Drug Gene Type Source PP242 CRTC2 Text_Mining(decreases(activity)) CTD PP242 MTOR Text_Mining(decreases(activity)) CTD PP242 PML Text_Mining(decreases(response to substance)) CTD PP242 PML Text_Mining(increases(expression)) CTD PP242 AHR AhR Potency (uM)=3.61632(uM) D4 PubChem PP242 AHR Potency-Replicate_1=3.7578(uM) D4 PubChem PP242 CYP19A1 Potency-Replicate_1=0.3349(uM) D4 PubChem PP242 MAPK1 Inhibition=None(Unspecified) D4 ChEMBL PP242 MAPK3 Inhibition=None(Unspecified) D4 ChEMBL PP242 TDP1 Potency=0.0944(uM) D4 PubChem PP242 TDP1 Potency=0.1679(uM) D4 PubChem