Drug Gene Type Source Tegaserod CYP1A2 Text_Mining(decreases(activity)) CTD Tegaserod CYP2D6 Text_Mining(increases(metabolic processing)) CTD Tegaserod CYP2D6 Text_Mining(decreases(reaction)) CTD Tegaserod CYP2D6 Text_Mining(decreases(activity)) CTD Tegaserod HTR4 Text_Mining(affects(binding)) CTD Tegaserod HTR4 Text_Mining(increases(activity)) CTD Tegaserod HTR2B None=None(uM) D4 PubChem Tegaserod HTR4 None=None(uM) D4 PubChem Tegaserod VDR Potency-Replicate_1=13.4481(uM) D4 PubChem