Drug Gene Type Source PI-103 ABCB1 Text_Mining(decreases(expression)) CTD PI-103 ABCC1 Text_Mining(decreases(expression)) CTD PI-103 AKT1 Text_Mining(affects(binding)) CTD PI-103 AKT1 Text_Mining(decreases(response to substance)) CTD PI-103 AKT1 Text_Mining(decreases(reaction)) CTD PI-103 AKT1 Text_Mining(increases(phosphorylation)) CTD PI-103 AKT1 Text_Mining(decreases(phosphorylation)) CTD PI-103 BAK1 Text_Mining(affects(cotreatment)) CTD PI-103 BAK1 Text_Mining(increases(response to substance)) CTD PI-103 BAX Text_Mining(affects(cotreatment)) CTD PI-103 BAX Text_Mining(increases(response to substance)) CTD PI-103 BAX Text_Mining(decreases(reaction)) CTD PI-103 BAX Text_Mining(increases(activity)) CTD PI-103 BAX Text_Mining(increases(expression)) CTD PI-103 BAX Text_Mining(increases(reaction)) CTD PI-103 BBC3 Text_Mining(affects(cotreatment)) CTD PI-103 BBC3 Text_Mining(increases(expression)) CTD PI-103 BBC3 Text_Mining(increases(reaction)) CTD PI-103 BCL2 Text_Mining(decreases(reaction)) CTD PI-103 BCL2 Text_Mining(increases(activity)) CTD PI-103 BCL2 Text_Mining(increases(cleavage)) CTD PI-103 BCL2 Text_Mining(increases(localization)) CTD PI-103 BCL2 Text_Mining(increases(reaction)) CTD PI-103 BCL2 Text_Mining(increases(expression)) CTD PI-103 BCL2 Text_Mining(affects(cotreatment)) CTD PI-103 BCL2 Text_Mining(decreases(response to substance)) CTD PI-103 BCL2L1 Text_Mining(increases(expression)) CTD PI-103 BCL2L11 Text_Mining(affects(cotreatment)) CTD PI-103 BCL2L11 Text_Mining(decreases(phosphorylation)) CTD PI-103 BID Text_Mining(decreases(reaction)) CTD PI-103 BID Text_Mining(increases(activity)) CTD PI-103 BID Text_Mining(increases(cleavage)) CTD PI-103 BID Text_Mining(increases(localization)) CTD PI-103 BID Text_Mining(increases(reaction)) CTD PI-103 CA9 Text_Mining(decreases(phosphorylation)) CTD PI-103 CASP3 Text_Mining(decreases(reaction)) CTD PI-103 CASP3 Text_Mining(increases(cleavage)) CTD PI-103 CASP3 Text_Mining(increases(reaction)) CTD PI-103 CASP3 Text_Mining(increases(activity)) CTD PI-103 CASP7 Text_Mining(increases(activity)) CTD PI-103 CASP7 Text_Mining(increases(reaction)) CTD PI-103 CASP7 Text_Mining(increases(cleavage)) CTD PI-103 CASP8 Text_Mining(decreases(reaction)) CTD PI-103 CASP8 Text_Mining(increases(cleavage)) CTD PI-103 CASP8 Text_Mining(increases(reaction)) CTD PI-103 CASP9 Text_Mining(decreases(reaction)) CTD PI-103 CASP9 Text_Mining(increases(cleavage)) CTD PI-103 CASP9 Text_Mining(increases(reaction)) CTD PI-103 EGF Text_Mining(decreases(reaction)) CTD PI-103 EGF Text_Mining(increases(phosphorylation)) CTD PI-103 EGF Text_Mining(affects(cotreatment)) CTD PI-103 H2AFX Text_Mining(increases(phosphorylation)) CTD PI-103 H2AFX Text_Mining(increases(reaction)) CTD PI-103 HIF1A Text_Mining(decreases(phosphorylation)) CTD PI-103 MAP2K1 Text_Mining(increases(phosphorylation)) CTD PI-103 MAP2K1 Text_Mining(affects(cotreatment)) CTD PI-103 MAP2K1 Text_Mining(decreases(reaction)) CTD PI-103 MAP2K2 Text_Mining(increases(phosphorylation)) CTD PI-103 MAP2K2 Text_Mining(affects(cotreatment)) CTD PI-103 MAP2K2 Text_Mining(decreases(reaction)) CTD PI-103 MAPK1 Text_Mining(increases(phosphorylation)) CTD PI-103 MAPK1 Text_Mining(affects(cotreatment)) CTD PI-103 MAPK1 Text_Mining(decreases(reaction)) CTD PI-103 MAPK3 Text_Mining(increases(phosphorylation)) CTD PI-103 MAPK3 Text_Mining(affects(cotreatment)) CTD PI-103 MAPK3 Text_Mining(decreases(reaction)) CTD PI-103 MCL1 Text_Mining(affects(cotreatment)) CTD PI-103 MCL1 Text_Mining(decreases(response to substance)) CTD PI-103 MCL1 Text_Mining(decreases(expression)) CTD PI-103 MCL1 Text_Mining(decreases(reaction)) CTD PI-103 MCL1 Text_Mining(increases(expression)) CTD PI-103 MTOR Text_Mining(decreases(reaction)) CTD PI-103 MTOR Text_Mining(increases(phosphorylation)) CTD PI-103 MTOR Text_Mining(affects(cotreatment)) CTD PI-103 PDK1 Text_Mining(affects(binding)) CTD PI-103 PDK1 Text_Mining(decreases(response to substance)) CTD PI-103 PMAIP1 Text_Mining(affects(cotreatment)) CTD PI-103 PMAIP1 Text_Mining(increases(expression)) CTD PI-103 PMAIP1 Text_Mining(increases(response to substance)) CTD PI-103 RPS6 Text_Mining(decreases(expression)) CTD PI-103 RPS6 Text_Mining(decreases(phosphorylation)) CTD PI-103 TP53 Text_Mining(decreases(reaction)) CTD PI-103 TP53 Text_Mining(increases(expression)) CTD PI-103 TP53 Text_Mining(affects(cotreatment)) CTD PI-103 TP53 Text_Mining(increases(reaction)) CTD PI-103 TP53 Text_Mining(increases(activity)) CTD PI-103 TP53 Text_Mining(increases(cleavage)) CTD PI-103 TP53 Text_Mining(increases(response to substance)) CTD PI-103 XIAP Text_Mining(affects(cotreatment)) CTD PI-103 XIAP Text_Mining(decreases(expression)) CTD PI-103 PIK3CA None=1.5(uM) D4 PubChem