Drug Gene Type Source Tyrphostin AG 879 AHR Text_Mining(decreases(reaction)) CTD Tyrphostin AG 879 AHR Text_Mining(increases(activity)) CTD Tyrphostin AG 879 IL6 Text_Mining(decreases(reaction)) CTD Tyrphostin AG 879 IL6 Text_Mining(increases(expression)) CTD Tyrphostin AG 879 IL6 Text_Mining(decreases(activity)) CTD Tyrphostin AG 879 KLK3 Text_Mining(decreases(reaction)) CTD Tyrphostin AG 879 KLK3 Text_Mining(increases(expression)) CTD Tyrphostin AG 879 ALDH1A1 Potency=2.8184(uM) D4 PubChem Tyrphostin AG 879 ALDH1A1 Potency=2818.4(nM) D4 ChEMBL Tyrphostin AG 879 ALOX15B Potency=12589.3(nM) D4 ChEMBL Tyrphostin AG 879 CBX1 Potency=11.2202(uM) D4 PubChem Tyrphostin AG 879 CBX1 Potency=11220.2(nM) D4 ChEMBL Tyrphostin AG 879 CYP1A2 None=None(uM) D4 PubChem Tyrphostin AG 879 CYP1A2 AC50=12589.2(nM) D4 ChEMBL Tyrphostin AG 879 CYP2C19 Potency=10.0(uM) D4 PubChem Tyrphostin AG 879 CYP2C19 None=None(uM) D4 PubChem Tyrphostin AG 879 CYP2C19 AC50=10000.0(nM) D4 ChEMBL Tyrphostin AG 879 CYP2C19 Potency=10000.0(nM) D4 ChEMBL Tyrphostin AG 879 CYP2C9 Potency=0.1(uM) D4 PubChem Tyrphostin AG 879 CYP2C9 None=None(uM) D4 PubChem Tyrphostin AG 879 CYP2C9 AC50=100.0(nM) D4 ChEMBL Tyrphostin AG 879 CYP2C9 Potency=100.0(nM) D4 ChEMBL Tyrphostin AG 879 CYP3A4 Potency=3.9811(uM) D4 PubChem Tyrphostin AG 879 CYP3A4 None=None(uM) D4 PubChem Tyrphostin AG 879 CYP3A4 AC50=3981.07(nM) D4 ChEMBL Tyrphostin AG 879 CYP3A4 Potency=3981.1(nM) D4 ChEMBL Tyrphostin AG 879 EHMT2 Potency=28.1838(uM) D4 PubChem Tyrphostin AG 879 EHMT2 Potency=28183.8(nM) D4 ChEMBL Tyrphostin AG 879 GLS Potency=4.4668(uM) D4 PubChem Tyrphostin AG 879 GMNN Potency=3.1623(uM) D4 PubChem Tyrphostin AG 879 GMNN Potency=3162.3(nM) D4 ChEMBL Tyrphostin AG 879 HIF1A Potency=0.631(uM) D4 PubChem Tyrphostin AG 879 HIF1A Potency=631.0(nM) D4 ChEMBL Tyrphostin AG 879 HSD17B10 Potency=12589.3(nM) D4 ChEMBL Tyrphostin AG 879 KCNH2 Potency=11.2202(uM) D4 PubChem Tyrphostin AG 879 MPHOSPH8 Potency=11.2202(uM) D4 PubChem Tyrphostin AG 879 MPHOSPH8 Potency=11220.2(nM) D4 ChEMBL Tyrphostin AG 879 RGS4 Potency=10.6213(uM) D4 PubChem Tyrphostin AG 879 TDP1 Potency=0.5623(uM) D4 PubChem Tyrphostin AG 879 TDP1 Potency=0.7079(uM) D4 PubChem Tyrphostin AG 879 TDP1 Potency=4.1095(uM) D4 PubChem Tyrphostin AG 879 TDP1 Potency=5.8048(uM) D4 PubChem Tyrphostin AG 879 THPO Potency=10.0(uM) D4 PubChem Tyrphostin AG 879 THPO Potency=10000.0(nM) D4 ChEMBL Tyrphostin AG 879 TSHR Potency=3.1623(uM) D4 PubChem Tyrphostin AG 879 TSHR Potency=3162.3(nM) D4 ChEMBL Tyrphostin AG 879 VDR Potency=35.4813(uM) D4 PubChem