Drug Gene Type Source Tanespimycin ADAMTS1 Text_Mining(increases(expression)) CTD Tanespimycin AKT1 Text_Mining(decreases(expression)) CTD Tanespimycin AKT1 Text_Mining(increases(reaction)) CTD Tanespimycin ALB Text_Mining(affects(binding)) CTD Tanespimycin ALB Text_Mining(decreases(reaction)) CTD Tanespimycin ALB Text_Mining(increases(oxidation)) CTD Tanespimycin ALK Text_Mining(decreases(activity)) CTD Tanespimycin ALK Text_Mining(decreases(expression)) CTD Tanespimycin APAF1 Text_Mining(increases(expression)) CTD Tanespimycin APAF1 Text_Mining(increases(response to substance)) CTD Tanespimycin AR Text_Mining(decreases(expression)) CTD Tanespimycin BCL2 Text_Mining(decreases(expression)) CTD Tanespimycin BCL2L1 Text_Mining(decreases(expression)) CTD Tanespimycin CASP3 Text_Mining(increases(activity)) CTD Tanespimycin CASP3 Text_Mining(increases(response to substance)) CTD Tanespimycin CASP3 Text_Mining(affects(cotreatment)) CTD Tanespimycin CASP3 Text_Mining(increases(cleavage)) CTD Tanespimycin CASP8 Text_Mining(affects(cotreatment)) CTD Tanespimycin CASP8 Text_Mining(increases(cleavage)) CTD Tanespimycin CASP9 Text_Mining(affects(cotreatment)) CTD Tanespimycin CASP9 Text_Mining(increases(cleavage)) CTD Tanespimycin CCND1 Text_Mining(affects(cotreatment)) CTD Tanespimycin CCND1 Text_Mining(decreases(expression)) CTD Tanespimycin CDC25C Text_Mining(affects(cotreatment)) CTD Tanespimycin CDC25C Text_Mining(decreases(expression)) CTD Tanespimycin CDK1 Text_Mining(affects(cotreatment)) CTD Tanespimycin CDK1 Text_Mining(decreases(expression)) CTD Tanespimycin CDK4 Text_Mining(decreases(expression)) CTD Tanespimycin CDK8 Text_Mining(decreases(expression)) CTD Tanespimycin COMMD1 Text_Mining(increases(degradation)) CTD Tanespimycin COMMD1 Text_Mining(increases(reaction)) CTD Tanespimycin CYP3A5 Text_Mining(affects(metabolic processing)) CTD Tanespimycin EGFR Text_Mining(decreases(expression)) CTD Tanespimycin EGFR Text_Mining(increases(degradation)) CTD Tanespimycin ERBB2 Text_Mining(decreases(expression)) CTD Tanespimycin ERBB2 Text_Mining(increases(degradation)) CTD Tanespimycin FGFR3 Text_Mining(decreases(expression)) CTD Tanespimycin FGFR3 Text_Mining(increases(degradation)) CTD Tanespimycin FLT3 Text_Mining(decreases(expression)) CTD Tanespimycin GSK3B Text_Mining(decreases(expression)) CTD Tanespimycin HIF1A Text_Mining(increases(degradation)) CTD Tanespimycin HIF1A Text_Mining(increases(reaction)) CTD Tanespimycin HSF1 Text_Mining(affects(localization)) CTD Tanespimycin HSF1 Text_Mining(increases(expression)) CTD Tanespimycin HSP90AA1 Text_Mining(decreases(expression)) CTD Tanespimycin HSPA1A Text_Mining(affects(localization)) CTD Tanespimycin HSPA1A Text_Mining(increases(expression)) CTD Tanespimycin HSPA4 Text_Mining(increases(expression)) CTD Tanespimycin HSPA4 Text_Mining(decreases(response to substance)) CTD Tanespimycin HSPA5 Text_Mining(increases(expression)) CTD Tanespimycin KIT Text_Mining(decreases(expression)) CTD Tanespimycin KIT Text_Mining(increases(degradation)) CTD Tanespimycin MAPK1 Text_Mining(decreases(phosphorylation)) CTD