Drug Gene Type Source purvalanol A BIRC5 Text_Mining(decreases(expression)) CTD purvalanol A BIRC5 Text_Mining(increases(reaction)) CTD purvalanol A CASP3 Text_Mining(affects(cotreatment)) CTD purvalanol A CASP3 Text_Mining(increases(activity)) CTD purvalanol A CASP9 Text_Mining(affects(cotreatment)) CTD purvalanol A CASP9 Text_Mining(increases(activity)) CTD purvalanol A CDK2 Text_Mining(decreases(activity)) CTD purvalanol A CDKN1A Text_Mining(increases(expression)) CTD purvalanol A CDKN2A Text_Mining(increases(expression)) CTD purvalanol A CSK Text_Mining(decreases(activity)) CTD purvalanol A DYRK1A Text_Mining(decreases(activity)) CTD purvalanol A GSK3B Text_Mining(decreases(activity)) CTD purvalanol A LCK Text_Mining(decreases(activity)) CTD purvalanol A MAPK1 Text_Mining(decreases(activity)) CTD purvalanol A MDM2 Text_Mining(decreases(expression)) CTD purvalanol A RPS6KA1 Text_Mining(decreases(activity)) CTD purvalanol A TP53 Text_Mining(increases(expression)) CTD purvalanol A CYP1A2 None=None(uM) D4 PubChem purvalanol A CYP1A2 AC50=316.23(nM) D4 ChEMBL purvalanol A CYP2C9 Potency=7.9433(uM) D4 PubChem purvalanol A CYP2C9 Potency=7943.3(nM) D4 ChEMBL purvalanol A CYP3A4 Potency=12.5893(uM) D4 PubChem purvalanol A CYP3A4 None=None(uM) D4 PubChem purvalanol A CYP3A4 AC50=12589.2(nM) D4 ChEMBL purvalanol A CYP3A4 Potency=12589.3(nM) D4 ChEMBL purvalanol A HIF1A Potency=10.0(uM) D4 PubChem purvalanol A HIF1A Potency=10000.0(nM) D4 ChEMBL purvalanol A HSD17B10 Potency=31622.8(nM) D4 ChEMBL purvalanol A STAT6 Potency=5.0119(uM) D4 PubChem purvalanol A STAT6 Potency=5011.9(nM) D4 ChEMBL purvalanol A TDP1 Potency=9.4411(uM) D4 PubChem