Drug Gene Type Source SB 202190 ATF2 Text_Mining(decreases(reaction)) CTD SB 202190 ATF2 Text_Mining(increases(phosphorylation)) CTD SB 202190 ATF2 Text_Mining(decreases(response to substance)) CTD SB 202190 ATF2 Text_Mining(increases(activity)) CTD SB 202190 ATF2 Text_Mining(affects(phosphorylation)) CTD SB 202190 BAX Text_Mining(affects(localization)) CTD SB 202190 BAX Text_Mining(decreases(reaction)) CTD SB 202190 BCL2 Text_Mining(decreases(expression)) CTD SB 202190 BCL2 Text_Mining(decreases(reaction)) CTD SB 202190 BCL2L1 Text_Mining(decreases(expression)) CTD SB 202190 BCL2L1 Text_Mining(decreases(reaction)) CTD SB 202190 BIRC5 Text_Mining(decreases(expression)) CTD SB 202190 BIRC5 Text_Mining(decreases(reaction)) CTD SB 202190 CASP3 Text_Mining(decreases(reaction)) CTD SB 202190 CASP3 Text_Mining(increases(activity)) CTD SB 202190 CCL11 Text_Mining(decreases(reaction)) CTD SB 202190 CCL11 Text_Mining(increases(expression)) CTD SB 202190 CCL2 Text_Mining(decreases(reaction)) CTD SB 202190 CCL2 Text_Mining(increases(expression)) CTD SB 202190 CCL26 Text_Mining(decreases(reaction)) CTD SB 202190 CCL26 Text_Mining(increases(expression)) CTD SB 202190 CCNB1 Text_Mining(decreases(reaction)) CTD SB 202190 CCNB1 Text_Mining(increases(degradation)) CTD SB 202190 CCNB1 Text_Mining(increases(ubiquitination)) CTD SB 202190 CCNB1 Text_Mining(increases(expression)) CTD SB 202190 CCND3 Text_Mining(decreases(reaction)) CTD SB 202190 CCND3 Text_Mining(increases(expression)) CTD SB 202190 CCND3 Text_Mining(increases(reaction)) CTD SB 202190 CCR2 Text_Mining(decreases(expression)) CTD SB 202190 CCR2 Text_Mining(decreases(reaction)) CTD SB 202190 CD14 Text_Mining(increases(expression)) CTD SB 202190 CD14 Text_Mining(increases(reaction)) CTD SB 202190 CDC20 Text_Mining(affects(binding)) CTD SB 202190 CDC20 Text_Mining(decreases(reaction)) CTD SB 202190 CDC20 Text_Mining(increases(reaction)) CTD SB 202190 CDC20 Text_Mining(decreases(expression)) CTD SB 202190 CDC27 Text_Mining(affects(binding)) CTD SB 202190 CDC27 Text_Mining(decreases(reaction)) CTD SB 202190 CDC27 Text_Mining(increases(reaction)) CTD SB 202190 CDK1 Text_Mining(decreases(activity)) CTD SB 202190 CDK1 Text_Mining(decreases(reaction)) CTD SB 202190 CDKN1A Text_Mining(decreases(reaction)) CTD SB 202190 CDKN1A Text_Mining(increases(expression)) CTD SB 202190 CEBPB Text_Mining(increases(expression)) CTD SB 202190 CEBPB Text_Mining(increases(reaction)) CTD SB 202190 CHRNA5 Text_Mining(decreases(reaction)) CTD SB 202190 CHRNA5 Text_Mining(increases(expression)) CTD SB 202190 CHRNA7 Text_Mining(decreases(reaction)) CTD SB 202190 CHRNA7 Text_Mining(increases(expression)) CTD SB 202190 CREB1 Text_Mining(decreases(reaction)) CTD SB 202190 CREB1 Text_Mining(increases(phosphorylation)) CTD SB 202190 CXCL8 Text_Mining(decreases(reaction)) CTD SB 202190 CXCL8 Text_Mining(increases(secretion)) CTD SB 202190 CXCL8 Text_Mining(increases(expression)) CTD SB 202190 CXCL8 Text_Mining(increases(reaction)) CTD SB 202190 CYP1A1 Text_Mining(decreases(reaction)) CTD SB 202190 CYP1A1 Text_Mining(increases(expression)) CTD SB 202190 FAS Text_Mining(decreases(reaction)) CTD SB 202190 FAS Text_Mining(increases(expression)) CTD SB 202190 FASLG Text_Mining(decreases(reaction)) CTD SB 202190 FASLG Text_Mining(increases(expression)) CTD SB 202190 FGF9 Text_Mining(decreases(reaction)) CTD SB 202190 FGF9 Text_Mining(increases(expression)) CTD SB 202190 FOS Text_Mining(affects(cotreatment)) CTD SB 202190 FOS Text_Mining(affects(localization)) CTD SB 202190 FOS Text_Mining(decreases(reaction)) CTD SB 