Drug Gene Type Source alsterpaullone AR Text_Mining(increases(activity)) CTD alsterpaullone CDK2 Text_Mining(decreases(activity)) CTD alsterpaullone GSK3B Text_Mining(decreases(activity)) CTD alsterpaullone KLK3 Text_Mining(increases(expression)) CTD alsterpaullone LCK Text_Mining(decreases(activity)) CTD alsterpaullone TP53 Text_Mining(affects(localization)) CTD alsterpaullone TP53 Text_Mining(decreases(degradation)) CTD alsterpaullone TP53 Text_Mining(increases(expression)) CTD alsterpaullone CFTR None=None(uM) D4 PubChem alsterpaullone IL1B None=None(uM) D4 PubChem alsterpaullone NCOA2 None=None(uM) D4 PubChem alsterpaullone NCOA3 None=None(uM) D4 PubChem alsterpaullone NFE2L2 Potency=2.3109(uM) D4 PubChem alsterpaullone NFE2L2 Potency=2310.9(nM) D4 ChEMBL alsterpaullone NR2E3 None=None(uM) D4 PubChem alsterpaullone NR2F2 None=None(uM) D4 PubChem alsterpaullone OPRD1 None=None(uM) D4 PubChem alsterpaullone OPRM1 None=None(uM) D4 PubChem alsterpaullone SMAD3 Potency=0.1636(uM) D4 PubChem alsterpaullone SMAD3 Potency=0.5012(uM) D4 PubChem alsterpaullone SMAD3 Potency=1.2995(uM) D4 PubChem alsterpaullone SMARCA2 None=None(uM) D4 PubChem alsterpaullone STK33 None=None(uM) D4 PubChem alsterpaullone TDP1 Potency=1.8356(uM) D4 PubChem