Drug Gene Type Source HELENALIN ATF4 Text_Mining(increases(expression)) CTD HELENALIN CASP3 Text_Mining(decreases(reaction)) CTD HELENALIN CASP3 Text_Mining(increases(activity)) CTD HELENALIN CASP8 Text_Mining(decreases(reaction)) CTD HELENALIN CASP8 Text_Mining(increases(activity)) CTD HELENALIN CD40 Text_Mining(decreases(reaction)) CTD HELENALIN CD40 Text_Mining(increases(expression)) CTD HELENALIN CD80 Text_Mining(decreases(reaction)) CTD HELENALIN CD80 Text_Mining(increases(expression)) CTD HELENALIN CD83 Text_Mining(decreases(reaction)) CTD HELENALIN CD83 Text_Mining(increases(expression)) CTD HELENALIN CD86 Text_Mining(decreases(reaction)) CTD HELENALIN CD86 Text_Mining(increases(expression)) CTD HELENALIN DDIT3 Text_Mining(increases(expression)) CTD HELENALIN DDIT4 Text_Mining(increases(expression)) CTD HELENALIN ICAM1 Text_Mining(decreases(reaction)) CTD HELENALIN ICAM1 Text_Mining(increases(expression)) CTD HELENALIN IL10 Text_Mining(decreases(reaction)) CTD HELENALIN IL10 Text_Mining(increases(secretion)) CTD HELENALIN IL12A Text_Mining(affects(binding)) CTD HELENALIN IL12A Text_Mining(decreases(reaction)) CTD HELENALIN IL12A Text_Mining(increases(secretion)) CTD HELENALIN IL12B Text_Mining(affects(binding)) CTD HELENALIN IL12B Text_Mining(decreases(reaction)) CTD HELENALIN IL12B Text_Mining(increases(secretion)) CTD HELENALIN IL6 Text_Mining(decreases(reaction)) CTD HELENALIN IL6 Text_Mining(increases(secretion)) CTD HELENALIN NFKBIA Text_Mining(decreases(expression)) CTD HELENALIN NFKBIA Text_Mining(decreases(reaction)) CTD HELENALIN RELA Text_Mining(decreases(reaction)) CTD HELENALIN RELA Text_Mining(increases(activity)) CTD HELENALIN RELA Text_Mining(increases(localization)) CTD HELENALIN RELA Text_Mining(decreases(activity)) CTD HELENALIN SOD2 Text_Mining(decreases(reaction)) CTD HELENALIN SOD2 Text_Mining(increases(expression)) CTD HELENALIN TNFRSF10A Text_Mining(decreases(reaction)) CTD HELENALIN TNFRSF10A Text_Mining(increases(expression)) CTD HELENALIN ABHD5 None=None(uM) D4 PubChem HELENALIN AGTR1 IC50=18.639(uM) D4 PubChem HELENALIN AGTR1 IC50=18639.0(nM) D4 ChEMBL HELENALIN APLNR None=None(uM) D4 PubChem HELENALIN ATAD5 Potency=0.0045(uM) D4 PubChem HELENALIN ATAD5 Potency=0.0056(uM) D4 PubChem HELENALIN ATAD5 Potency=2.81(uM) D4 PubChem HELENALIN ATAD5 Potency=4.1078(uM) D4 PubChem HELENALIN ATAD5 Potency=7.308(uM) D4 PubChem HELENALIN ATAD5 Potency=4107.8(nM) D4 ChEMBL HELENALIN ATXN2 Potency=19.9526(uM) D4 PubChem HELENALIN CFTR AC50_uM=0.989(uM) D4 PubChem HELENALIN CFTR None=None(uM) D4 PubChem HELENALIN DRD3 None=None(uM) D4 PubChem HELENALIN EHMT2 Potency=11.2202(uM) D4 PubChem HELENALIN EHMT2 Potency=11220.2(nM) D4 ChEMBL HELENALIN EPAS1 None=None(uM) D4 PubChem HELENALIN GLP1R Potency=2.5119(uM) D4 PubChem HELENALIN GMNN Potency=0.92(uM) D4 PubChem HELENALIN GPR183 None=None(uM) D4 PubChem HELENALIN GPR55 IC50=2.64228(uM) D4 PubChem HELENALIN GPR55 IC50=2642.28(nM) D4 ChEMBL HELENALIN HNF4A None=None(uM) D4 PubChem HELENALIN HTT Potency=2.2387(uM) D4 PubChem HELENALIN HTT Potency=2238.7(nM) D4 ChEMBL HELENALIN IDH1 Potency=1.4581(uM) D4 PubChem HELENALIN IL1B None=None(uM) D4 PubChem HELENALIN MAPT Potency=3.5481(uM) D4 PubChem HELENALIN MAPT Potency=3.9811(uM) D4 PubChem HELENALIN MAPT Potency=8912.5(nM) D4 ChEMBL HELENALIN MAPT Potency=3981.1(nM) D4 ChEMBL HELENALIN MAPT Potency=3548.1(nM) D4 ChEMBL HELENALIN MDM2 Mean Wild-type EC50=0.18(uM) D4 PubChem HELENALIN MDM2 EC50=0.42(uM) D4 PubChem HELENALIN MDM2 Mean Mutant EC50=1.11(uM) D4 PubChem HELENALIN MDM2 None=None(uM) D4 PubChem HELENALIN MDM2 EC50=420.0(nM) D4 ChEMBL HELENALIN MDM4 None=None(uM) D4 PubChem HELENALIN MITF None=None(uM) D4 PubChem HELENALIN NCOA2 None=None(uM) D4 PubChem HELENALIN NFE2L2 Potency=3.6626(uM) D4 PubChem HELENALIN NFE2L2 Potency=3662.6(nM) D4 ChEMBL HELENALIN NR2E3 IC50=1.921(uM) D4 PubChem HELENALIN NR2E3 None=None(uM) D4 PubChem HELENALIN NR2F2 None=None(uM) D4 PubChem HELENALIN NR5A2 None=None(uM) D4 PubChem HELENALIN PAX8 None=None(uM) D4 PubChem HELENALIN PLIN5 None=None(uM) D4 PubChem HELENALIN PRNP None=None(uM) D4 PubChem HELENALIN RGS4 Potency=21.1923(uM) D4 PubChem HELENALIN RGS4 None=None(uM) D4 PubChem HELENALIN SMAD3 Potency=3.9811(uM) D4 PubChem HELENALIN TNF None=None(uM) D4 PubChem HELENALIN TNFRSF10B None=None(uM) D4 PubChem HELENALIN TNFSF10 None=None(uM) D4 PubChem HELENALIN XBP1 Absolute IC50 (XBP1)=2.43(uM) D4 PubChem HELENALIN XBP1 IC50=2430.0(nM) D4 ChEMBL