Drug Gene Type Source Sitaxentan ABCB11 Text_Mining(decreases(activity)) CTD Sitaxentan CYP2C19 Text_Mining(decreases(reaction)) CTD Sitaxentan CYP2C19 Text_Mining(increases(metabolic processing)) CTD Sitaxentan CYP2C8 Text_Mining(decreases(reaction)) CTD Sitaxentan CYP2C8 Text_Mining(increases(metabolic processing)) CTD Sitaxentan CYP2C9 Text_Mining(decreases(reaction)) CTD Sitaxentan CYP2C9 Text_Mining(increases(metabolic processing)) CTD Sitaxentan CYP3A4 Text_Mining(decreases(activity)) CTD Sitaxentan EDNRA Text_Mining(affects(binding)) CTD Sitaxentan EDNRA Text_Mining(decreases(activity)) CTD Sitaxentan FN1 Text_Mining(decreases(reaction)) CTD Sitaxentan FN1 Text_Mining(increases(expression)) CTD Sitaxentan RELA Text_Mining(decreases(reaction)) CTD Sitaxentan RELA Text_Mining(increases(activity)) CTD Sitaxentan PPARG None=None(uM) D4 PubChem