Drug Gene Type Source rottlerin ABL1 Text_Mining(decreases(activity)) CTD rottlerin ABL1 Text_Mining(decreases(reaction)) CTD rottlerin ABL1 Text_Mining(increases(expression)) CTD rottlerin ABL1 Text_Mining(increases(phosphorylation)) CTD rottlerin AKT1 Text_Mining(decreases(reaction)) CTD rottlerin AKT1 Text_Mining(increases(activity)) CTD rottlerin AKT1 Text_Mining(increases(phosphorylation)) CTD rottlerin AKT1 Text_Mining(decreases(phosphorylation)) CTD rottlerin ATG7 Text_Mining(decreases(reaction)) CTD rottlerin ATG7 Text_Mining(increases(expression)) CTD rottlerin BAK1 Text_Mining(decreases(reaction)) CTD rottlerin BAK1 Text_Mining(increases(activity)) CTD rottlerin BAX Text_Mining(increases(expression)) CTD rottlerin BCL2 Text_Mining(decreases(expression)) CTD rottlerin BCL2L1 Text_Mining(decreases(expression)) CTD rottlerin BECN1 Text_Mining(decreases(reaction)) CTD rottlerin BECN1 Text_Mining(increases(expression)) CTD rottlerin BIRC3 Text_Mining(decreases(reaction)) CTD rottlerin BIRC3 Text_Mining(increases(expression)) CTD rottlerin CASP3 Text_Mining(decreases(reaction)) CTD rottlerin CASP3 Text_Mining(increases(activity)) CTD rottlerin CASP3 Text_Mining(increases(cleavage)) CTD rottlerin CASP6 Text_Mining(decreases(reaction)) CTD rottlerin CASP6 Text_Mining(increases(cleavage)) CTD rottlerin CASP9 Text_Mining(increases(cleavage)) CTD rottlerin CCND1 Text_Mining(affects(cotreatment)) CTD rottlerin CCND1 Text_Mining(decreases(expression)) CTD rottlerin CCND3 Text_Mining(affects(cotreatment)) CTD rottlerin CCND3 Text_Mining(decreases(expression)) CTD rottlerin CD38 Text_Mining(decreases(reaction)) CTD rottlerin CD38 Text_Mining(increases(expression)) CTD rottlerin CDK4 Text_Mining(affects(cotreatment)) CTD rottlerin CDK4 Text_Mining(decreases(expression)) CTD rottlerin CDK6 Text_Mining(affects(cotreatment)) CTD rottlerin CDK6 Text_Mining(decreases(expression)) CTD rottlerin CDKN1A Text_Mining(decreases(reaction)) CTD rottlerin CDKN1A Text_Mining(increases(expression)) CTD rottlerin CEBPA Text_Mining(decreases(expression)) CTD rottlerin CEBPA Text_Mining(decreases(reaction)) CTD rottlerin CEBPA Text_Mining(increases(ubiquitination)) CTD rottlerin COL1A1 Text_Mining(decreases(activity)) CTD rottlerin COL1A1 Text_Mining(decreases(reaction)) CTD rottlerin COL1A1 Text_Mining(increases(expression)) CTD rottlerin COL1A1 Text_Mining(increases(phosphorylation)) CTD rottlerin CXCL8 Text_Mining(decreases(reaction)) CTD rottlerin CXCL8 Text_Mining(increases(expression)) CTD rottlerin CYP19A1 Text_Mining(decreases(activity)) CTD rottlerin DDIT3 Text_Mining(decreases(reaction)) CTD rottlerin DDIT3 Text_Mining(increases(expression)) CTD rottlerin EGFR Text_Mining(decreases(reaction)) CTD rottlerin EGFR Text_Mining(increases(phosphorylation)) CTD rottlerin EGFR Text_Mining(increases(activity)) CTD rottlerin EIF4E Text_Mining(affects(binding)) CTD rottlerin EIF4E Text_Mining(increases(reaction)) CTD rottlerin EIF4EBP1 Text_Mining(decreases(reaction)) CTD rottlerin EIF4EBP1 Text_Mining(increases(phosphorylation)) CTD rottlerin EIF4EBP1 Text_Mining(affects(binding)) CTD rottlerin EIF4EBP1 Text_Mining(increases(reaction)) CTD rottlerin FOS Text_Mining(affects(localization)) CTD rottlerin FOS Text_Mining(decreases(reaction)) CTD rottlerin GCLC Text_Mining(decreases(reaction)) CTD rottlerin GCLC