Drug Gene Type Source Bexarotene ADD3 Text_Mining(increases(expression)) CTD Bexarotene ADIRF Text_Mining(increases(expression)) CTD Bexarotene ADRB2 Text_Mining(decreases(expression)) CTD Bexarotene AKR1C1 Text_Mining(increases(expression)) CTD Bexarotene AKR1C3 Text_Mining(increases(expression)) CTD Bexarotene AMOTL2 Text_Mining(decreases(expression)) CTD Bexarotene ARL6IP5 Text_Mining(increases(expression)) CTD Bexarotene ASNS Text_Mining(decreases(expression)) CTD Bexarotene ATM Text_Mining(increases(activity)) CTD Bexarotene BAX Text_Mining(increases(activity)) CTD Bexarotene BAX Text_Mining(increases(expression)) CTD Bexarotene BIRC5 Text_Mining(decreases(expression)) CTD Bexarotene BNIP2 Text_Mining(decreases(expression)) CTD Bexarotene C10ORF10 Text_Mining(increases(expression)) CTD Bexarotene CCNB1 Text_Mining(decreases(expression)) CTD Bexarotene CDK1 Text_Mining(decreases(expression)) CTD Bexarotene CDKN1A Text_Mining(increases(expression)) CTD Bexarotene CEBPG Text_Mining(decreases(expression)) CTD Bexarotene COX2 Text_Mining(decreases(expression)) CTD Bexarotene CTH Text_Mining(decreases(expression)) CTD Bexarotene CTSH Text_Mining(increases(expression)) CTD Bexarotene CYCS Text_Mining(decreases(expression)) CTD Bexarotene CYP26A1 Text_Mining(increases(expression)) CTD Bexarotene CYR61 Text_Mining(decreases(expression)) CTD Bexarotene DDIT4 Text_Mining(increases(expression)) CTD Bexarotene DHRS3 Text_Mining(increases(expression)) CTD Bexarotene DKK1 Text_Mining(increases(expression)) CTD Bexarotene DUSP1 Text_Mining(decreases(expression)) CTD Bexarotene DUSP5 Text_Mining(decreases(expression)) CTD Bexarotene EGR3 Text_Mining(decreases(expression)) CTD Bexarotene EIF1 Text_Mining(decreases(expression)) CTD Bexarotene EPHA2 Text_Mining(decreases(expression)) CTD Bexarotene GARS Text_Mining(decreases(expression)) CTD Bexarotene GPM6B Text_Mining(increases(expression)) CTD Bexarotene HERPUD1 Text_Mining(decreases(expression)) CTD Bexarotene ID1 Text_Mining(increases(expression)) CTD Bexarotene IER2 Text_Mining(decreases(expression)) CTD Bexarotene IGFBP6 Text_Mining(increases(expression)) CTD Bexarotene IL15 Text_Mining(increases(expression)) CTD Bexarotene IL4 Text_Mining(decreases(expression)) CTD Bexarotene ITGB6 Text_Mining(increases(expression)) CTD Bexarotene ITM2A Text_Mining(increases(expression)) CTD Bexarotene ITPR1 Text_Mining(increases(expression)) CTD Bexarotene KLF10 Text_Mining(decreases(expression)) CTD Bexarotene KRT15 Text_Mining(increases(expression)) CTD Bexarotene KRT17 Text_Mining(decreases(expression)) CTD Bexarotene LOXL2 Text_Mining(increases(expression)) CTD Bexarotene MAF Text_Mining(increases(expression)) CTD Bexarotene MAFF Text_Mining(decreases(expression)) CTD Bexarotene MLLT11 Text_Mining(increases(expression)) CTD Bexarotene MMP1 Text_Mining(decreases(expression)) CTD Bexarotene MTHFD2 Text_Mining(decreases(expression)) CTD Bexarotene ODC1 Text_Mining(decreases(expression)) CTD Bexarotene PER2 Text_Mining(decreases(expression)) CTD Bexarotene PIK3R1 Text_Mining(increases(expression)) CTD Bexarotene PIK3R1 Text_Mining(increases(reaction)) CTD Bexarotene PLAT Text_Mining(increases(expression)) CTD Bexarotene PLAUR Text_Mining(decreases(expression)) CTD Bexarotene PLOD2 Text_Mining(increases(expression)) CTD Bexarotene PNO1 Text_Mining(decreases(expression)) CTD Bexarotene PNRC1 Text_Mining(increases(expression)) CTD Bexarotene RARB Text_Mining(increases(expression)) CTD Bexarotene RB1 Text_Mining(decreases(phosphorylation)) CTD Bexarotene RXRA Text_Mining(affects(binding)) CTD Bexarotene RXRA Text_Mining(increases(activity)) CTD Bexarotene RXRB Text_Mining(affects(binding)) CTD Bexarotene RXRG Text_Mining(affects(binding)) CTD Bexarotene S100A9 Text_Mining(increases(expression)) CTD Bexarotene SCD Text_Mining(increases(expression)) CTD Bexarotene SIAH2 Text_Mining(decreases(expression)) CTD Bexarotene SLC2A4 Text_Mining(affects(cotreatment)) CTD Bexarotene SLC2A4 Text_Mining(increases(expression)) CTD Bexarotene SLC7A1 Text_Mining(decreases(expression)) CTD Bexarotene SLC7A5 Text_Mining(decreases(expression)) CTD Bexarotene SMAD5 Text_Mining(increases(expression)) CTD Bexarotene SPARC Text_Mining(increases(expression)) CTD Bexarotene SRSF2 Text_Mining(decreases(expression)) CTD Bexarotene TGM2 Text_Mining(increases(expression)) CTD Bexarotene TM4SF1 Text_Mining(increases(expression)) CTD Bexarotene TP53 Text_Mining(increases(activity)) CTD Bexarotene TP53 Text_Mining(increases(phosphorylation)) CTD Bexarotene TP73 Text_Mining(increases(expression)) CTD Bexarotene TSC22D3 Text_Mining(increases(expression)) CTD Bexarotene UAP1 Text_Mining(decreases(expression)) CTD Bexarotene UCP2 Text_Mining(increases(expression)) CTD Bexarotene UCP2 Text_Mining(increases(reaction)) CTD Bexarotene VAMP8 Text_Mining(increases(expression)) CTD Bexarotene XBP1 Text_Mining(decreases(expression)) CTD Bexarotene BLM Potency=68.0496(uM) D4 PubChem Bexarotene BLM Potency=68049.6(nM) D4 ChEMBL Bexarotene CYP19A1 Potency-Replicate_1=61.1306(uM) D4 PubChem Bexarotene ESR1 Potency-Replicate_1=3.7578(uM) D4 PubChem Bexarotene ESR1 Ratio Potency (uM)=10.9622(uM) D4 PubChem Bexarotene ESR1 Potency-Replicate_1=17.3739(uM) D4 PubChem Bexarotene ESR1 ER Potency (uM)=18.8336(uM) D4 PubChem Bexarotene HSPB1 Ratio Potency (uM)=21.13(uM) D4 PubChem Bexarotene KAT2A Potency=6.3096(uM) D4 PubChem Bexarotene KAT2A Potency=6309.6(nM) D4 ChEMBL Bexarotene NR1H3 Activity=None(Unspecified) D4 ChEMBL Bexarotene NR3C1 Potency-Replicate_1=9.77(uM) D4 PubChem Bexarotene PPARG Ratio Potency (uM)=None(uM) D4 PubChem Bexarotene RXRA Activity=None(Unspecified) D4 ChEMBL Bexarotene USP1 Potency=22.3872(uM) D4 PubChem