Drug Gene Type Source Erlotinib ACACA Text_Mining(increases(phosphorylation)) CTD Erlotinib AREG Text_Mining(affects(response to substance)) CTD Erlotinib ATG5 Text_Mining(decreases(response to substance)) CTD Erlotinib ATG5 Text_Mining(increases(expression)) CTD Erlotinib ATG7 Text_Mining(increases(expression)) CTD Erlotinib AXL Text_Mining(decreases(response to substance)) CTD Erlotinib AXL Text_Mining(decreases(activity)) CTD Erlotinib AXL Text_Mining(increases(response to substance)) CTD Erlotinib BCL2 Text_Mining(increases(expression)) CTD Erlotinib BCL2 Text_Mining(decreases(reaction)) CTD Erlotinib BCL2 Text_Mining(increases(response to substance)) CTD Erlotinib BCL2L2 Text_Mining(increases(expression)) CTD Erlotinib BCL2L2 Text_Mining(decreases(reaction)) CTD Erlotinib BCL2L2 Text_Mining(increases(response to substance)) CTD Erlotinib BECN1 Text_Mining(decreases(response to substance)) CTD Erlotinib BRCA1 Text_Mining(decreases(activity)) CTD Erlotinib BRCA1 Text_Mining(decreases(phosphorylation)) CTD Erlotinib CCND1 Text_Mining(decreases(reaction)) CTD Erlotinib CCND1 Text_Mining(increases(expression)) CTD Erlotinib CDH1 Text_Mining(decreases(glycosylation)) CTD Erlotinib CDH1 Text_Mining(increases(degradation)) CTD Erlotinib CDH1 Text_Mining(increases(reaction)) CTD Erlotinib CHFR Text_Mining(affects(cotreatment)) CTD Erlotinib CHFR Text_Mining(affects(response to substance)) CTD Erlotinib CYP3A4 Text_Mining(decreases(activity)) CTD Erlotinib CYP3A4 Text_Mining(increases(expression)) CTD Erlotinib DDIT3 Text_Mining(increases(expression)) CTD Erlotinib EGF Text_Mining(decreases(reaction)) CTD Erlotinib EGF Text_Mining(decreases(response to substance)) CTD Erlotinib EGF Text_Mining(increases(reaction)) CTD Erlotinib EGF Text_Mining(affects(binding)) CTD Erlotinib EGFR Text_Mining(affects(cotreatment)) CTD Erlotinib EGFR Text_Mining(increases(response to substance)) CTD Erlotinib EGFR Text_Mining(affects(response to substance)) CTD Erlotinib EGFR Text_Mining(decreases(response to substance)) CTD Erlotinib EGFR Text_Mining(decreases(reaction)) CTD Erlotinib EGFR Text_Mining(increases(activity)) CTD Erlotinib EGFR Text_Mining(increases(phosphorylation)) CTD Erlotinib EGFR Text_Mining(decreases(expression)) CTD Erlotinib EGFR Text_Mining(decreases(glycosylation)) CTD Erlotinib EGFR Text_Mining(increases(reaction)) CTD Erlotinib EGFR Text_Mining(affects(binding)) CTD Erlotinib EGFR Text_Mining(decreases(activity)) CTD Erlotinib EGFR Text_Mining(decreases(phosphorylation)) CTD Erlotinib HBEGF Text_Mining(decreases(reaction)) CTD Erlotinib HBEGF Text_Mining(decreases(response to substance)) CTD Erlotinib JAK2 Text_Mining(decreases(phosphorylation)) CTD Erlotinib KCNH2 Text_Mining(affects(activity)) CTD Erlotinib KRAS Text_Mining(increases(response to substance)) CTD Erlotinib MAPK1 Text_Mining(decreases(phosphorylation)) CTD Erlotinib MAPK3 Text_Mining(decreases(phosphorylation)) CTD Erlotinib MET