Drug Gene Type Source Lapatinib ABCB11 Text_Mining(decreases(activity)) CTD Lapatinib AKT1 Text_Mining(affects(cotreatment)) CTD Lapatinib AKT1 Text_Mining(decreases(phosphorylation)) CTD Lapatinib AKT1 Text_Mining(decreases(activity)) CTD Lapatinib AKT1 Text_Mining(decreases(expression)) CTD Lapatinib BIRC5 Text_Mining(decreases(expression)) CTD Lapatinib CCND1 Text_Mining(affects(cotreatment)) CTD Lapatinib CCND1 Text_Mining(decreases(expression)) CTD Lapatinib CCNE1 Text_Mining(affects(binding)) CTD Lapatinib CCNE1 Text_Mining(affects(cotreatment)) CTD Lapatinib CCNE1 Text_Mining(decreases(activity)) CTD Lapatinib CCNE1 Text_Mining(increases(reaction)) CTD Lapatinib CDK2 Text_Mining(affects(binding)) CTD Lapatinib CDK2 Text_Mining(affects(cotreatment)) CTD Lapatinib CDK2 Text_Mining(decreases(activity)) CTD Lapatinib CDK2 Text_Mining(increases(reaction)) CTD Lapatinib CDKN1B Text_Mining(affects(binding)) CTD Lapatinib CDKN1B Text_Mining(affects(cotreatment)) CTD Lapatinib CDKN1B Text_Mining(decreases(activity)) CTD Lapatinib CDKN1B Text_Mining(increases(reaction)) CTD Lapatinib CDKN1B Text_Mining(increases(expression)) CTD Lapatinib EGFR Text_Mining(decreases(activity)) CTD Lapatinib ERBB2 Text_Mining(decreases(phosphorylation)) CTD Lapatinib ERBB2 Text_Mining(increases(reaction)) CTD Lapatinib ERBB2 Text_Mining(decreases(activity)) CTD Lapatinib ERBB2 Text_Mining(decreases(expression)) CTD Lapatinib ERBB3 Text_Mining(decreases(activity)) CTD Lapatinib ERBB3 Text_Mining(decreases(expression)) CTD Lapatinib ESR1 Text_Mining(affects(cotreatment)) CTD Lapatinib ESR1 Text_Mining(decreases(activity)) CTD Lapatinib MAPK1 Text_Mining(decreases(reaction)) CTD Lapatinib MAPK1 Text_Mining(increases(phosphorylation)) CTD Lapatinib MAPK1 Text_Mining(decreases(expression)) CTD Lapatinib MAPK1 Text_Mining(decreases(phosphorylation)) CTD Lapatinib MAPK3 Text_Mining(decreases(reaction)) CTD Lapatinib MAPK3 Text_Mining(increases(phosphorylation)) CTD Lapatinib MAPK3 Text_Mining(decreases(expression)) CTD Lapatinib MAPK3 Text_Mining(decreases(phosphorylation)) CTD Lapatinib EGFR None=0.92(uM) D4 PubChem Lapatinib EGFR None=1.2(uM) D4 PubChem Lapatinib EGFR None=2.1(uM) D4 PubChem Lapatinib EGFR None=2.2(uM) D4 PubChem Lapatinib EGFR None=2.4(uM) D4 PubChem Lapatinib EGFR None=2.8(uM) D4 PubChem Lapatinib EGFR None=3.5(uM) D4 PubChem Lapatinib EGFR None=3.9(uM) D4 PubChem Lapatinib EGFR None=4.2(uM) D4 PubChem Lapatinib EGFR None=8.6(uM) D4 PubChem Lapatinib EGFR Inhibition=None(Unspecified) D4 ChEMBL Lapatinib ERBB2 None=7.0(uM) D4 PubChem Lapatinib ERBB2 Inhibition=None(Unspecified) D4 ChEMBL Lapatinib HSPB1 Ratio Potency (uM)=26.6011(uM) D4 PubChem Lapatinib NFE2L2 Ratio Potency (uM)=4.216(uM) D4 PubChem Lapatinib YES1 Potency=4.3432(uM) D4 PubChem