Drug Gene Type Source Gefitinib ABCB11 Text_Mining(decreases(activity)) CTD Gefitinib ABCG2 Text_Mining(decreases(reaction)) CTD Gefitinib ABCG2 Text_Mining(decreases(response to substance)) CTD Gefitinib ABCG2 Text_Mining(affects(localization)) CTD Gefitinib ABCG2 Text_Mining(decreases(activity)) CTD Gefitinib ABCG2 Text_Mining(decreases(export)) CTD Gefitinib ADORA1 Text_Mining(decreases(expression)) CTD Gefitinib AKT1 Text_Mining(decreases(reaction)) CTD Gefitinib AKT1 Text_Mining(increases(phosphorylation)) CTD Gefitinib AREG Text_Mining(affects(response to substance)) CTD Gefitinib AREG Text_Mining(decreases(response to substance)) CTD Gefitinib AREG Text_Mining(decreases(reaction)) CTD Gefitinib AREG Text_Mining(increases(expression)) CTD Gefitinib AREG Text_Mining(affects(cotreatment)) CTD Gefitinib AREG Text_Mining(increases(phosphorylation)) CTD Gefitinib ATG5 Text_Mining(increases(expression)) CTD Gefitinib ATG7 Text_Mining(increases(expression)) CTD Gefitinib AURKA Text_Mining(decreases(response to substance)) CTD Gefitinib AURKA Text_Mining(increases(degradation)) CTD Gefitinib AURKA Text_Mining(decreases(expression)) CTD Gefitinib AURKA Text_Mining(increases(response to substance)) CTD Gefitinib AVEN Text_Mining(affects(response to substance)) CTD Gefitinib BCL2L11 Text_Mining(increases(response to substance)) CTD Gefitinib BIRC5 Text_Mining(increases(expression)) CTD Gefitinib BIRC5 Text_Mining(decreases(reaction)) CTD Gefitinib CASP3 Text_Mining(increases(activity)) CTD Gefitinib CASP3 Text_Mining(increases(cleavage)) CTD Gefitinib CAV1 Text_Mining(increases(expression)) CTD Gefitinib CCND1 Text_Mining(decreases(expression)) CTD Gefitinib CCND3 Text_Mining(decreases(expression)) CTD Gefitinib CD14 Text_Mining(decreases(reaction)) CTD Gefitinib CD14 Text_Mining(increases(expression)) CTD Gefitinib CD14 Text_Mining(increases(reaction)) CTD Gefitinib CDKN1A Text_Mining(increases(expression)) CTD Gefitinib CDKN1B Text_Mining(affects(cotreatment)) CTD Gefitinib CDKN1B Text_Mining(decreases(expression)) CTD Gefitinib CDKN1B Text_Mining(increases(reaction)) CTD Gefitinib CDKN1B Text_Mining(increases(expression)) CTD Gefitinib CDKN2B Text_Mining(increases(expression)) CTD Gefitinib CGRRF1 Text_Mining(increases(expression)) CTD Gefitinib COL4A3BP Text_Mining(affects(response to substance)) CTD Gefitinib CORO1C Text_Mining(affects(response to substance)) CTD Gefitinib CXCL8 Text_Mining(decreases(reaction)) CTD Gefitinib CXCL8 Text_Mining(increases(expression)) CTD Gefitinib CYCS Text_Mining(affects(localization)) CTD Gefitinib CYP2D6 Text_Mining(affects(metabolic processing)) CTD Gefitinib CYP2F1 Text_Mining(decreases(expression)) CTD Gefitinib CYP3A4 Text_Mining(affects(metabolic processing)) CTD Gefitinib CYP3A5 Text_Mining(affects(metabolic processing)) CTD Gefitinib DUSP3 Text_Mining(affects(response to substance)) CTD Gefitinib DUSP9 Text_Mining(decreases(expression)) CTD Gefitinib E2F1 Text_Mining(decreases(expression)) CTD Gefitinib EGF Text_Mining(affects(localization)) CTD Gefitinib EGF Text_Mining(decreases(reaction)) CTD Gefitinib EGF Text_Mining(increases(phosphorylation)) CTD Gefitinib EGF Text_Mining(increases(activity)) CTD Gefitinib EGF Text_Mining(affects(binding)) CTD Gefitinib EGF Text_Mining(increases(reaction)) CTD Gefitinib EGF Text_Mining(increases(abundance)) CTD Gefitinib EGFR Text_Mining(affects(response to substance)) CTD Gefitinib EGFR Text_Mining(decreases(response to substance)) CTD Gefitinib EGFR Text_Mining(increases(response to substance)) CTD Gefitinib EGFR Text_Mining(affects(cotreatment)) CTD Gefitinib EGFR Text_Mining(decreases(phosphorylation)) CTD Gefitinib EGFR Text_Mining(decreases(reaction)) CTD Gefitinib EGFR