Drug Gene Type Source dorsomorphin ABCB1 Text_Mining(decreases(expression)) CTD dorsomorphin ABCB1 Text_Mining(decreases(reaction)) CTD dorsomorphin ACACA Text_Mining(decreases(reaction)) CTD dorsomorphin ACACA Text_Mining(increases(phosphorylation)) CTD dorsomorphin AKT1 Text_Mining(decreases(phosphorylation)) CTD dorsomorphin AKT1 Text_Mining(decreases(reaction)) CTD dorsomorphin AKT1 Text_Mining(increases(phosphorylation)) CTD dorsomorphin ALB Text_Mining(decreases(reaction)) CTD dorsomorphin ALB Text_Mining(increases(expression)) CTD dorsomorphin APP Text_Mining(decreases(expression)) CTD dorsomorphin APP Text_Mining(decreases(reaction)) CTD dorsomorphin ATM Text_Mining(increases(phosphorylation)) CTD dorsomorphin ATM Text_Mining(decreases(reaction)) CTD dorsomorphin BAX Text_Mining(increases(expression)) CTD dorsomorphin CAMP Text_Mining(affects(localization)) CTD dorsomorphin CAMP Text_Mining(decreases(reaction)) CTD dorsomorphin CASP3 Text_Mining(increases(cleavage)) CTD dorsomorphin CASP3 Text_Mining(decreases(reaction)) CTD dorsomorphin CCNB1 Text_Mining(decreases(expression)) CTD dorsomorphin CCNB1 Text_Mining(decreases(reaction)) CTD dorsomorphin CDK1 Text_Mining(decreases(expression)) CTD dorsomorphin CDK1 Text_Mining(decreases(phosphorylation)) CTD dorsomorphin CDK1 Text_Mining(decreases(reaction)) CTD dorsomorphin CDKN1A Text_Mining(increases(expression)) CTD dorsomorphin CDKN1A Text_Mining(decreases(reaction)) CTD dorsomorphin CHEK2 Text_Mining(increases(phosphorylation)) CTD dorsomorphin CHEK2 Text_Mining(decreases(reaction)) CTD dorsomorphin CREB1 Text_Mining(increases(phosphorylation)) CTD dorsomorphin CYBA Text_Mining(decreases(reaction)) CTD dorsomorphin CYBA Text_Mining(increases(expression)) CTD dorsomorphin CYP4F2 Text_Mining(decreases(reaction)) CTD dorsomorphin CYP4F2 Text_Mining(increases(expression)) CTD dorsomorphin FAS Text_Mining(decreases(reaction)) CTD dorsomorphin FAS Text_Mining(increases(expression)) CTD dorsomorphin G6PC3 Text_Mining(decreases(expression)) CTD dorsomorphin G6PC3 Text_Mining(decreases(reaction)) CTD dorsomorphin GCLC Text_Mining(decreases(reaction)) CTD dorsomorphin GCLC Text_Mining(increases(activity)) CTD dorsomorphin GCLC Text_Mining(increases(expression)) CTD dorsomorphin GDF2 Text_Mining(decreases(reaction)) CTD dorsomorphin GDF2 Text_Mining(increases(phosphorylation)) CTD dorsomorphin GSK3B Text_Mining(decreases(reaction)) CTD dorsomorphin GSK3B Text_Mining(increases(phosphorylation)) CTD dorsomorphin GSK3B Text_Mining(decreases(activity)) CTD dorsomorphin H2AFX Text_Mining(increases(phosphorylation)) CTD dorsomorphin H2AFX Text_Mining(decreases(reaction)) CTD dorsomorphin HMOX1 Text_Mining(decreases(reaction)) CTD dorsomorphin HMOX1 Text_Mining(increases(activity)) CTD dorsomorphin HMOX1 Text_Mining(increases(expression)) CTD dorsomorphin ICAM1 Text_Mining(decreases(reaction)) CTD dorsomorphin ICAM1 Text_Mining(increases(expression)) CTD dorsomorphin