Drug Gene Type Source clobenpropit ADRB2 Text_Mining(increases(activity)) CTD clobenpropit ADRB2 Text_Mining(increases(reaction)) CTD clobenpropit CCL2 Text_Mining(decreases(expression)) CTD clobenpropit CCND1 Text_Mining(decreases(expression)) CTD clobenpropit CCND1 Text_Mining(increases(response to substance)) CTD clobenpropit CDK2 Text_Mining(decreases(expression)) CTD clobenpropit CDK2 Text_Mining(increases(response to substance)) CTD clobenpropit CDKN1A Text_Mining(increases(expression)) CTD clobenpropit CDKN1A Text_Mining(increases(response to substance)) CTD clobenpropit CDKN1B Text_Mining(increases(expression)) CTD clobenpropit CDKN1B Text_Mining(increases(response to substance)) CTD clobenpropit HRH2 Text_Mining(increases(expression)) CTD clobenpropit HRH2 Text_Mining(increases(reaction)) CTD clobenpropit HRH3 Text_Mining(affects(binding)) CTD clobenpropit HRH3 Text_Mining(decreases(activity)) CTD clobenpropit HRH4 Text_Mining(affects(binding)) CTD clobenpropit HRH4 Text_Mining(decreases(reaction)) CTD clobenpropit HRH4 Text_Mining(increases(abundance)) CTD clobenpropit HRH4 Text_Mining(increases(activity)) CTD clobenpropit HRH4 Text_Mining(increases(response to substance)) CTD clobenpropit HRH4 Text_Mining(decreases(expression)) CTD clobenpropit HRH4 Text_Mining(increases(expression)) CTD clobenpropit IFNG Text_Mining(affects(expression)) CTD clobenpropit IL16 Text_Mining(increases(expression)) CTD clobenpropit IL16 Text_Mining(increases(reaction)) CTD clobenpropit IL5 Text_Mining(affects(expression)) CTD clobenpropit SLC22A3 Text_Mining(decreases(reaction)) CTD clobenpropit SLC22A3 Text_Mining(increases(uptake)) CTD clobenpropit CYP1A2 None=None(uM) D4 PubChem clobenpropit CYP1A2 AC50=15848.9(nM) D4 ChEMBL clobenpropit CYP2C19 Potency=15.8489(uM) D4 PubChem clobenpropit CYP2C19 None=None(uM) D4 PubChem clobenpropit CYP2C19 Potency=15848.9(nM) D4 ChEMBL clobenpropit CYP2C19 AC50=15848.9(nM) D4 ChEMBL clobenpropit CYP2C9 Potency=12.5893(uM) D4 PubChem clobenpropit CYP2C9 None=None(uM) D4 PubChem clobenpropit CYP2C9 AC50=12589.2(nM) D4 ChEMBL clobenpropit CYP2C9 Potency=12589.3(nM) D4 ChEMBL clobenpropit CYP2D6 Potency=12.5893(uM) D4 PubChem clobenpropit CYP2D6 None=None(uM) D4 PubChem clobenpropit CYP2D6 Potency=12589.3(nM) D4 ChEMBL clobenpropit CYP2D6 AC50=12589.2(nM) D4 ChEMBL clobenpropit CYP3A4 Potency=1.5849(uM) D4 PubChem clobenpropit CYP3A4 None=None(uM) D4 PubChem clobenpropit CYP3A4 AC50=1584.89(nM) D4 ChEMBL clobenpropit CYP3A4 Potency=1584.9(nM) D4 ChEMBL clobenpropit TDP1 Potency=21.136(uM) D4 PubChem