Drug Gene Type Source MEPAZINE SLC22A2 Text_Mining(decreases(reaction)) CTD MEPAZINE SLC22A2 Text_Mining(increases(uptake)) CTD MEPAZINE ESR1 Potency-Replicate_1=18.9959(uM) D4 PubChem MEPAZINE ESR1 Ratio Potency (uM)=23.0141(uM) D4 PubChem