Drug Gene Type Source GW9662 ABCA1 Text_Mining(decreases(reaction)) CTD GW9662 ABCA1 Text_Mining(increases(expression)) CTD GW9662 ABCA1 Text_Mining(decreases(expression)) CTD GW9662 ADIPOQ Text_Mining(decreases(reaction)) CTD GW9662 ADIPOQ Text_Mining(increases(expression)) CTD GW9662 AGER Text_Mining(affects(binding)) CTD GW9662 AGER Text_Mining(decreases(activity)) CTD GW9662 AGER Text_Mining(decreases(reaction)) CTD GW9662 AGER Text_Mining(increases(expression)) CTD GW9662 AKT1 Text_Mining(decreases(phosphorylation)) CTD GW9662 AKT1 Text_Mining(decreases(reaction)) CTD GW9662 BAX Text_Mining(decreases(reaction)) CTD GW9662 BAX Text_Mining(increases(expression)) CTD GW9662 BCL2 Text_Mining(decreases(expression)) CTD GW9662 BCL2 Text_Mining(decreases(reaction)) CTD GW9662 BSG Text_Mining(decreases(reaction)) CTD GW9662 BSG Text_Mining(increases(expression)) CTD GW9662 BSG Text_Mining(decreases(expression)) CTD GW9662 CASP3 Text_Mining(decreases(reaction)) CTD GW9662 CASP3 Text_Mining(increases(activity)) CTD GW9662 CASP3 Text_Mining(increases(reaction)) CTD GW9662 CAV1 Text_Mining(decreases(reaction)) CTD GW9662 CAV1 Text_Mining(increases(expression)) CTD GW9662 CCND1 Text_Mining(decreases(expression)) CTD GW9662 CCND1 Text_Mining(decreases(reaction)) CTD GW9662 CCR2 Text_Mining(affects(binding)) CTD GW9662 CCR2 Text_Mining(decreases(activity)) CTD GW9662 CCR2 Text_Mining(decreases(expression)) CTD GW9662 CCR2 Text_Mining(decreases(reaction)) CTD GW9662 CD1A Text_Mining(decreases(expression)) CTD GW9662 CD1A Text_Mining(decreases(reaction)) CTD GW9662 CD36 Text_Mining(decreases(expression)) CTD GW9662 CD36 Text_Mining(decreases(reaction)) CTD GW9662 CD36 Text_Mining(increases(expression)) CTD GW9662 CD80 Text_Mining(decreases(expression)) CTD GW9662 CD80 Text_Mining(decreases(reaction)) CTD GW9662 CD86 Text_Mining(decreases(reaction)) CTD GW9662 CD86 Text_Mining(increases(expression)) CTD GW9662 CDKN1A Text_Mining(decreases(reaction)) CTD GW9662 CDKN1A Text_Mining(increases(expression)) CTD GW9662 CXCL8 Text_Mining(decreases(degradation)) CTD GW9662 CXCL8 Text_Mining(increases(reaction)) CTD GW9662 CYCS Text_Mining(affects(binding)) CTD GW9662 CYCS Text_Mining(affects(localization)) CTD GW9662 CYCS Text_Mining(decreases(activity)) CTD GW9662 CYCS Text_Mining(decreases(reaction)) CTD GW9662 CYP27A1 Text_Mining(decreases(reaction)) CTD GW9662 CYP27A1 Text_Mining(increases(expression)) CTD GW9662 CYP27A1 Text_Mining(decreases(expression)) CTD GW9662 FA2H Text_Mining(decreases(reaction)) CTD GW9662 FA2H Text_Mining(increases(expression)) CTD GW9662 FABP1 Text_Mining(decreases(reaction)) CTD GW9662 FABP1 Text_Mining(increases(expression)) CTD GW9662 FABP4 Text_Mining(decreases(reaction)) CTD