGS2 Text_Mining(increases(expression)) CTD Calcimycin PTGS2 Text_Mining(increases(reaction)) CTD Calcimycin PTGS2 Text_Mining(increases(activity)) CTD Calcimycin PTGS2 Text_Mining(decreases(reaction)) CTD Calcimycin RCAN1 Text_Mining(increases(expression)) CTD Calcimycin RELA Text_Mining(affects(cotreatment)) CTD Calcimycin RELA Text_Mining(affects(localization)) CTD Calcimycin RELA Text_Mining(decreases(reaction)) CTD Calcimycin RELA Text_Mining(increases(activity)) CTD Calcimycin RELA Text_Mining(increases(response to substance)) CTD Calcimycin RELA Text_Mining(increases(expression)) CTD Calcimycin SELL Text_Mining(decreases(expression)) CTD Calcimycin SELL Text_Mining(decreases(reaction)) CTD Calcimycin SP1 Text_Mining(affects(cotreatment)) CTD Calcimycin SP1 Text_Mining(affects(localization)) CTD Calcimycin TNF Text_Mining(affects(cotreatment)) CTD Calcimycin TNF Text_Mining(decreases(reaction)) CTD Calcimycin TNF Text_Mining(increases(expression)) CTD Calcimycin TNF Text_Mining(increases(secretion)) CTD Calcimycin TNFSF10 Text_Mining(affects(cotreatment)) CTD Calcimycin TNFSF10 Text_Mining(decreases(reaction)) CTD Calcimycin TNFSF10 Text_Mining(increases(expression)) CTD Calcimycin TNFSF10 Text_Mining(increases(reaction)) CTD Calcimycin UHRF1 Text_Mining(decreases(expression)) CTD Calcimycin VEGFA Text_Mining(decreases(reaction)) CTD Calcimycin VEGFA Text_Mining(increases(expression)) CTD Calcimycin VEGFA Text_Mining(increases(secretion)) CTD Calcimycin XBP1 Text_Mining(increases(splicing)) CTD Calcimycin XBP1 Text_Mining(decreases(reaction)) CTD Calcimycin APLNR IC50_CXCR6_Mean=None(uM) D4 PubChem Calcimycin APLNR None=None(uM) D4 PubChem Calcimycin ATAD5 Potency=5.8024(uM) D4 PubChem Calcimycin ATAD5 Potency=12.99(uM) D4 PubChem Calcimycin ATAD5 Potency=5802.4(nM) D4 ChEMBL Calcimycin ATAD5 Potency=12990.0(nM) D4 ChEMBL Calcimycin ATXN2 Potency=3.1623(uM) D4 PubChem Calcimycin ATXN2 Potency=3.5481(uM) D4 PubChem Calcimycin ATXN2 Potency=7.0795(uM) D4 PubChem Calcimycin AVPR1A None=None(uM) D4 PubChem Calcimycin CACNA1H None=None(uM) D4 PubChem Calcimycin CBX1 Potency=0.006(uM) D4 PubChem Calcimycin CBX1 Potency=6.0(nM) D4 ChEMBL Calcimycin CCR6 None=None(uM) D4 PubChem Calcimycin CCR6 IC50_CXCR6_Mean=None(uM) D4 PubChem Calcimycin CHRM1 None=None(uM) D4 PubChem Calcimycin CRHBP None=None(uM) D4 PubChem Calcimycin CRHR2 None=None(uM) D4 PubChem Calcimycin CXCR6 None=None(uM) D4 PubChem Calcimycin CXCR6 IC50_CXCR6_Mean=None(uM) D4 PubChem Calcimycin DRD1 Potency=0.3981(uM) D4 PubChem Calcimycin DRD1 None=None(uM) D4 PubChem Calcimycin