Text_Mining(affects(cotreatment)) CTD Erlotinib MET Text_Mining(decreases(phosphorylation)) CTD Erlotinib MTOR Text_Mining(decreases(phosphorylation)) CTD Erlotinib NOX4 Text_Mining(increases(expression)) CTD Erlotinib NOX4 Text_Mining(increases(stability)) CTD Erlotinib NOX4 Text_Mining(decreases(response to substance)) CTD Erlotinib NR1I2 Text_Mining(affects(binding)) CTD Erlotinib NR1I2 Text_Mining(increases(activity)) CTD Erlotinib PML Text_Mining(increases(expression)) CTD Erlotinib PML Text_Mining(increases(localization)) CTD Erlotinib PML Text_Mining(decreases(response to substance)) CTD Erlotinib PTPN9 Text_Mining(decreases(expression)) CTD Erlotinib PTPN9 Text_Mining(decreases(response to substance)) CTD Erlotinib RAD50 Text_Mining(decreases(activity)) CTD Erlotinib RAD50 Text_Mining(decreases(expression)) CTD Erlotinib RAD51 Text_Mining(decreases(activity)) CTD Erlotinib RAD51 Text_Mining(decreases(expression)) CTD Erlotinib RPS6 Text_Mining(decreases(phosphorylation)) CTD Erlotinib RPS6KB1 Text_Mining(decreases(phosphorylation)) CTD Erlotinib SRC Text_Mining(decreases(phosphorylation)) CTD Erlotinib STAT3 Text_Mining(increases(phosphorylation)) CTD Erlotinib STAT3 Text_Mining(decreases(reaction)) CTD Erlotinib STAT3 Text_Mining(increases(response to substance)) CTD Erlotinib TGFA Text_Mining(decreases(reaction)) CTD Erlotinib TGFA Text_Mining(decreases(response to substance)) CTD Erlotinib TGFB1 Text_Mining(decreases(reaction)) CTD Erlotinib TGFB1 Text_Mining(decreases(response to substance)) CTD Erlotinib TGFB1 Text_Mining(increases(reaction)) CTD Erlotinib AHR AhR Potency (uM)=1.88336(uM) D4 PubChem Erlotinib AHR Potency-Replicate_1=2.6603(uM) D4 PubChem Erlotinib AR Potency-Replicate_1=21.1317(uM) D4 PubChem Erlotinib CLK4 Potency=20.6665(uM) D4 PubChem Erlotinib CLK4 Potency=20666.5(nM) D4 ChEMBL Erlotinib CYP19A1 Potency-Replicate_1=18.8336(uM) D4 PubChem Erlotinib CYP19A1 None=None(uM) D4 PubChem Erlotinib EGFR Potency=0.0008(uM) D4 PubChem Erlotinib EGFR Potency=0.0009(uM) D4 PubChem Erlotinib EGFR EGFR IC50=0.001(uM) D4 PubChem Erlotinib EGFR None=0.35(uM) D4 PubChem Erlotinib EGFR None=0.47(uM) D4 PubChem Erlotinib EGFR None=0.48(uM) D4 PubChem Erlotinib EGFR None=0.52(uM) D4 PubChem Erlotinib EGFR None=0.67(uM) D4 PubChem Erlotinib EGFR None=0.85(uM) D4 PubChem Erlotinib EGFR None=0.97(uM) D4 PubChem Erlotinib EGFR None=1.2(uM) D4 PubChem Erlotinib EGFR None=1.6(uM) D4 PubChem Erlotinib EGFR Inhibition=None(Unspecified) D4 ChEMBL Erlotinib EGFR Potency=0.9(nM) D4 ChEMBL Erlotinib EGFR Potency=0.8(nM) D4 ChEMBL Erlotinib GAK None=3.1(uM) D4 PubChem Erlotinib JAK2 irf1 Inhibition [HEL cells] (IC50)=0.835(uM) D4 PubChem Erlotinib JAK2 Activity=0.835(um) D4 ChEMBL Erlotinib NFE2L2 Ratio Potency (uM)=2.37083(uM) D4 PubChem Erlotinib NR3C1 Ratio Potency (uM)=20.5113(uM) D4 PubChem Erlotinib SLK None=None(uM) D4 PubChem Erlotinib TDP1 Potency=13.3359(uM) D4 PubChem Erlotinib YES1 Potency=0.9723(uM) D4 PubChem