Drug Gene Type Source Carfilzomib MAPK8 Text_Mining(increases(activity)) CTD Carfilzomib AR Ratio Potency (uM)=0.0337801(uM) D4 PubChem Carfilzomib AR Potency-Replicate_1=0.1059(uM) D4 PubChem Carfilzomib AR AR Potency (uM)=0.138548(uM) D4 PubChem Carfilzomib CYP19A1 Potency-Replicate_1=0.0335(uM) D4 PubChem Carfilzomib ESR1 Ratio Potency (uM)=0.0600704(uM) D4 PubChem Carfilzomib ESR1 ER Potency (uM)=0.174422(uM) D4 PubChem Carfilzomib ESR1 Potency-Replicate_1=0.1883(uM) D4 PubChem Carfilzomib ESR1 Potency-Replicate_1=0.6007(uM) D4 PubChem Carfilzomib HSPB1 Ratio Potency (uM)=0.188322(uM) D4 PubChem Carfilzomib NFE2L2 Ratio Potency (uM)=0.0446581(uM) D4 PubChem Carfilzomib NFE2L2 Potency-Replicate_1=0.0668(uM) D4 PubChem Carfilzomib PSMA1 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMA2 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMA3 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMA4 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMA5 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMA6 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMA7 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMA8 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMB1 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMB10 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMB11 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMB2 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMB3 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMB4 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMB5 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMB6 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMB7 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMB8 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib PSMB9 Inhibition=None(Unspecified) D4 ChEMBL Carfilzomib TDP1 Potency=0.0042(uM) D4 PubChem Carfilzomib TDP1 Potency=0.0067(uM) D4 PubChem Carfilzomib VDR None=None(uM) D4 PubChem