Drug Gene Type Source Imatinib ABCB1 Text_Mining(increases(expression)) CTD Imatinib ABCB1 Text_Mining(increases(activity)) CTD Imatinib ABCB11 Text_Mining(decreases(reaction)) CTD Imatinib ABCB11 Text_Mining(increases(transport)) CTD Imatinib ABCB11 Text_Mining(decreases(activity)) CTD Imatinib ABCC10 Text_Mining(decreases(abundance)) CTD Imatinib ABCC10 Text_Mining(decreases(reaction)) CTD Imatinib ABCC10 Text_Mining(increases(secretion)) CTD Imatinib ABCC10 Text_Mining(decreases(response to substance)) CTD Imatinib ABCG2 Text_Mining(increases(expression)) CTD Imatinib ABCG2 Text_Mining(increases(activity)) CTD Imatinib ABL1 Text_Mining(increases(response to substance)) CTD Imatinib ABL1 Text_Mining(decreases(response to substance)) CTD Imatinib ABL1 Text_Mining(affects(binding)) CTD Imatinib ABL1 Text_Mining(decreases(phosphorylation)) CTD Imatinib ABL1 Text_Mining(increases(reaction)) CTD Imatinib ABL1 Text_Mining(decreases(reaction)) CTD Imatinib ABL1 Text_Mining(increases(phosphorylation)) CTD Imatinib ABL1 Text_Mining(increases(activity)) CTD Imatinib ABL1 Text_Mining(increases(chemical synthesis)) CTD Imatinib ABL1 Text_Mining(increases(expression)) CTD Imatinib ABL1 Text_Mining(decreases(activity)) CTD Imatinib ABL1 Text_Mining(decreases(expression)) CTD Imatinib ABL1 Text_Mining(affects(cotreatment)) CTD Imatinib AICDA Text_Mining(decreases(expression)) CTD Imatinib AICDA Text_Mining(increases(reaction)) CTD Imatinib AKT1 Text_Mining(decreases(reaction)) CTD Imatinib AKT1 Text_Mining(increases(phosphorylation)) CTD Imatinib AKT1 Text_Mining(increases(reaction)) CTD Imatinib AKT1 Text_Mining(decreases(expression)) CTD Imatinib AKT1 Text_Mining(decreases(phosphorylation)) CTD Imatinib ALDH2 Text_Mining(affects(cotreatment)) CTD Imatinib ALDH2 Text_Mining(decreases(expression)) CTD Imatinib ALDOC Text_Mining(affects(cotreatment)) CTD Imatinib ALDOC Text_Mining(decreases(expression)) CTD Imatinib BAD Text_Mining(affects(cotreatment)) CTD Imatinib BAD Text_Mining(decreases(expression)) CTD Imatinib BAX Text_Mining(affects(cotreatment)) CTD Imatinib BAX Text_Mining(increases(expression)) CTD Imatinib BCL2 Text_Mining(affects(cotreatment)) CTD Imatinib BCL2 Text_Mining(decreases(expression)) CTD Imatinib BCL2L1 Text_Mining(decreases(expression)) CTD Imatinib BCL2L1 Text_Mining(affects(cotreatment)) CTD Imatinib BCL2L11 Text_Mining(increases(response to substance)) CTD Imatinib BCR Text_Mining(affects(binding)) CTD Imatinib BCR Text_Mining(decreases(phosphorylation)) CTD Imatinib BCR Text_Mining(increases(reaction)) CTD Imatinib BCR Text_Mining(decreases(reaction)) CTD Imatinib BCR Text_Mining(increases(chemical synthesis)) CTD Imatinib BCR Text_Mining(increases(expression)) CTD Imatinib BCR Text_Mining(decreases(activity)) CTD Imatinib BCR Text_Mining(decreases(expression)) CTD Imatinib BCR Text_Mining(affects(cotreatment)) CTD Imatinib BID Text_Mining(affects(cotreatment)) CTD Imatinib BID Text_Mining(increases(activity)) CTD Imatinib BIRC2 Text_Mining(affects(cotreatment)) CTD Imatinib BIRC2 Text_Mining(decreases(expression)) CTD Imatinib BIRC5 Text_Mining(decreases(response