Text_Mining(increases(activity)) CTD Gefitinib EGFR Text_Mining(increases(phosphorylation)) CTD Gefitinib EGFR Text_Mining(increases(degradation)) CTD Gefitinib EGFR Text_Mining(affects(binding)) CTD Gefitinib EGFR Text_Mining(increases(reaction)) CTD Gefitinib EGFR Text_Mining(decreases(activity)) CTD Gefitinib EGFR Text_Mining(affects(localization)) CTD Gefitinib EGFR Text_Mining(decreases(export)) CTD Gefitinib EGFR Text_Mining(decreases(expression)) CTD Gefitinib EPOR Text_Mining(increases(expression)) CTD Gefitinib EPS15 Text_Mining(increases(expression)) CTD Gefitinib ERBB2 Text_Mining(decreases(reaction)) CTD Gefitinib ERBB2 Text_Mining(increases(activity)) CTD Gefitinib ERBB2 Text_Mining(increases(phosphorylation)) CTD Gefitinib ERBB2 Text_Mining(affects(binding)) CTD Gefitinib ERBB2 Text_Mining(decreases(activity)) CTD Gefitinib ERBB2 Text_Mining(decreases(phosphorylation)) CTD Gefitinib ERCC1 Text_Mining(affects(response to substance)) CTD Gefitinib ERCC1 Text_Mining(affects(cotreatment)) CTD Gefitinib ESR1 Text_Mining(decreases(phosphorylation)) CTD Gefitinib ESR2 Text_Mining(increases(expression)) CTD Gefitinib FGF6 Text_Mining(increases(expression)) CTD Gefitinib FOXO3 Text_Mining(increases(response to substance)) CTD Gefitinib FOXO3 Text_Mining(affects(localization)) CTD Gefitinib FOXO3 Text_Mining(decreases(phosphorylation)) CTD Gefitinib GADD45A Text_Mining(increases(expression)) CTD Gefitinib GADD45G Text_Mining(decreases(expression)) CTD Gefitinib GARS Text_Mining(increases(expression)) CTD Gefitinib GCLC Text_Mining(affects(response to substance)) CTD Gefitinib GNB2 Text_Mining(decreases(expression)) CTD Gefitinib GUCY2D Text_Mining(decreases(expression)) CTD Gefitinib HBEGF Text_Mining(decreases(reaction)) CTD Gefitinib HBEGF Text_Mining(increases(expression)) CTD Gefitinib IFI6 Text_Mining(decreases(expression)) CTD Gefitinib IGF1R Text_Mining(affects(binding)) CTD Gefitinib IGF1R Text_Mining(increases(reaction)) CTD Gefitinib IGF1R Text_Mining(increases(phosphorylation)) CTD Gefitinib IGF1R Text_Mining(decreases(reaction)) CTD Gefitinib ITGAM Text_Mining(decreases(reaction)) CTD Gefitinib ITGAM Text_Mining(increases(expression)) CTD Gefitinib ITGAM Text_Mining(increases(reaction)) CTD Gefitinib ITGB1 Text_Mining(decreases(response to substance)) CTD Gefitinib ITGB1 Text_Mining(increases(activity)) CTD Gefitinib KRAS Text_Mining(affects(response to substance)) CTD Gefitinib LEPR Text_Mining(decreases(expression)) CTD Gefitinib MAPK1 Text_Mining(decreases(reaction)) CTD Gefitinib MAPK1 Text_Mining(increases(phosphorylation)) CTD Gefitinib MAPK1 Text_Mining(affects(localization)) CTD Gefitinib MAPK1 Text_Mining(increases(activity)) CTD Gefitinib MAPK1 Text_Mining(affects(cotreatment)) CTD Gefitinib MAPK1 Text_Mining(decreases(phosphorylation)) CTD Gefitinib MAPK1 Text_Mining(increases(reaction)) CTD Gefitinib MAPK1 Text_Mining(decreases(expression)) CTD Gefitinib MAPK3 Text_Mining(decreases(reaction)) CTD Gefitinib MAPK3 Text_Mining(increases(phosphorylation)) CTD Gefitinib MAPK3 Text_Mining(affects(localization)) CTD Gefitinib MAPK3 Text_Mining(increases(activity)) CTD Gefitinib MAPK3 Text_Mining(affects(cotreatment)) CTD Gefitinib MAPK3 Text_Mining(decreases(phosphorylation)) CTD Gefitinib MAPK3 Text_Mining(increases(reaction)) CTD Gefitinib MAPK3 Text_Mining(decreases(expression)) CTD Gefitinib MAPK8 Text_Mining(increases(phosphorylation)) CTD Gefitinib MLH1 Text_Mining(decreases(expression)) CTD Gefitinib MTOR Text_Mining(decreases(phosphorylation)) CTD Gefitinib MYC Text_Mining(decreases(expression)) CTD Gefitinib NFKB1 Text_Mining(decreases(expression)) CTD Gefitinib NFKBIA Text_Mining(decreases(response to substance)) CTD Gefitinib NFKBIA