Drug Gene Type Source GW0742 AKT1 Text_Mining(decreases(reaction)) CTD GW0742 AKT1 Text_Mining(increases(phosphorylation)) CTD GW0742 AKT1 Text_Mining(increases(reaction)) CTD GW0742 ANGPTL4 Text_Mining(decreases(reaction)) CTD GW0742 ANGPTL4 Text_Mining(increases(expression)) CTD GW0742 NOS3 Text_Mining(decreases(reaction)) CTD GW0742 NOS3 Text_Mining(increases(phosphorylation)) CTD GW0742 NOS3 Text_Mining(increases(reaction)) CTD GW0742 PARP1 Text_Mining(increases(cleavage)) CTD GW0742 PARP1 Text_Mining(increases(reaction)) CTD GW0742 PLIN2 Text_Mining(decreases(reaction)) CTD GW0742 PLIN2 Text_Mining(increases(expression)) CTD GW0742 PPARD Text_Mining(decreases(reaction)) CTD GW0742 PPARD Text_Mining(increases(activity)) CTD GW0742 PPARD Text_Mining(affects(binding)) CTD GW0742 PPARD Text_Mining(increases(phosphorylation)) CTD GW0742 PPARD Text_Mining(increases(reaction)) CTD GW0742 YWHAE Text_Mining(affects(cotreatment)) CTD GW0742 YWHAE Text_Mining(increases(expression)) CTD GW0742 CYP3A4 Potency=7.9433(uM) D4 PubChem GW0742 CYP3A4 Potency=7943.3(nM) D4 ChEMBL GW0742 HPGD Potency=10.0(uM) D4 PubChem GW0742 HPGD Potency=10000.0(nM) D4 ChEMBL GW0742 KAT2A Potency=31.6228(uM) D4 PubChem GW0742 KAT2A Potency=31622.8(nM) D4 ChEMBL GW0742 MYC None=None(uM) D4 PubChem GW0742 NFE2L2 Potency=68.5896(uM) D4 PubChem GW0742 NR1I2 Potency-Replicate_1=44.6684(uM) D4 PubChem GW0742 PPARD Ratio Potency (uM)=0.001(uM) D4 PubChem GW0742 PPARD Activity=None(Unspecified) D4 ChEMBL GW0742 PPARG Ratio Potency (uM)=1.1391(uM) D4 PubChem GW0742 PPARG Potency-Replicate_1=2.4541(uM) D4 PubChem GW0742 VDR Potency=19.9526(uM) D4 PubChem GW0742 VDR Potency=25.1189(uM) D4 PubChem