202190 FOS Text_Mining(increases(expression)) CTD SB 202190 FOS Text_Mining(increases(reaction)) CTD SB 202190 GDF15 Text_Mining(decreases(reaction)) CTD SB 202190 GDF15 Text_Mining(increases(expression)) CTD SB 202190 HIF1A Text_Mining(decreases(reaction)) CTD SB 202190 HIF1A Text_Mining(increases(expression)) CTD SB 202190 HMOX1 Text_Mining(decreases(reaction)) CTD SB 202190 HMOX1 Text_Mining(increases(expression)) CTD SB 202190 ICAM1 Text_Mining(decreases(reaction)) CTD SB 202190 ICAM1 Text_Mining(increases(expression)) CTD SB 202190 IFNG Text_Mining(decreases(reaction)) CTD SB 202190 IFNG Text_Mining(increases(expression)) CTD SB 202190 IL10 Text_Mining(decreases(reaction)) CTD SB 202190 IL10 Text_Mining(increases(reaction)) CTD SB 202190 IL10 Text_Mining(increases(secretion)) CTD SB 202190 IL1A Text_Mining(decreases(reaction)) CTD SB 202190 IL1A Text_Mining(increases(expression)) CTD SB 202190 IL1B Text_Mining(decreases(reaction)) CTD SB 202190 IL1B Text_Mining(increases(secretion)) CTD SB 202190 IL1B Text_Mining(increases(reaction)) CTD SB 202190 IL1B Text_Mining(increases(expression)) CTD SB 202190 IL2 Text_Mining(decreases(reaction)) CTD SB 202190 IL2 Text_Mining(increases(expression)) CTD SB 202190 IL4 Text_Mining(decreases(reaction)) CTD SB 202190 IL4 Text_Mining(increases(expression)) CTD SB 202190 IL6 Text_Mining(decreases(reaction)) CTD SB 202190 IL6 Text_Mining(increases(expression)) CTD SB 202190 IL6 Text_Mining(increases(secretion)) CTD SB 202190 IL6 Text_Mining(decreases(activity)) CTD SB 202190 ITGAM Text_Mining(decreases(reaction)) CTD SB 202190 ITGAM Text_Mining(increases(expression)) CTD SB 202190 ITGAM Text_Mining(increases(reaction)) CTD SB 202190 ITGB6 Text_Mining(decreases(reaction)) CTD SB 202190 ITGB6 Text_Mining(increases(expression)) CTD SB 202190 JUN Text_Mining(affects(cotreatment)) CTD SB 202190 JUN Text_Mining(affects(localization)) CTD SB 202190 JUN Text_Mining(decreases(reaction)) CTD SB 202190 JUN Text_Mining(increases(phosphorylation)) CTD SB 202190 KLK3 Text_Mining(decreases(reaction)) CTD SB 202190 KLK3 Text_Mining(increases(expression)) CTD SB 202190 MAD2L1 Text_Mining(affects(binding)) CTD SB 202190 MAD2L1 Text_Mining(decreases(reaction)) CTD SB 202190 MAD2L1 Text_Mining(increases(reaction)) CTD SB 202190 MAPK1 Text_Mining(increases(activity)) CTD SB 202190 MAPK1 Text_Mining(increases(phosphorylation)) CTD SB 202190 MAPK1 Text_Mining(increases(reaction)) CTD SB 202190 MAPK14 Text_Mining(decreases(activity)) CTD SB 202190 MAPK3 Text_Mining(increases(activity)) CTD SB 202190 MAPK3 Text_Mining(increases(phosphorylation)) CTD SB 202190 MAPK3 Text_Mining(increases(reaction)) CTD SB 202190 MAPK8 Text_Mining(decreases(reaction)) CTD SB 202190 MAPK8 Text_Mining(increases(phosphorylation)) CTD SB 202190 MAPK9 Text_Mining(decreases(reaction)) CTD SB 202190 MAPK9 Text_Mining(increases(phosphorylation)) CTD SB 202190 MMP9 Text_Mining(decreases(reaction)) CTD SB 202190 MMP9 Text_Mining(increases(secretion)) CTD SB 202190 MMP9 Text_Mining(increases(activity)) CTD SB 202190 NGFR Text_Mining(decreases(reaction)) CTD SB 202190 NGFR Text_Mining(increases(expression)) CTD SB 202190 NOD1 Text_Mining(decreases(reaction)) CTD SB 202190 NOD1 Text_Mining(increases(secretion)) CTD SB 202190 PLAT Text_Mining(affects(binding)) CTD SB 202190 PLAT Text_Mining(decreases(reaction)) CTD SB 202190 PLAT Text_Mining(increases(reaction)) CTD SB 202190 PLAT Text_Mining(increases(expression)) CTD SB 202190 PLAT Text_Mining(increases(secretion)) CTD SB 202190 PLAU Text_Mining(decreases(reaction)) CTD SB 202190 PLAU