to substance)) CTD Imatinib BIRC5 Text_Mining(decreases(expression)) CTD Imatinib CASP3 Text_Mining(increases(activity)) CTD Imatinib CASP3 Text_Mining(increases(reaction)) CTD Imatinib CASP3 Text_Mining(affects(cotreatment)) CTD Imatinib CASP3 Text_Mining(increases(cleavage)) CTD Imatinib CASP8 Text_Mining(affects(cotreatment)) CTD Imatinib CASP8 Text_Mining(increases(activity)) CTD Imatinib CASP8 Text_Mining(increases(expression)) CTD Imatinib CBL Text_Mining(affects(cotreatment)) CTD Imatinib CBL Text_Mining(increases(expression)) CTD Imatinib CCL2 Text_Mining(affects(cotreatment)) CTD Imatinib CCL2 Text_Mining(decreases(reaction)) CTD Imatinib CCL2 Text_Mining(increases(secretion)) CTD Imatinib CCNA2 Text_Mining(affects(cotreatment)) CTD Imatinib CCNA2 Text_Mining(decreases(expression)) CTD Imatinib CCND3 Text_Mining(affects(cotreatment)) CTD Imatinib CCND3 Text_Mining(decreases(expression)) CTD Imatinib CDK1 Text_Mining(affects(cotreatment)) CTD Imatinib CDK1 Text_Mining(decreases(expression)) CTD Imatinib CDK2 Text_Mining(decreases(expression)) CTD Imatinib CDK4 Text_Mining(affects(cotreatment)) CTD Imatinib CDK4 Text_Mining(decreases(expression)) CTD Imatinib CDKN1B Text_Mining(affects(cotreatment)) CTD Imatinib CDKN1B Text_Mining(increases(expression)) CTD Imatinib CEBPB Text_Mining(increases(expression)) CTD Imatinib CFLAR Text_Mining(affects(cotreatment)) CTD Imatinib CFLAR Text_Mining(decreases(expression)) CTD Imatinib COL1A1 Text_Mining(decreases(reaction)) CTD Imatinib COL1A1 Text_Mining(increases(expression)) CTD Imatinib CRKL Text_Mining(decreases(reaction)) CTD Imatinib CRKL Text_Mining(increases(phosphorylation)) CTD Imatinib CRKL Text_Mining(decreases(phosphorylation)) CTD Imatinib CUL1 Text_Mining(affects(cotreatment)) CTD Imatinib CUL1 Text_Mining(increases(expression)) CTD Imatinib CXCL10 Text_Mining(affects(cotreatment)) CTD Imatinib CXCL10 Text_Mining(decreases(reaction)) CTD Imatinib CXCL10 Text_Mining(increases(secretion)) CTD Imatinib CXCL8 Text_Mining(affects(cotreatment)) CTD Imatinib CXCL8 Text_Mining(decreases(reaction)) CTD Imatinib CXCL8 Text_Mining(increases(expression)) CTD Imatinib CXCL8 Text_Mining(increases(secretion)) CTD Imatinib CXCL9 Text_Mining(affects(cotreatment)) CTD Imatinib CXCL9 Text_Mining(decreases(reaction)) CTD Imatinib CXCL9 Text_Mining(increases(secretion)) CTD Imatinib DEDD2 Text_Mining(affects(cotreatment)) CTD Imatinib DEDD2 Text_Mining(increases(expression)) CTD Imatinib DIABLO Text_Mining(affects(cotreatment)) CTD Imatinib DIABLO Text_Mining(increases(secretion)) CTD Imatinib DOK1 Text_Mining(decreases(phosphorylation)) CTD Imatinib EIF4B Text_Mining(decreases(expression)) CTD Imatinib EIF4E Text_Mining(decreases(expression)) CTD Imatinib EIF4EBP1 Text_Mining(decreases(expression)) CTD Imatinib EIF4EBP1 Text_Mining(increases(reaction)) CTD Imatinib FADD Text_Mining(affects(cotreatment)) CTD Imatinib FADD Text_Mining(increases(expression)) CTD Imatinib FBXO16 Text_Mining(affects(cotreatment)) CTD Imatinib FBXO16 Text_Mining(increases(expression)) CTD Imatinib FBXW4P1 Text_Mining(affects(cotreatment)) CTD