Text_Mining(increases(degradation)) CTD Gefitinib NPTX2 Text_Mining(decreases(expression)) CTD Gefitinib NRL Text_Mining(decreases(expression)) CTD Gefitinib OSMR Text_Mining(affects(response to substance)) CTD Gefitinib PARP1 Text_Mining(affects(reaction)) CTD Gefitinib PARP1 Text_Mining(increases(cleavage)) CTD Gefitinib PHLDA2 Text_Mining(affects(response to substance)) CTD Gefitinib PLBD1 Text_Mining(affects(response to substance)) CTD Gefitinib PTGS2 Text_Mining(affects(cotreatment)) CTD Gefitinib PTGS2 Text_Mining(decreases(expression)) CTD Gefitinib PTGS2 Text_Mining(increases(reaction)) CTD Gefitinib PTTG1 Text_Mining(decreases(expression)) CTD Gefitinib PTTG1 Text_Mining(decreases(stability)) CTD Gefitinib PTTG1 Text_Mining(decreases(response to substance)) CTD Gefitinib QSOX1 Text_Mining(increases(expression)) CTD Gefitinib RBM7 Text_Mining(affects(response to substance)) CTD Gefitinib RELA Text_Mining(decreases(reaction)) CTD Gefitinib RELA Text_Mining(increases(phosphorylation)) CTD Gefitinib RELA Text_Mining(decreases(response to substance)) CTD Gefitinib RPA1 Text_Mining(increases(expression)) CTD Gefitinib RPS6KB1 Text_Mining(decreases(phosphorylation)) CTD Gefitinib RRM1 Text_Mining(affects(response to substance)) CTD Gefitinib SFN Text_Mining(decreases(expression)) CTD Gefitinib SKI Text_Mining(increases(expression)) CTD Gefitinib SNAI2 Text_Mining(affects(response to substance)) CTD Gefitinib SOX17 Text_Mining(decreases(localization)) CTD Gefitinib STAT3 Text_Mining(decreases(reaction)) CTD Gefitinib STAT3 Text_Mining(increases(phosphorylation)) CTD Gefitinib TERT Text_Mining(decreases(expression)) CTD Gefitinib TGFA Text_Mining(decreases(reaction)) CTD Gefitinib TGFA Text_Mining(increases(reaction)) CTD Gefitinib TGFA Text_Mining(increases(response to substance)) CTD Gefitinib TGFA Text_Mining(increases(secretion)) CTD Gefitinib TGFA Text_Mining(decreases(response to substance)) CTD Gefitinib TNFRSF1B Text_Mining(decreases(expression)) CTD Gefitinib TP53 Text_Mining(affects(response to substance)) CTD Gefitinib TP53 Text_Mining(decreases(expression)) CTD Gefitinib TP53 Text_Mining(increases(response to substance)) CTD Gefitinib TYMS Text_Mining(decreases(expression)) CTD Gefitinib TYMS Text_Mining(affects(cotreatment)) CTD Gefitinib TYMS Text_Mining(affects(response to substance)) CTD Gefitinib XRCC1 Text_Mining(affects(response to substance)) CTD Gefitinib AHR AhR Potency (uM)=7.21552(uM) D4 PubChem Gefitinib AHR Potency-Replicate_1=14.9601(uM) D4 PubChem Gefitinib EGFR Potency=0.0032(uM) D4 PubChem Gefitinib EGFR EGFR IC50=0.004(uM) D4 PubChem Gefitinib EGFR None=0.52(uM) D4 PubChem Gefitinib EGFR None=0.54(uM) D4 PubChem Gefitinib EGFR None=0.57(uM) D4 PubChem Gefitinib EGFR None=0.94(uM) D4 PubChem Gefitinib EGFR None=0.98(uM) D4 PubChem Gefitinib EGFR None=1.0(uM) D4 PubChem Gefitinib EGFR None=1.1(uM) D4 PubChem Gefitinib EGFR Potency=1.122(uM) D4 PubChem Gefitinib EGFR None=1.4(uM) D4 PubChem Gefitinib EGFR None=2.0(uM) D4 PubChem Gefitinib EGFR Inhibition=None(Unspecified) D4 ChEMBL Gefitinib EGFR Potency=1122.0(nM) D4 ChEMBL Gefitinib EGFR Potency=3.2(nM) D4 ChEMBL Gefitinib ERBB2 Inhibition=None(Unspecified) D4 ChEMBL Gefitinib ESR1 Ratio Potency (uM)=16.9301(uM) D4 PubChem Gefitinib ESR1 Potency-Replicate_1=16.9301(uM) D4 PubChem Gefitinib GMNN Potency=29.8554(uM) D4 PubChem Gefitinib MAPT Potency=39.8107(uM) D4 PubChem Gefitinib MAPT Potency=39810.7(nM) D4 ChEMBL Gefitinib MET Inhibition=None(Unspecified) D4 ChEMBL Gefitinib NFE2L2 Ratio Potency (uM)=4.73043(uM) D4 PubChem Gefitinib PIM1 None=None(uM) D4 PubChem Gefitinib SLK None=None(uM) D4 PubChem Gefitinib YES1 Potency=1.3734(uM) D4 PubChem Gefitinib YES1 Potency=1.7291(uM) D4 PubChem