Drug Gene Type Source Deguelin ADM Text_Mining(decreases(reaction)) CTD Deguelin ADM Text_Mining(increases(expression)) CTD Deguelin AKT1 Text_Mining(decreases(reaction)) CTD Deguelin AKT1 Text_Mining(increases(activity)) CTD Deguelin AKT1 Text_Mining(increases(phosphorylation)) CTD Deguelin AKT1 Text_Mining(decreases(expression)) CTD Deguelin AKT1 Text_Mining(decreases(phosphorylation)) CTD Deguelin ANGPTL4 Text_Mining(decreases(reaction)) CTD Deguelin ANGPTL4 Text_Mining(increases(expression)) CTD Deguelin ATM Text_Mining(decreases(expression)) CTD Deguelin ATR Text_Mining(decreases(expression)) CTD Deguelin BCL2 Text_Mining(decreases(reaction)) CTD Deguelin BCL2 Text_Mining(increases(expression)) CTD Deguelin BCL2 Text_Mining(decreases(expression)) CTD Deguelin BCL2L1 Text_Mining(decreases(reaction)) CTD Deguelin BCL2L1 Text_Mining(increases(expression)) CTD Deguelin BCL2L1 Text_Mining(decreases(expression)) CTD Deguelin BIRC5 Text_Mining(decreases(reaction)) CTD Deguelin BIRC5 Text_Mining(increases(expression)) CTD Deguelin BIRC5 Text_Mining(decreases(expression)) CTD Deguelin BRCA1 Text_Mining(decreases(expression)) CTD Deguelin CA9 Text_Mining(decreases(reaction)) CTD Deguelin CA9 Text_Mining(increases(expression)) CTD Deguelin CASP3 Text_Mining(increases(activity)) CTD Deguelin CASP3 Text_Mining(increases(cleavage)) CTD Deguelin CASP7 Text_Mining(increases(expression)) CTD Deguelin CCND1 Text_Mining(decreases(expression)) CTD Deguelin CCND1 Text_Mining(decreases(reaction)) CTD Deguelin CCND1 Text_Mining(increases(expression)) CTD Deguelin CCND1 Text_Mining(increases(degradation)) CTD Deguelin CDH3 Text_Mining(increases(expression)) CTD Deguelin CDH7 Text_Mining(increases(expression)) CTD Deguelin CDH9 Text_Mining(increases(expression)) CTD Deguelin CDK4 Text_Mining(decreases(expression)) CTD Deguelin CDKN1A Text_Mining(decreases(expression)) CTD Deguelin CFLAR Text_Mining(decreases(reaction)) CTD Deguelin CFLAR Text_Mining(increases(expression)) CTD Deguelin CFLAR Text_Mining(decreases(expression)) CTD Deguelin CLDN2 Text_Mining(increases(expression)) CTD Deguelin CLDN5 Text_Mining(increases(expression)) CTD Deguelin CTNNB1 Text_Mining(decreases(expression)) CTD Deguelin CTNNB1 Text_Mining(decreases(reaction)) CTD Deguelin CTNNB1 Text_Mining(increases(degradation)) CTD Deguelin CXCL8 Text_Mining(decreases(reaction)) CTD Deguelin CXCL8 Text_Mining(increases(expression)) CTD Deguelin CXCR4 Text_Mining(decreases(reaction)) CTD Deguelin CXCR4 Text_Mining(increases(expression)) CTD Deguelin DKK2 Text_Mining(decreases(expression)) CTD Deguelin DKK4 Text_Mining(increases(expression)) CTD Deguelin EGFR Text_Mining(decreases(expression)) CTD Deguelin EGLN3 Text_Mining(decreases(reaction)) CTD Deguelin EGLN3 Text_Mining(increases(expression)) CTD Deguelin EIF4EBP1 Text_Mining(decreases(expression)) CTD Deguelin EPAS1 Text_Mining(decreases(expression)) CTD Deguelin FRZB Text_Mining(increases(expression)) CTD Deguelin FZD10 Text_Mining(increases(expression)) CTD Deguelin FZD4 Text_Mining(increases(expression)) CTD Deguelin FZD8 Text_Mining(increases(expression)) CTD Deguelin GSK3B Text_Mining(decreases(phosphorylation)) CTD Deguelin HIF1A Text_Mining(decreases(reaction)) CTD Deguelin HIF1A Text_Mining(increases(degradation)) CTD Deguelin HIF1A Text_Mining(increases(expression)) CTD Deguelin ICAM1 Text_Mining(decreases(reaction)) CTD Deguelin ICAM1 Text_Mining(increases(expression)) CTD Deguelin IGF1 Text_Mining(decreases(reaction)) CTD Deguelin IGF1 Text_Mining(increases(expression)) CTD Deguelin IGF1R Text_Mining(decreases(expression)) CTD Deguelin IHH Text_Mining(increases(expression)) CTD Deguelin IL10 Text_Mining(decreases(reaction)) CTD Deguelin IL10 Text_Mining(increases(expression)) CTD Deguelin KDR Text_Mining(decreases(expression)) CTD Deguelin LOX Text_Mining(decreases(reaction)) CTD Deguelin LOX Text_Mining(increases(expression)) CTD Deguelin MAP2K1 Text_Mining(decreases(expression)) CTD Deguelin MAP2K2 Text_Mining(decreases(expression)) CTD Deguelin MCL1 Text_Mining(decreases(expression)) CTD Deguelin MGMT Text_Mining(decreases(expression)) CTD