Imatinib FBXW4P1 Text_Mining(increases(expression)) CTD Imatinib FGFR3 Text_Mining(decreases(expression)) CTD Imatinib GCK Text_Mining(affects(cotreatment)) CTD Imatinib GCK Text_Mining(decreases(expression)) CTD Imatinib H2AFX Text_Mining(increases(expression)) CTD Imatinib HDC Text_Mining(affects(binding)) CTD Imatinib HDC Text_Mining(decreases(reaction)) CTD Imatinib HDC Text_Mining(increases(expression)) CTD Imatinib HDC Text_Mining(decreases(expression)) CTD Imatinib HMOX1 Text_Mining(decreases(reaction)) CTD Imatinib HMOX1 Text_Mining(increases(expression)) CTD Imatinib HSF1 Text_Mining(increases(expression)) CTD Imatinib HSPB1 Text_Mining(increases(expression)) CTD Imatinib ICAM1 Text_Mining(increases(expression)) CTD Imatinib IFNG Text_Mining(affects(cotreatment)) CTD Imatinib IFNG Text_Mining(decreases(reaction)) CTD Imatinib IFNG Text_Mining(increases(expression)) CTD Imatinib IFNG Text_Mining(increases(phosphorylation)) CTD Imatinib IFNG Text_Mining(increases(secretion)) CTD Imatinib IGF1 Text_Mining(decreases(reaction)) CTD Imatinib IGF1 Text_Mining(increases(phosphorylation)) CTD Imatinib IGF1 Text_Mining(increases(reaction)) CTD Imatinib IGFBP4 Text_Mining(increases(expression)) CTD Imatinib IL1B Text_Mining(affects(cotreatment)) CTD Imatinib IL1B Text_Mining(decreases(reaction)) CTD Imatinib IL1B Text_Mining(increases(expression)) CTD Imatinib IL1B Text_Mining(increases(phosphorylation)) CTD Imatinib IL1B Text_Mining(increases(secretion)) CTD Imatinib IL4R Text_Mining(increases(expression)) CTD Imatinib JUN Text_Mining(affects(cotreatment)) CTD Imatinib JUN Text_Mining(increases(activity)) CTD Imatinib KIT Text_Mining(decreases(reaction)) CTD Imatinib KIT Text_Mining(increases(expression)) CTD Imatinib KRT14 Text_Mining(increases(expression)) CTD Imatinib KRT5 Text_Mining(increases(expression)) CTD Imatinib LCK Text_Mining(decreases(phosphorylation)) CTD Imatinib LYN Text_Mining(decreases(response to substance)) CTD Imatinib LYN Text_Mining(affects(cotreatment)) CTD Imatinib LYN Text_Mining(decreases(phosphorylation)) CTD Imatinib MAPK1 Text_Mining(decreases(reaction)) CTD Imatinib MAPK1 Text_Mining(increases(activity)) CTD Imatinib MAPK1 Text_Mining(increases(phosphorylation)) CTD Imatinib MAPK1 Text_Mining(decreases(phosphorylation)) CTD Imatinib MAPK3 Text_Mining(decreases(reaction)) CTD Imatinib MAPK3 Text_Mining(increases(activity)) CTD Imatinib MAPK3 Text_Mining(increases(phosphorylation)) CTD Imatinib MAPK3 Text_Mining(decreases(phosphorylation)) CTD Imatinib MCL1 Text_Mining(affects(cotreatment)) CTD Imatinib MCL1 Text_Mining(decreases(expression)) CTD Imatinib MTOR Text_Mining(decreases(reaction)) CTD Imatinib MTOR Text_Mining(increases(phosphorylation)) CTD Imatinib MTOR Text_Mining(increases(reaction)) CTD Imatinib MTOR Text_Mining(decreases(expression)) CTD Imatinib NAB2 Text_Mining(increases(expression)) CTD Imatinib NFKB1 Text_Mining(affects(binding)) CTD Imatinib NFKB1 Text_Mining(decreases(activity)) CTD Imatinib NFKBIA Text_Mining(affects(cotreatment)) CTD Imatinib NFKBIA Text_Mining(decreases(reaction)) CTD Imatinib NFKBIA