Text_Mining(increases(activity)) CTD rottlerin GCLC Text_Mining(increases(expression)) CTD rottlerin GDF15 Text_Mining(decreases(reaction)) CTD rottlerin GDF15 Text_Mining(increases(expression)) CTD rottlerin GDF15 Text_Mining(affects(response to substance)) CTD rottlerin HMOX1 Text_Mining(decreases(reaction)) CTD rottlerin HMOX1 Text_Mining(increases(expression)) CTD rottlerin HMOX1 Text_Mining(increases(activity)) CTD rottlerin HNRNPK Text_Mining(decreases(expression)) CTD rottlerin HNRNPK Text_Mining(decreases(reaction)) CTD rottlerin HSPA5 Text_Mining(increases(expression)) CTD rottlerin IFNA2 Text_Mining(decreases(reaction)) CTD rottlerin IFNA2 Text_Mining(increases(expression)) CTD rottlerin IFNA2 Text_Mining(increases(activity)) CTD rottlerin IFNA2 Text_Mining(increases(phosphorylation)) CTD rottlerin IL2 Text_Mining(affects(cotreatment)) CTD rottlerin IL2 Text_Mining(decreases(reaction)) CTD rottlerin IL2 Text_Mining(increases(expression)) CTD rottlerin IL2 Text_Mining(increases(reaction)) CTD rottlerin JUN Text_Mining(affects(localization)) CTD rottlerin JUN Text_Mining(decreases(reaction)) CTD rottlerin JUN Text_Mining(increases(activity)) CTD rottlerin JUN Text_Mining(increases(expression)) CTD rottlerin JUN Text_Mining(increases(phosphorylation)) CTD rottlerin MAP2K1 Text_Mining(decreases(phosphorylation)) CTD rottlerin MAPK1 Text_Mining(decreases(reaction)) CTD rottlerin MAPK1 Text_Mining(increases(activity)) CTD rottlerin MAPK1 Text_Mining(increases(phosphorylation)) CTD rottlerin MAPK1 Text_Mining(affects(cotreatment)) CTD rottlerin MAPK1 Text_Mining(decreases(phosphorylation)) CTD rottlerin MAPK14 Text_Mining(decreases(phosphorylation)) CTD rottlerin MAPK3 Text_Mining(decreases(reaction)) CTD rottlerin MAPK3 Text_Mining(increases(activity)) CTD rottlerin MAPK3 Text_Mining(increases(phosphorylation)) CTD rottlerin MAPK3 Text_Mining(affects(cotreatment)) CTD rottlerin MAPK3 Text_Mining(decreases(phosphorylation)) CTD rottlerin MAPK8 Text_Mining(decreases(reaction)) CTD rottlerin MAPK8 Text_Mining(increases(phosphorylation)) CTD rottlerin MAPK9 Text_Mining(decreases(reaction)) CTD rottlerin MAPK9 Text_Mining(increases(phosphorylation)) CTD rottlerin MIF Text_Mining(decreases(reaction)) CTD rottlerin MIF Text_Mining(increases(expression)) CTD rottlerin MMP2 Text_Mining(decreases(reaction)) CTD rottlerin MMP2 Text_Mining(increases(expression)) CTD rottlerin MMP2 Text_Mining(increases(activity)) CTD rottlerin MTOR Text_Mining(decreases(reaction)) CTD rottlerin MTOR Text_Mining(increases(phosphorylation)) CTD rottlerin MTOR Text_Mining(decreases(phosphorylation)) CTD rottlerin NFE2L2 Text_Mining(decreases(reaction)) CTD rottlerin NFE2L2 Text_Mining(increases(activity)) CTD rottlerin NFE2L2 Text_Mining(increases(expression)) CTD rottlerin NFE2L2 Text_Mining(affects(localization)) CTD rottlerin NTS Text_Mining(decreases(reaction)) CTD rottlerin NTS Text_Mining(increases(activity)) CTD rottlerin NTS Text_Mining(increases(phosphorylation)) CTD rottlerin PARP1 Text_Mining(increases(cleavage)) CTD rottlerin PLD1 Text_Mining(decreases(reaction)) CTD rottlerin PLD1 Text_Mining(increases(expression)) CTD rottlerin PLD1 Text_Mining(increases(reaction)) CTD rottlerin PLSCR1 Text_Mining(decreases(reaction)) CTD rottlerin PLSCR1 Text_Mining(increases(expression)) CTD rottlerin PPARG Text_Mining(decreases(activity)) CTD