DRD1 Potency=398.1(nM) D4 ChEMBL Calcimycin DRD2 None=None(uM) D4 PubChem Calcimycin EHMT2 Potency=17.7828(uM) D4 PubChem Calcimycin EPAS1 None=None(uM) D4 PubChem Calcimycin GLS Potency=3.5481(uM) D4 PubChem Calcimycin GMNN Potency=1.5849(uM) D4 PubChem Calcimycin GMNN Potency=4.6109(uM) D4 PubChem Calcimycin GMNN Potency=1584.9(nM) D4 ChEMBL Calcimycin GNA15 None=None(uM) D4 PubChem Calcimycin GSTO1 None=None(uM) D4 PubChem Calcimycin HCRTR1 None=None(uM) D4 PubChem Calcimycin HSP90AA1 AC50_uM=1.074(uM) D4 PubChem Calcimycin IDH1 Potency=1.4581(uM) D4 PubChem Calcimycin KCNH2 Potency=3.1623(uM) D4 PubChem Calcimycin KCNQ1 None=None(uM) D4 PubChem Calcimycin MAPK1 Potency=14.1254(uM) D4 PubChem Calcimycin MAPK1 Potency=14125.4(nM) D4 ChEMBL Calcimycin MDM2 None=None(uM) D4 PubChem Calcimycin MDM4 None=None(uM) D4 PubChem Calcimycin MITF None=None(uM) D4 PubChem Calcimycin MRGPRX1 None=None(uM) D4 PubChem Calcimycin MTOR Potency=2.6122(uM) D4 PubChem Calcimycin MTOR Potency=14.6892(uM) D4 PubChem Calcimycin MTOR Potency=2612.2(nM) D4 ChEMBL Calcimycin MTOR Potency=14689.2(nM) D4 ChEMBL Calcimycin NFE2L2 Potency=1.1582(uM) D4 PubChem Calcimycin NFE2L2 Potency=1158.2(nM) D4 ChEMBL Calcimycin NOD1 EC50=None(uM) D4 PubChem Calcimycin NPSR1 Potency=0.0158(uM) D4 PubChem Calcimycin NPSR1 Potency=1.2589(uM) D4 PubChem Calcimycin NPSR1 Potency=7.9433(uM) D4 PubChem Calcimycin NPSR1 Potency=1258.9(nM) D4 ChEMBL Calcimycin NPSR1 Potency=7943.3(nM) D4 ChEMBL Calcimycin NPSR1 Potency=15.8(nM) D4 ChEMBL Calcimycin OXTR None=None(uM) D4 PubChem Calcimycin PADI4 None=None(uM) D4 PubChem Calcimycin PAX8 None=None(uM) D4 PubChem Calcimycin PLA2G7 None=None(uM) D4 PubChem Calcimycin PPP1CA None=None(uM) D4 PubChem Calcimycin PRMT1 None=None(uM) D4 PubChem Calcimycin PTGER2 None=None(uM) D4 PubChem Calcimycin RGS4 Potency=26.6795(uM) D4 PubChem Calcimycin SLC12A5 None=None(uM) D4 PubChem Calcimycin SMAD3 Potency=1.0323(uM) D4 PubChem Calcimycin SMAD3 Potency=2.0596(uM) D4 PubChem Calcimycin SMAD3 Potency=5.0119(uM) D4 PubChem Calcimycin SMAD3 Potency=6.5131(uM) D4 PubChem Calcimycin STK33 None=None(uM) D4 PubChem Calcimycin TAAR1 None=None(uM) D4 PubChem Calcimycin TDP1 Potency=0.0259(uM) D4 PubChem Calcimycin TDP1 Potency=0.1836(uM) D4 PubChem Calcimycin TDP2 None=None(uM) D4 PubChem Calcimycin TNFRSF10B None=None(uM) D4 PubChem Calcimycin TRHR None=None(uM) D4 PubChem Calcimycin TSHR None=None(uM) D4 PubChem Calcimycin VDR Potency=44.6684(uM) D4 PubChem Calcimycin XBP1 Absolute IC50 (XBP1)=1.41(uM) D4 PubChem Calcimycin XBP1 IC50=1410.0(nM) D4 ChEMBL