GW9662 FABP4 Text_Mining(increases(expression)) CTD GW9662 FADS2 Text_Mining(decreases(activity)) CTD GW9662 FADS2 Text_Mining(decreases(reaction)) CTD GW9662 FADS2 Text_Mining(increases(expression)) CTD GW9662 FN1 Text_Mining(decreases(expression)) CTD GW9662 FN1 Text_Mining(decreases(reaction)) CTD GW9662 FSHB Text_Mining(affects(binding)) CTD GW9662 FSHB Text_Mining(decreases(activity)) CTD GW9662 FSHB Text_Mining(decreases(reaction)) CTD GW9662 FSHB Text_Mining(increases(reaction)) CTD GW9662 FSHB Text_Mining(increases(secretion)) CTD GW9662 FSHB Text_Mining(decreases(response to substance)) CTD GW9662 GCLC Text_Mining(increases(expression)) CTD GW9662 GCLM Text_Mining(increases(expression)) CTD GW9662 GDF15 Text_Mining(decreases(activity)) CTD GW9662 GDF15 Text_Mining(decreases(reaction)) CTD GW9662 GDF15 Text_Mining(increases(expression)) CTD GW9662 HMOX1 Text_Mining(decreases(expression)) CTD GW9662 HMOX1 Text_Mining(decreases(reaction)) CTD GW9662 IDE Text_Mining(decreases(reaction)) CTD GW9662 IDE Text_Mining(increases(expression)) CTD GW9662 IL10 Text_Mining(decreases(reaction)) CTD GW9662 IL10 Text_Mining(increases(secretion)) CTD GW9662 IL10 Text_Mining(increases(expression)) CTD GW9662 IL12A Text_Mining(affects(binding)) CTD GW9662 IL12A Text_Mining(decreases(reaction)) CTD GW9662 IL12A Text_Mining(increases(secretion)) CTD GW9662 IL12B Text_Mining(affects(binding)) CTD GW9662 IL12B Text_Mining(decreases(reaction)) CTD GW9662 IL12B Text_Mining(increases(secretion)) CTD GW9662 INS Text_Mining(decreases(expression)) CTD GW9662 INS Text_Mining(decreases(reaction)) CTD GW9662 MMP9 Text_Mining(decreases(reaction)) CTD GW9662 MMP9 Text_Mining(increases(secretion)) CTD GW9662 MMP9 Text_Mining(increases(activity)) CTD GW9662 MMP9 Text_Mining(affects(expression)) CTD GW9662 NFE2L2 Text_Mining(decreases(expression)) CTD GW9662 NFE2L2 Text_Mining(decreases(reaction)) CTD GW9662 NQO1 Text_Mining(increases(expression)) CTD GW9662 PPARA Text_Mining(decreases(reaction)) CTD GW9662 PPARA Text_Mining(increases(activity)) CTD GW9662 PPARG Text_Mining(affects(localization)) CTD GW9662 PPARG Text_Mining(affects(reaction)) CTD GW9662 PPARG Text_Mining(affects(binding)) CTD GW9662 PPARG Text_Mining(decreases(activity)) CTD GW9662 PPARG Text_Mining(decreases(reaction)) CTD GW9662 PPARG Text_Mining(increases(reaction)) CTD GW9662 PPARG Text_Mining(increases(secretion)) CTD GW9662 PPARG Text_Mining(decreases(abundance)) CTD GW9662 PPARG Text_Mining(increases(expression)) CTD GW9662 PPARG Text_Mining(decreases(expression)) CTD GW9662 PPARG Text_Mining(decreases(response to substance)) CTD GW9662 PPARG Text_Mining(increases(abundance)) CTD GW9662 PPARG