Text_Mining(increases(expression)) CTD SB 202190 PTGS2 Text_Mining(decreases(reaction)) CTD SB 202190 PTGS2 Text_Mining(increases(expression)) CTD SB 202190 RB1 Text_Mining(increases(expression)) CTD SB 202190 RB1 Text_Mining(increases(reaction)) CTD SB 202190 SP1 Text_Mining(affects(binding)) CTD SB 202190 SP1 Text_Mining(decreases(reaction)) CTD SB 202190 SP1 Text_Mining(increases(reaction)) CTD SB 202190 TERT Text_Mining(affects(cotreatment)) CTD SB 202190 TERT Text_Mining(decreases(reaction)) CTD SB 202190 TERT Text_Mining(increases(expression)) CTD SB 202190 TGFA Text_Mining(decreases(reaction)) CTD SB 202190 TGFA Text_Mining(increases(secretion)) CTD SB 202190 TGFB1 Text_Mining(decreases(reaction)) CTD SB 202190 TGFB1 Text_Mining(increases(expression)) CTD SB 202190 TNF Text_Mining(decreases(reaction)) CTD SB 202190 TNF Text_Mining(increases(secretion)) CTD SB 202190 TP53 Text_Mining(decreases(reaction)) CTD SB 202190 TP53 Text_Mining(increases(expression)) CTD SB 202190 TP53 Text_Mining(increases(phosphorylation)) CTD SB 202190 TPP2 Text_Mining(affects(localization)) CTD SB 202190 TPP2 Text_Mining(decreases(reaction)) CTD SB 202190 VEGFA Text_Mining(decreases(reaction)) CTD SB 202190 VEGFA Text_Mining(increases(expression)) CTD SB 202190 CBX1 Potency=56.2341(uM) D4 PubChem SB 202190 CBX1 Potency=56234.1(nM) D4 ChEMBL SB 202190 CSNK1E Inhibition=None(Unspecified) D4 ChEMBL SB 202190 CYP1A2 None=None(uM) D4 PubChem SB 202190 CYP1A2 AC50=15848.9(nM) D4 ChEMBL SB 202190 CYP2C19 Potency=0.7943(uM) D4 PubChem SB 202190 CYP2C19 Potency=794.3(nM) D4 ChEMBL SB 202190 CYP2C9 Potency=7.9433(uM) D4 PubChem SB 202190 CYP2C9 Potency=7943.3(nM) D4 ChEMBL SB 202190 CYP2D6 Potency=5.0119(uM) D4 PubChem SB 202190 CYP2D6 Potency=12.5893(uM) D4 PubChem SB 202190 CYP2D6 None=None(uM) D4 PubChem SB 202190 CYP2D6 AC50=5011.87(nM) D4 ChEMBL SB 202190 CYP2D6 Potency=5011.9(nM) D4 ChEMBL SB 202190 CYP2D6 Potency=12589.3(nM) D4 ChEMBL SB 202190 CYP3A4 Potency=1.0(uM) D4 PubChem SB 202190 CYP3A4 None=None(uM) D4 PubChem SB 202190 CYP3A4 AC50=501.19(nM) D4 ChEMBL SB 202190 CYP3A4 Potency=1000.0(nM) D4 ChEMBL SB 202190 EGFR Inhibition=None(Unspecified) D4 ChEMBL SB 202190 EHMT2 Potency=12.5893(uM) D4 PubChem SB 202190 EHMT2 Potency=12589.3(nM) D4 ChEMBL SB 202190 FRK Inhibition=None(Unspecified) D4 ChEMBL SB 202190 GAK Inhibition=None(Unspecified) D4 ChEMBL SB 202190 GMNN Potency=3.5481(uM) D4 PubChem SB 202190 HSD17B10 Potency=31622.8(nM) D4 ChEMBL SB 202190 MAPK1 Potency=7.9433(uM) D4 PubChem SB 202190 MAPK1 Potency=7943.3(nM) D4 ChEMBL SB 202190 MAPK10 Inhibition=None(Unspecified) D4 ChEMBL SB 202190 MAPK11 Inhibition=None(Unspecified) D4 ChEMBL SB 202190 MAPK12 Inhibition=None(Unspecified) D4 ChEMBL SB 202190 MAPK14 None=9.8(uM) D4 PubChem SB 202190 MAPK14 Inhibition=None(Unspecified) D4 ChEMBL SB 202190 MAPK8 Inhibition=None(Unspecified) D4 ChEMBL SB 202190 MAPK9 Inhibition=None(Unspecified) D4 ChEMBL SB 202190 MDM2 None=None(uM) D4 PubChem SB 202190 MDM4 None=None(uM) D4 PubChem SB 202190 MPHOSPH8 Potency=31.6228(uM) D4 PubChem SB 202190 MPHOSPH8 Potency=31622.8(nM) D4 ChEMBL SB 202190 PTK6 Inhibition=None(Unspecified) D4 ChEMBL SB 202190 RIPK2 Inhibition=None(Unspecified) D4 ChEMBL SB 202190 STK36 Inhibition=None(Unspecified) D4 ChEMBL SB 202190 TDP1 Potency=6.5131(uM) D4 PubChem SB 202190 TDP1 Potency=15.0672(uM) D4 PubChem SB 202190 TNIK Inhibition=None(Unspecified) D4 ChEMBL SB 202190 TNNC1 None=None(uM) D4 PubChem SB 202190 TNNI3 None=None(uM) D4 PubChem SB 202190 TNNT2 None=None(uM) D4 PubChem SB 202190 YES1 Potency=17.2906(uM) D4 PubChem