Drug Gene Type Source kenpaullone ABCB1 Text_Mining(increases(expression)) CTD kenpaullone AR Text_Mining(affects(localization)) CTD kenpaullone AR Text_Mining(increases(activity)) CTD kenpaullone CASP3 Text_Mining(decreases(reaction)) CTD kenpaullone CASP3 Text_Mining(increases(activity)) CTD kenpaullone CDK2 Text_Mining(decreases(activity)) CTD kenpaullone CTNNB1 Text_Mining(affects(localization)) CTD kenpaullone GSK3B Text_Mining(decreases(phosphorylation)) CTD kenpaullone GSK3B Text_Mining(decreases(reaction)) CTD kenpaullone GSK3B Text_Mining(decreases(activity)) CTD kenpaullone KLK3 Text_Mining(increases(expression)) CTD kenpaullone LCK Text_Mining(decreases(activity)) CTD kenpaullone ATAD5 Potency=0.4108(uM) D4 PubChem kenpaullone ATAD5 Potency=410.8(nM) D4 ChEMBL kenpaullone CFTR IC50_CF-PAF_Mean=None(uM) D4 PubChem kenpaullone CFTR None=None(uM) D4 PubChem kenpaullone CYP1A2 None=None(uM) D4 PubChem kenpaullone CYP1A2 AC50=158.49(nM) D4 ChEMBL kenpaullone CYP2D6 Potency=0.3981(uM) D4 PubChem kenpaullone CYP2D6 None=None(uM) D4 PubChem kenpaullone CYP2D6 AC50=398.11(nM) D4 ChEMBL kenpaullone CYP2D6 Potency=398.1(nM) D4 ChEMBL kenpaullone CYP3A4 Potency=12.5893(uM) D4 PubChem kenpaullone CYP3A4 None=None(uM) D4 PubChem kenpaullone CYP3A4 AC50=12589.2(nM) D4 ChEMBL kenpaullone CYP3A4 Potency=12589.3(nM) D4 ChEMBL kenpaullone EHMT2 Potency=39.8107(uM) D4 PubChem kenpaullone EHMT2 Potency=39810.7(nM) D4 ChEMBL kenpaullone GMNN Potency=4.1095(uM) D4 PubChem kenpaullone GMNN Potency=6.3096(uM) D4 PubChem kenpaullone GMNN Potency=6309.6(nM) D4 ChEMBL kenpaullone HTT Potency=2.2387(uM) D4 PubChem kenpaullone HTT Potency=3.5481(uM) D4 PubChem kenpaullone HTT None=None(uM) D4 PubChem kenpaullone HTT Potency=3548.1(nM) D4 ChEMBL kenpaullone HTT Potency=2238.7(nM) D4 ChEMBL kenpaullone IL1B None=None(uM) D4 PubChem kenpaullone ITPKC None=None(uM) D4 PubChem kenpaullone MAPT None=None(uM) D4 PubChem kenpaullone NPC1 Potency=0.5174(uM) D4 PubChem kenpaullone NPC1 Potency=517.4(nM) D4 ChEMBL kenpaullone NR0B1 IC50=0.83352(uM) D4 PubChem kenpaullone NR0B1 None=None(uM) D4 PubChem kenpaullone PAK4 None=None(uM) D4 PubChem kenpaullone PAK6 None=None(uM) D4 PubChem kenpaullone PAK7 None=None(uM) D4 PubChem kenpaullone PARK2 Potency=2.5929(uM) D4 PubChem kenpaullone PARK2 Potency=5.8048(uM) D4 PubChem kenpaullone PIM1 None=None(uM) D4 PubChem kenpaullone RAB9A Potency=0.3663(uM) D4 PubChem kenpaullone RAB9A Potency=366.3(nM) D4 ChEMBL kenpaullone SMAD3 Potency=0.92(uM) D4 PubChem kenpaullone SMAD3 Potency=2.8184(uM) D4 PubChem kenpaullone SMAD3 Potency=2.9093(uM) D4 PubChem kenpaullone SMARCA2 None=None(uM) D4 PubChem kenpaullone SMN1; SMN2 Potency=11220.2(nM) D4 ChEMBL kenpaullone SMN1; SMN2 Potency=15848.9(nM) D4 ChEMBL kenpaullone SMN2 Potency=11.2202(uM) D4 PubChem kenpaullone SMN2 Potency=15.8489(uM) D4 PubChem kenpaullone STK33 None=None(uM) D4 PubChem kenpaullone THPO Potency=0.1585(uM) D4 PubChem kenpaullone THPO Potency=158.5(nM) D4 ChEMBL