rottlerin PPARG Text_Mining(decreases(reaction)) CTD rottlerin PPARG Text_Mining(increases(expression)) CTD rottlerin PPARG Text_Mining(increases(phosphorylation)) CTD rottlerin PRKCD Text_Mining(decreases(response to substance)) CTD rottlerin PRKCD Text_Mining(decreases(reaction)) CTD rottlerin PRKCD Text_Mining(increases(phosphorylation)) CTD rottlerin PRKCD Text_Mining(increases(activity)) CTD rottlerin PRKCD Text_Mining(increases(cleavage)) CTD rottlerin PRKCD Text_Mining(decreases(activity)) CTD rottlerin PRKCD Text_Mining(increases(expression)) CTD rottlerin PRKCD Text_Mining(increases(reaction)) CTD rottlerin PRKCQ Text_Mining(decreases(activity)) CTD rottlerin PTGS2 Text_Mining(decreases(reaction)) CTD rottlerin PTGS2 Text_Mining(increases(expression)) CTD rottlerin PTGS2 Text_Mining(increases(reaction)) CTD rottlerin RAF1 Text_Mining(decreases(phosphorylation)) CTD rottlerin RB1 Text_Mining(decreases(phosphorylation)) CTD rottlerin SOD2 Text_Mining(decreases(reaction)) CTD rottlerin SOD2 Text_Mining(increases(expression)) CTD rottlerin STS Text_Mining(decreases(reaction)) CTD rottlerin STS Text_Mining(increases(activity)) CTD rottlerin TFF1 Text_Mining(decreases(activity)) CTD rottlerin TFF1 Text_Mining(decreases(reaction)) CTD rottlerin TFF1 Text_Mining(increases(expression)) CTD rottlerin TFF1 Text_Mining(increases(reaction)) CTD rottlerin TGFA Text_Mining(decreases(reaction)) CTD rottlerin TGFA Text_Mining(increases(secretion)) CTD rottlerin TNFRSF10B Text_Mining(decreases(reaction)) CTD rottlerin TNFRSF10B Text_Mining(increases(expression)) CTD rottlerin VEGFA Text_Mining(decreases(reaction)) CTD rottlerin VEGFA Text_Mining(increases(abundance)) CTD rottlerin XIAP Text_Mining(decreases(expression)) CTD rottlerin ALDH1A1 Potency=14.1254(uM) D4 PubChem rottlerin ALDH1A1 Potency=17.7828(uM) D4 PubChem rottlerin ALDH1A1 Potency=17782.8(nM) D4 ChEMBL rottlerin ALDH1A1 Potency=14125.4(nM) D4 ChEMBL rottlerin ATM Potency=10.0(uM) D4 PubChem rottlerin ATM Potency=29.1921(uM) D4 PubChem rottlerin ATM None=None(uM) D4 PubChem rottlerin CBX1 Potency=12.5893(uM) D4 PubChem rottlerin CBX1 Potency=12589.3(nM) D4 ChEMBL rottlerin EHMT2 Potency=2.1192(uM) D4 PubChem rottlerin EHMT2 Potency=14.1254(uM) D4 PubChem rottlerin EHMT2 Potency=14125.4(nM) D4 ChEMBL rottlerin EHMT2 Potency=2119.2(nM) D4 ChEMBL rottlerin KAT2A Potency=11.2202(uM) D4 PubChem rottlerin KAT2A Potency=11220.2(nM) D4 ChEMBL rottlerin MAPT Potency=12.5893(uM) D4 PubChem rottlerin MAPT Potency=15.8489(uM) D4 PubChem rottlerin MAPT Potency=17.7828(uM) D4 PubChem rottlerin MAPT Potency=15848.9(nM) D4 ChEMBL rottlerin MAPT Potency=17782.8(nM) D4 ChEMBL rottlerin MAPT Potency=12589.3(nM) D4 ChEMBL rottlerin POLI Potency=50.1187(uM) D4 PubChem rottlerin PRKCD Inhibition=None(Unspecified) D4 ChEMBL rottlerin RGS4 Potency=10.6213(uM) D4 PubChem rottlerin RHOA Inhibition=None(Unspecified) D4 ChEMBL rottlerin TDP1 Potency=8.9125(uM) D4 PubChem rottlerin TDP1 Potency=13.3359(uM) D4 PubChem rottlerin TDP1 Potency=19.7612(uM) D4 PubChem rottlerin TDP1 Potency=29.8554(uM) D4 PubChem rottlerin USP1 Potency=41.8398(uM) D4 PubChem rottlerin USP1 Potency=56.2341(uM) D4 PubChem rottlerin USP1 Potency=79.4328(uM) D4 PubChem rottlerin VDR Potency=8.9125(uM) D4 PubChem rottlerin VDR Potency=14.1254(uM) D4 PubChem rottlerin VDR Potency=39.8107(uM) D4 PubChem