Drug Gene Type Source Crizotinib ABCB1 Text_Mining(decreases(reaction)) CTD Crizotinib ABCB1 Text_Mining(decreases(response to substance)) CTD Crizotinib ABCB1 Text_Mining(increases(hydrolysis)) CTD Crizotinib ABCB1 Text_Mining(increases(reaction)) CTD Crizotinib ACACA Text_Mining(increases(phosphorylation)) CTD Crizotinib AKT1 Text_Mining(decreases(phosphorylation)) CTD Crizotinib AKT1 Text_Mining(decreases(reaction)) CTD Crizotinib AKT1 Text_Mining(increases(reaction)) CTD Crizotinib ALK Text_Mining(decreases(response to substance)) CTD Crizotinib ALK Text_Mining(decreases(phosphorylation)) CTD Crizotinib ALK Text_Mining(decreases(reaction)) CTD Crizotinib ALK Text_Mining(affects(binding)) CTD Crizotinib ALK Text_Mining(decreases(activity)) CTD Crizotinib ALK Text_Mining(increases(reaction)) CTD Crizotinib ALK Text_Mining(increases(phosphorylation)) CTD Crizotinib ALK Text_Mining(increases(expression)) CTD Crizotinib ALK Text_Mining(decreases(stability)) CTD Crizotinib ALK Text_Mining(increases(mutagenesis)) CTD Crizotinib ALK Text_Mining(increases(activity)) CTD Crizotinib BCL2L11 Text_Mining(affects(reaction)) CTD Crizotinib BCL2L11 Text_Mining(increases(cleavage)) CTD Crizotinib BCL2L11 Text_Mining(affects(response to substance)) CTD Crizotinib BCL2L11 Text_Mining(increases(expression)) CTD Crizotinib BCL2L11 Text_Mining(increases(reaction)) CTD Crizotinib BIRC2 Text_Mining(decreases(expression)) CTD Crizotinib BIRC2 Text_Mining(increases(expression)) CTD Crizotinib BIRC2 Text_Mining(increases(reaction)) CTD Crizotinib BIRC5 Text_Mining(decreases(expression)) CTD Crizotinib BIRC5 Text_Mining(increases(expression)) CTD Crizotinib BIRC5 Text_Mining(increases(reaction)) CTD Crizotinib CACNA1C Text_Mining(decreases(activity)) CTD Crizotinib CASP3 Text_Mining(affects(reaction)) CTD Crizotinib CASP3 Text_Mining(increases(cleavage)) CTD Crizotinib CASP3 Text_Mining(increases(activity)) CTD Crizotinib CASP3 Text_Mining(increases(reaction)) CTD Crizotinib CASP7 Text_Mining(increases(activity)) CTD Crizotinib CD44 Text_Mining(decreases(expression)) CTD Crizotinib CDA Text_Mining(decreases(expression)) CTD Crizotinib CDA Text_Mining(increases(response to substance)) CTD Crizotinib CRKL Text_Mining(decreases(phosphorylation)) CTD Crizotinib CRKL Text_Mining(increases(expression)) CTD Crizotinib CRKL Text_Mining(increases(phosphorylation)) CTD Crizotinib CYP3A4 Text_Mining(increases(expression)) CTD Crizotinib EGF Text_Mining(decreases(phosphorylation)) CTD Crizotinib EGF Text_Mining(decreases(reaction)) CTD Crizotinib EGF Text_Mining(decreases(response to substance)) CTD Crizotinib EGF Text_Mining(increases(reaction)) CTD Crizotinib EGFR Text_Mining(decreases(response to substance)) CTD Crizotinib EGFR Text_Mining(increases(reaction)) CTD Crizotinib EGFR Text_Mining(increases(phosphorylation)) CTD Crizotinib EML4 Text_Mining(decreases(stability)) CTD Crizotinib EML4 Text_Mining(increases(mutagenesis)) CTD Crizotinib EML4 Text_Mining(decreases(response to substance)) CTD Crizotinib EPCAM Text_Mining(decreases(expression)) CTD Crizotinib FADS2 Text_Mining(increases(expression)) CTD Crizotinib FASN Text_Mining(increases(expression)) CTD Crizotinib FGFR1 Text_Mining(decreases(activity)) CTD Crizotinib FGFR1 Text_Mining(decreases(phosphorylation)) CTD Crizotinib FGFR1 Text_Mining(decreases(reaction)) CTD Crizotinib FGFR1 Text_Mining(increases(expression)) CTD Crizotinib FSHB Text_Mining(decreases(secretion)) CTD Crizotinib HBEGF Text_Mining(decreases(response