Deguelin MKI67 Text_Mining(decreases(expression)) CTD Deguelin MMP9 Text_Mining(decreases(reaction)) CTD Deguelin MMP9 Text_Mining(increases(expression)) CTD Deguelin MTOR Text_Mining(decreases(expression)) CTD Deguelin MYC Text_Mining(decreases(expression)) CTD Deguelin MYC Text_Mining(decreases(reaction)) CTD Deguelin MYC Text_Mining(increases(expression)) CTD Deguelin MYC Text_Mining(increases(degradation)) CTD Deguelin NCOA3 Text_Mining(decreases(expression)) CTD Deguelin NFKBIA Text_Mining(decreases(reaction)) CTD Deguelin NFKBIA Text_Mining(increases(degradation)) CTD Deguelin NFKBIA Text_Mining(increases(phosphorylation)) CTD Deguelin NOS3 Text_Mining(decreases(expression)) CTD Deguelin NUP98 Text_Mining(decreases(expression)) CTD Deguelin ODC1 Text_Mining(increases(activity)) CTD Deguelin PARP1 Text_Mining(decreases(reaction)) CTD Deguelin PARP1 Text_Mining(increases(cleavage)) CTD Deguelin PARP1 Text_Mining(increases(expression)) CTD Deguelin PDK1 Text_Mining(decreases(expression)) CTD Deguelin PIK3CA Text_Mining(decreases(expression)) CTD Deguelin PRKDC Text_Mining(decreases(expression)) CTD Deguelin PTGS2 Text_Mining(decreases(reaction)) CTD Deguelin PTGS2 Text_Mining(increases(expression)) CTD Deguelin RB1 Text_Mining(decreases(expression)) CTD Deguelin RELA Text_Mining(affects(localization)) CTD Deguelin RELA Text_Mining(decreases(reaction)) CTD Deguelin RELA Text_Mining(increases(phosphorylation)) CTD Deguelin RELA Text_Mining(decreases(expression)) CTD Deguelin RELA Text_Mining(decreases(phosphorylation)) CTD Deguelin RPS6 Text_Mining(decreases(expression)) CTD Deguelin RPS6KB1 Text_Mining(decreases(expression)) CTD Deguelin SFRP2 Text_Mining(decreases(expression)) CTD Deguelin SNAI1 Text_Mining(decreases(expression)) CTD Deguelin SOX14 Text_Mining(increases(expression)) CTD Deguelin SOX30 Text_Mining(increases(expression)) CTD Deguelin SOX5 Text_Mining(increases(expression)) CTD Deguelin SRC Text_Mining(increases(activity)) CTD Deguelin STAT3 Text_Mining(increases(activity)) CTD Deguelin STAT6 Text_Mining(increases(phosphorylation)) CTD Deguelin STS Text_Mining(decreases(reaction)) CTD Deguelin STS Text_Mining(increases(activity)) CTD Deguelin TCF4 Text_Mining(increases(expression)) CTD Deguelin TNF Text_Mining(decreases(reaction)) CTD Deguelin TNF Text_Mining(increases(cleavage)) CTD Deguelin TNF Text_Mining(increases(expression)) CTD Deguelin TNF Text_Mining(affects(localization)) CTD Deguelin TNF Text_Mining(increases(phosphorylation)) CTD Deguelin TNF Text_Mining(increases(activity)) CTD Deguelin TNF Text_Mining(increases(degradation)) CTD Deguelin TP53 Text_Mining(decreases(expression)) CTD Deguelin VEGFA Text_Mining(decreases(reaction)) CTD Deguelin VEGFA Text_Mining(increases(expression)) CTD Deguelin VEGFA Text_Mining(decreases(expression)) CTD Deguelin VEGFA Text_Mining(decreases(response to substance)) CTD Deguelin WIF1 Text_Mining(increases(expression)) CTD Deguelin WNT10A Text_Mining(increases(expression)) CTD Deguelin WNT11 Text_Mining(increases(expression)) CTD Deguelin WNT9A Text_Mining(decreases(expression)) CTD Deguelin WNT2 Text_Mining(increases(expression)) CTD Deguelin WNT2B Text_Mining(decreases(expression)) CTD Deguelin WNT3A Text_Mining(decreases(expression)) CTD Deguelin XIAP Text_Mining(decreases(expression)) CTD Deguelin CYP1A2 None=None(uM) D4 PubChem Deguelin CYP2C19 Potency=5.0119(uM) D4 PubChem Deguelin CYP2C19 None=None(uM) D4 PubChem Deguelin CYP2C19 Potency=5011.9(nM) D4 ChEMBL Deguelin CYP2C19 AC50=5011.87(nM) D4 ChEMBL Deguelin CYP2D6 Potency=0.0631(uM) D4 PubChem Deguelin CYP2D6 None=None(uM) D4 PubChem Deguelin CYP2D6 AC50=63.1(nM) D4 ChEMBL Deguelin CYP2D6 Potency=63.1(nM) D4 ChEMBL Deguelin CYP3A4 Potency=15.8489(uM) D4 PubChem Deguelin CYP3A4 None=None(uM) D4 PubChem Deguelin CYP3A4 Potency=15848.9(nM) D4 ChEMBL Deguelin CYP3A4 AC50=15848.9(nM) D4 ChEMBL Deguelin MITF None=None(uM) D4 PubChem Deguelin TDP1 Potency=0.1059(uM) D4 PubChem Deguelin TDP1 Potency=0.1496(uM) D4 PubChem Deguelin TSHR Potency=19.9526(uM) D4 PubChem Deguelin TSHR Potency=19952.6(nM) D4 ChEMBL