Text_Mining(increases(activity)) CTD GW9662 PPARG Text_Mining(increases(uptake)) CTD GW9662 PRODH Text_Mining(affects(binding)) CTD GW9662 PRODH Text_Mining(decreases(activity)) CTD GW9662 PRODH Text_Mining(decreases(reaction)) CTD GW9662 PRODH Text_Mining(increases(expression)) CTD GW9662 PTEN Text_Mining(decreases(reaction)) CTD GW9662 PTEN Text_Mining(increases(expression)) CTD GW9662 PTGS2 Text_Mining(decreases(reaction)) CTD GW9662 PTGS2 Text_Mining(increases(expression)) CTD GW9662 PTGS2 Text_Mining(decreases(expression)) CTD GW9662 SCD Text_Mining(decreases(activity)) CTD GW9662 SCD Text_Mining(decreases(reaction)) CTD GW9662 SCD Text_Mining(increases(expression)) CTD GW9662 TJP1 Text_Mining(affects(localization)) CTD GW9662 TJP1 Text_Mining(decreases(reaction)) CTD GW9662 TJP1 Text_Mining(decreases(expression)) CTD GW9662 TNF Text_Mining(affects(binding)) CTD GW9662 TNF Text_Mining(decreases(activity)) CTD GW9662 TNF Text_Mining(decreases(reaction)) CTD GW9662 TNF Text_Mining(increases(reaction)) CTD GW9662 TNF Text_Mining(increases(secretion)) CTD GW9662 TNF Text_Mining(decreases(response to substance)) CTD GW9662 TNF Text_Mining(decreases(secretion)) CTD GW9662 TNF Text_Mining(affects(cotreatment)) CTD GW9662 TNF Text_Mining(increases(expression)) CTD GW9662 VEGFA Text_Mining(decreases(reaction)) CTD GW9662 VEGFA Text_Mining(increases(expression)) CTD GW9662 AHR Potency=14.1254(uM) D4 PubChem GW9662 AHR AhR Potency (uM)=19.3312(uM) D4 PubChem GW9662 AHR Potency-Replicate_1=54.4827(uM) D4 PubChem GW9662 AHR None=None(uM) D4 PubChem GW9662 AR Ratio Potency (uM)=21.0489(uM) D4 PubChem GW9662 AR Potency-Replicate_1=24.5412(uM) D4 PubChem GW9662 CYP1A2 None=None(uM) D4 PubChem GW9662 CYP1A2 AC50=630.96(nM) D4 ChEMBL GW9662 CYP2C19 Potency=0.7943(uM) D4 PubChem GW9662 CYP2C19 None=None(uM) D4 PubChem GW9662 CYP2C19 AC50=794.33(nM) D4 ChEMBL GW9662 CYP2C19 Potency=794.3(nM) D4 ChEMBL GW9662 CYP2C9 Potency=6.3096(uM) D4 PubChem GW9662 CYP2C9 None=None(uM) D4 PubChem GW9662 CYP2C9 AC50=6309.57(nM) D4 ChEMBL GW9662 CYP2C9 Potency=6309.6(nM) D4 ChEMBL GW9662 NCF1 None=None(uM) D4 PubChem GW9662 NFE2L2 Potency=1.2197(uM) D4 PubChem GW9662 NFE2L2 Potency=1.4581(uM) D4 PubChem GW9662 NFE2L2 Potency-Replicate_1=3.0638(uM) D4 PubChem GW9662 NFE2L2 Potency-Replicate_1=7.6959(uM) D4 PubChem GW9662 NFE2L2 Ratio Potency (uM)=14.7772(uM) D4 PubChem GW9662 NR1I2 None=None(uM) D4 PubChem GW9662 NR3C1 None=None(uM) D4 PubChem GW9662 PPARD None=None(uM) D4 PubChem GW9662 PPARG None=None(uM) D4 PubChem GW9662 STK33 None=None(uM) D4 PubChem GW9662 TDP1 Potency=28.1838(uM) D4 PubChem GW9662 TDP1 Potency=29.8554(uM) D4 PubChem GW9662 THPO Potency=1.5849(uM) D4 PubChem GW9662 THPO Potency=1584.9(nM) D4 ChEMBL