to substance)) CTD Crizotinib HBEGF Text_Mining(increases(reaction)) CTD Crizotinib HBEGF Text_Mining(decreases(reaction)) CTD Crizotinib HBEGF Text_Mining(decreases(phosphorylation)) CTD Crizotinib HGF Text_Mining(decreases(phosphorylation)) CTD Crizotinib HGF Text_Mining(increases(expression)) CTD Crizotinib HGF Text_Mining(increases(phosphorylation)) CTD Crizotinib HGF Text_Mining(decreases(activity)) CTD Crizotinib HGF Text_Mining(decreases(reaction)) CTD Crizotinib HMGCR Text_Mining(increases(expression)) CTD Crizotinib HMGCS1 Text_Mining(increases(expression)) CTD Crizotinib INSIG1 Text_Mining(increases(expression)) CTD Crizotinib KCNH2 Text_Mining(decreases(activity)) CTD Crizotinib KIT Text_Mining(decreases(response to substance)) CTD Crizotinib KRAS Text_Mining(decreases(response to substance)) CTD Crizotinib LCK Text_Mining(decreases(activity)) CTD Crizotinib LHB Text_Mining(decreases(secretion)) CTD Crizotinib MAPK1 Text_Mining(decreases(reaction)) CTD Crizotinib MAPK1 Text_Mining(increases(phosphorylation)) CTD Crizotinib MAPK1 Text_Mining(decreases(phosphorylation)) CTD Crizotinib MAPK1 Text_Mining(increases(expression)) CTD Crizotinib MAPK1 Text_Mining(decreases(response to substance)) CTD Crizotinib MAPK1 Text_Mining(increases(reaction)) CTD Crizotinib MAPK3 Text_Mining(decreases(reaction)) CTD Crizotinib MAPK3 Text_Mining(increases(phosphorylation)) CTD Crizotinib MAPK3 Text_Mining(decreases(phosphorylation)) CTD Crizotinib MAPK3 Text_Mining(increases(expression)) CTD Crizotinib MAPK3 Text_Mining(decreases(response to substance)) CTD Crizotinib MAPK3 Text_Mining(increases(reaction)) CTD Crizotinib MET Text_Mining(decreases(response to substance)) CTD Crizotinib MET Text_Mining(increases(mutagenesis)) CTD Crizotinib MET Text_Mining(affects(binding)) CTD Crizotinib MET Text_Mining(decreases(activity)) CTD Crizotinib MET Text_Mining(decreases(reaction)) CTD Crizotinib MET Text_Mining(decreases(phosphorylation)) CTD Crizotinib MET Text_Mining(increases(expression)) CTD Crizotinib MET Text_Mining(increases(phosphorylation)) CTD Crizotinib MET Text_Mining(increases(reaction)) CTD Crizotinib MET Text_Mining(increases(cleavage)) CTD Crizotinib MET Text_Mining(increases(response to substance)) CTD Crizotinib MYCN Text_Mining(decreases(reaction)) CTD Crizotinib MYCN Text_Mining(increases(expression)) CTD Crizotinib PROM1 Text_Mining(decreases(expression)) CTD Crizotinib ROS1 Text_Mining(decreases(phosphorylation)) CTD Crizotinib RPS6 Text_Mining(decreases(phosphorylation)) CTD Crizotinib SCN5A Text_Mining(decreases(activity)) CTD Crizotinib SREBF2 Text_Mining(increases(expression)) CTD Crizotinib STAT3 Text_Mining(decreases(phosphorylation)) CTD Crizotinib STAT3 Text_Mining(increases(expression)) CTD Crizotinib STAT3 Text_Mining(increases(phosphorylation)) CTD Crizotinib STAT3 Text_Mining(increases(reaction)) CTD Crizotinib TGFA Text_Mining(decreases(response to substance)) CTD Crizotinib TGFA Text_Mining(increases(reaction)) CTD Crizotinib TGFA Text_Mining(decreases(reaction)) CTD Crizotinib TGFA Text_Mining(decreases(phosphorylation)) CTD Crizotinib TWIST1 Text_Mining(decreases(response to substance)) CTD Crizotinib VIM Text_Mining(decreases(expression)) CTD Crizotinib XIAP Text_Mining(decreases(expression)) CTD Crizotinib XIAP Text_Mining(increases(expression)) CTD Crizotinib XIAP Text_Mining(increases(reaction)) CTD Crizotinib ALK Inhibition=None(Unspecified) D4 ChEMBL Crizotinib YES1 Potency=0.6884(uM) D4 PubChem