KLF2 Text_Mining(decreases(expression)) CTD dorsomorphin MTOR Text_Mining(decreases(phosphorylation)) CTD dorsomorphin MTOR Text_Mining(decreases(reaction)) CTD dorsomorphin NFE2L2 Text_Mining(decreases(reaction)) CTD dorsomorphin NFE2L2 Text_Mining(increases(activity)) CTD dorsomorphin NFE2L2 Text_Mining(increases(expression)) CTD dorsomorphin NFE2L2 Text_Mining(affects(localization)) CTD dorsomorphin NOS3 Text_Mining(decreases(reaction)) CTD dorsomorphin NOS3 Text_Mining(increases(activity)) CTD dorsomorphin NR0B2 Text_Mining(decreases(reaction)) CTD dorsomorphin NR0B2 Text_Mining(increases(expression)) CTD dorsomorphin PARP1 Text_Mining(increases(cleavage)) CTD dorsomorphin PARP1 Text_Mining(decreases(reaction)) CTD dorsomorphin PCK1 Text_Mining(decreases(expression)) CTD dorsomorphin PCK1 Text_Mining(decreases(reaction)) CTD dorsomorphin PPARGC1A Text_Mining(decreases(expression)) CTD dorsomorphin PPARGC1A Text_Mining(decreases(reaction)) CTD dorsomorphin PRKAA1 Text_Mining(decreases(phosphorylation)) CTD dorsomorphin PRKAA1 Text_Mining(decreases(reaction)) CTD dorsomorphin PRKAA1 Text_Mining(increases(phosphorylation)) CTD dorsomorphin PRKAA2 Text_Mining(decreases(phosphorylation)) CTD dorsomorphin PRKAA2 Text_Mining(decreases(reaction)) CTD dorsomorphin PRKAA2 Text_Mining(increases(phosphorylation)) CTD dorsomorphin RPS6 Text_Mining(decreases(phosphorylation)) CTD dorsomorphin RPS6 Text_Mining(decreases(reaction)) CTD dorsomorphin SELE Text_Mining(decreases(reaction)) CTD dorsomorphin SELE Text_Mining(increases(expression)) CTD dorsomorphin SMAD1 Text_Mining(decreases(reaction)) CTD dorsomorphin SMAD1 Text_Mining(increases(phosphorylation)) CTD dorsomorphin SMAD5 Text_Mining(decreases(reaction)) CTD dorsomorphin SMAD5 Text_Mining(increases(phosphorylation)) CTD dorsomorphin SMAD9 Text_Mining(decreases(reaction)) CTD dorsomorphin SMAD9 Text_Mining(increases(phosphorylation)) CTD dorsomorphin SOX17 Text_Mining(decreases(localization)) CTD dorsomorphin SREBF1 Text_Mining(decreases(reaction)) CTD dorsomorphin SREBF1 Text_Mining(increases(expression)) CTD dorsomorphin SREBF1 Text_Mining(decreases(expression)) CTD dorsomorphin STK11 Text_Mining(decreases(reaction)) CTD dorsomorphin STK11 Text_Mining(increases(phosphorylation)) CTD dorsomorphin TP53 Text_Mining(affects(localization)) CTD dorsomorphin TP53 Text_Mining(decreases(reaction)) CTD dorsomorphin TP53 Text_Mining(increases(phosphorylation)) CTD dorsomorphin TP53 Text_Mining(increases(expression)) CTD dorsomorphin TP53 Text_Mining(decreases(expression)) CTD dorsomorphin TP53 Text_Mining(decreases(phosphorylation)) CTD dorsomorphin TP53 Text_Mining(increases(cleavage)) CTD dorsomorphin TP53 Text_Mining(increases(response to substance)) CTD dorsomorphin VCAM1 Text_Mining(decreases(reaction)) CTD dorsomorphin VCAM1 Text_Mining(increases(expression)) CTD dorsomorphin YES1 Potency=0.0547(uM) D4 PubChem dorsomorphin YES1 Potency=0.1959(uM) D4 PubChem