Text_Mining(increases(phosphorylation)) CTD Imatinib ODC1 Text_Mining(increases(expression)) CTD Imatinib PDGFB Text_Mining(decreases(expression)) CTD Imatinib PDGFRA Text_Mining(decreases(expression)) CTD Imatinib PDGFRA Text_Mining(increases(reaction)) CTD Imatinib PDGFRB Text_Mining(decreases(expression)) CTD Imatinib PDGFRB Text_Mining(decreases(phosphorylation)) CTD Imatinib PDHB Text_Mining(affects(cotreatment)) CTD Imatinib PDHB Text_Mining(decreases(expression)) CTD Imatinib PIK3R1 Text_Mining(decreases(expression)) CTD Imatinib PPARG Text_Mining(decreases(activity)) CTD Imatinib PPARG Text_Mining(decreases(reaction)) CTD Imatinib PPARG Text_Mining(increases(phosphorylation)) CTD Imatinib PPP2CA Text_Mining(increases(expression)) CTD Imatinib PRKCD Text_Mining(decreases(reaction)) CTD Imatinib PRKCD Text_Mining(increases(activity)) CTD Imatinib PRKCD Text_Mining(increases(phosphorylation)) CTD Imatinib PTEN Text_Mining(increases(reaction)) CTD Imatinib PTEN Text_Mining(increases(response to substance)) CTD Imatinib PTGS2 Text_Mining(decreases(expression)) CTD Imatinib PTGS2 Text_Mining(increases(reaction)) CTD Imatinib RB1 Text_Mining(decreases(expression)) CTD Imatinib RB1 Text_Mining(decreases(phosphorylation)) CTD Imatinib RELA Text_Mining(affects(binding)) CTD Imatinib RELA Text_Mining(decreases(activity)) CTD Imatinib RELA Text_Mining(increases(methylation)) CTD Imatinib RELA Text_Mining(increases(phosphorylation)) CTD Imatinib RET Text_Mining(decreases(phosphorylation)) CTD Imatinib RPS6 Text_Mining(affects(cotreatment)) CTD Imatinib RPS6 Text_Mining(decreases(phosphorylation)) CTD Imatinib RPS6KB1 Text_Mining(decreases(expression)) CTD Imatinib SLC22A2 Text_Mining(decreases(reaction)) CTD Imatinib SLC22A2 Text_Mining(increases(uptake)) CTD Imatinib SOX17 Text_Mining(decreases(localization)) CTD Imatinib STAT1 Text_Mining(affects(cotreatment)) CTD Imatinib STAT1 Text_Mining(decreases(reaction)) CTD Imatinib STAT1 Text_Mining(increases(phosphorylation)) CTD Imatinib STAT5A Text_Mining(affects(cotreatment)) CTD Imatinib STAT5A Text_Mining(decreases(phosphorylation)) CTD Imatinib TANK Text_Mining(increases(expression)) CTD Imatinib TNF Text_Mining(decreases(reaction)) CTD Imatinib TNF Text_Mining(increases(secretion)) CTD Imatinib TNFRSF10B Text_Mining(increases(expression)) CTD Imatinib TNFRSF1B Text_Mining(affects(cotreatment)) CTD Imatinib TNFRSF1B Text_Mining(decreases(expression)) CTD Imatinib VEGFA Text_Mining(decreases(secretion)) CTD Imatinib VEGFA Text_Mining(affects(cotreatment)) CTD Imatinib WT1 Text_Mining(decreases(expression)) CTD Imatinib ABL1 None=8.5(uM) D4 PubChem Imatinib ABL1 Inhibition=None(Unspecified) D4 ChEMBL Imatinib ABL2 None=10.0(uM) D4 PubChem Imatinib BCR Inhibition=None(Unspecified) D4 ChEMBL Imatinib DDR1 None=0.7(uM) D4 PubChem Imatinib EYA2 Potency=9.53(uM) D4 PubChem Imatinib NQO2 Activity=None(Unspecified) D4 ChEMBL Imatinib SFN Inhibition=None(Unspecified) D4 ChEMBL Imatinib SMAD3 Potency=12.5893(uM) D4 PubChem Imatinib TDP1 Potency=11.2202(uM) D4 PubChem Imatinib TDP1 Potency=17.7828(uM) D4 PubChem Imatinib YES1 Potency=27.4038(uM) D4 PubChem