Tanespimycin MAPK3 Text_Mining(decreases(phosphorylation)) CTD Tanespimycin MCL1 Text_Mining(decreases(expression)) CTD Tanespimycin MDM2 Text_Mining(increases(degradation)) CTD Tanespimycin MMP2 Text_Mining(affects(reaction)) CTD Tanespimycin MMP2 Text_Mining(increases(activity)) CTD Tanespimycin MMP2 Text_Mining(decreases(reaction)) CTD Tanespimycin MMP2 Text_Mining(increases(expression)) CTD Tanespimycin MMP9 Text_Mining(affects(reaction)) CTD Tanespimycin MMP9 Text_Mining(increases(activity)) CTD Tanespimycin MMP9 Text_Mining(decreases(reaction)) CTD Tanespimycin MMP9 Text_Mining(increases(expression)) CTD Tanespimycin MTSS1 Text_Mining(increases(expression)) CTD Tanespimycin NQO1 Text_Mining(decreases(abundance)) CTD Tanespimycin NQO1 Text_Mining(decreases(activity)) CTD Tanespimycin NQO1 Text_Mining(decreases(response to substance)) CTD Tanespimycin NQO1 Text_Mining(increases(abundance)) CTD Tanespimycin NQO1 Text_Mining(increases(reduction)) CTD Tanespimycin NQO1 Text_Mining(increases(chemical synthesis)) CTD Tanespimycin NQO1 Text_Mining(increases(response to substance)) CTD Tanespimycin NQO1 Text_Mining(affects(cotreatment)) CTD Tanespimycin NQO1 Text_Mining(decreases(expression)) CTD Tanespimycin PNN Text_Mining(increases(expression)) CTD Tanespimycin RAF1 Text_Mining(decreases(expression)) CTD Tanespimycin RB1 Text_Mining(affects(cotreatment)) CTD Tanespimycin RB1 Text_Mining(decreases(phosphorylation)) CTD Tanespimycin RPS6 Text_Mining(decreases(phosphorylation)) CTD Tanespimycin SERPINB5 Text_Mining(increases(expression)) CTD Tanespimycin SOD2 Text_Mining(increases(abundance)) CTD Tanespimycin SOD2 Text_Mining(increases(response to substance)) CTD Tanespimycin TIMP3 Text_Mining(increases(expression)) CTD Tanespimycin TNFSF10 Text_Mining(affects(cotreatment)) CTD Tanespimycin TNFSF10 Text_Mining(decreases(expression)) CTD Tanespimycin TNFSF10 Text_Mining(increases(activity)) CTD Tanespimycin TP53 Text_Mining(decreases(expression)) CTD Tanespimycin TYMS Text_Mining(decreases(expression)) CTD Tanespimycin XIAP Text_Mining(affects(cotreatment)) CTD Tanespimycin XIAP Text_Mining(decreases(expression)) CTD Tanespimycin AR Potency-Replicate_1=0.1188(uM) D4 PubChem Tanespimycin AR AR Potency (uM)=0.118832(uM) D4 PubChem Tanespimycin AR Ratio Potency (uM)=0.230141(uM) D4 PubChem Tanespimycin AR Potency-Replicate_1=0.2391(uM) D4 PubChem Tanespimycin ESR1 ER Potency (uM)=0.195704(uM) D4 PubChem Tanespimycin ESR1 Potency-Replicate_1=0.2371(uM) D4 PubChem Tanespimycin GMNN Potency=0.0668(uM) D4 PubChem Tanespimycin HIF1A Inhibition=None(Unspecified) D4 ChEMBL Tanespimycin HSP90AA1 Activity=None(Unspecified) D4 ChEMBL Tanespimycin HSP90AA1 Inhibition=None(Unspecified) D4 ChEMBL Tanespimycin HSP90AB1 Activity=None(Unspecified) D4 ChEMBL Tanespimycin HSP90AB1 Inhibition=None(Unspecified) D4 ChEMBL Tanespimycin MTOR Potency=0.2524(uM) D4 PubChem Tanespimycin MTOR Potency=0.515(uM) D4 PubChem Tanespimycin NR3C1 None=None(uM) D4 PubChem Tanespimycin TDP1 Potency=0.3759(uM) D4 PubChem Tanespimycin TDP1 Potency=1.0593(uM) D4 PubChem