Drug Gene Type Source bisindolylmaleimide i ABCB4 Text_Mining(decreases(expression)) CTD bisindolylmaleimide i ABCB4 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i ACE Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i ACE Text_Mining(increases(expression)) CTD bisindolylmaleimide i AGT Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i AGT Text_Mining(increases(expression)) CTD bisindolylmaleimide i AKT1 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i AKT1 Text_Mining(increases(activity)) CTD bisindolylmaleimide i AKT1 Text_Mining(increases(phosphorylation)) CTD bisindolylmaleimide i AKT1 Text_Mining(decreases(activity)) CTD bisindolylmaleimide i AKT1 Text_Mining(decreases(phosphorylation)) CTD bisindolylmaleimide i AREG Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i AREG Text_Mining(increases(expression)) CTD bisindolylmaleimide i AREG Text_Mining(increases(reaction)) CTD bisindolylmaleimide i ATP1A1 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i ATP1A1 Text_Mining(increases(expression)) CTD bisindolylmaleimide i CASR Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i CASR Text_Mining(increases(phosphorylation)) CTD bisindolylmaleimide i CASR Text_Mining(increases(reaction)) CTD bisindolylmaleimide i CD86 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i CD86 Text_Mining(increases(expression)) CTD bisindolylmaleimide i CNN1 Text_Mining(decreases(expression)) CTD bisindolylmaleimide i CREB1 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i CREB1 Text_Mining(increases(phosphorylation)) CTD bisindolylmaleimide i CSF2 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i CSF2 Text_Mining(increases(secretion)) CTD bisindolylmaleimide i CTGF Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i CTGF Text_Mining(increases(expression)) CTD bisindolylmaleimide i CXCL12 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i CXCL12 Text_Mining(increases(expression)) CTD bisindolylmaleimide i CXCL8 Text_Mining(affects(reaction)) CTD bisindolylmaleimide i CXCL8 Text_Mining(increases(expression)) CTD bisindolylmaleimide i CXCL8 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i EGFR Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i EGFR Text_Mining(increases(phosphorylation)) CTD bisindolylmaleimide i ERBB4 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i ERBB4 Text_Mining(increases(cleavage)) CTD bisindolylmaleimide i FOS Text_Mining(affects(cotreatment)) CTD bisindolylmaleimide i FOS Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i FOS Text_Mining(increases(expression)) CTD bisindolylmaleimide i HGF Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i HGF Text_Mining(increases(expression)) CTD bisindolylmaleimide i IL11 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i IL11 Text_Mining(increases(expression)) CTD bisindolylmaleimide i IL5 Text_Mining(decreases(activity)) CTD bisindolylmaleimide i INHBA Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i INHBA Text_Mining(increases(expression)) CTD bisindolylmaleimide i INS Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i INS Text_Mining(increases(expression)) CTD bisindolylmaleimide i INS Text_Mining(increases(activity)) CTD bisindolylmaleimide i INS Text_Mining(increases(phosphorylation)) CTD bisindolylmaleimide i ITGB2 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i ITGB2 Text_Mining(increases(activity)) CTD bisindolylmaleimide i JUN Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i JUN Text_Mining(increases(activity)) CTD bisindolylmaleimide i JUN Text_Mining(increases(expression)) CTD bisindolylmaleimide i JUN Text_Mining(increases(phosphorylation)) CTD bisindolylmaleimide i KDR Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i KDR Text_Mining(increases(expression)) CTD bisindolylmaleimide i MAP2K1 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i MAP2K1 Text_Mining(increases(activity)) CTD bisindolylmaleimide i MAP2K1 Text_Mining(increases(phosphorylation)) CTD bisindolylmaleimide i MAP2K2 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i MAP2K2 Text_Mining(increases(activity)) CTD bisindolylmaleimide i MAP2K2 Text_Mining(increases(phosphorylation)) CTD bisindolylmaleimide i MAPK1 Text_Mining(affects(cotreatment)) CTD bisindolylmaleimide i MAPK1 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i MAPK1 Text_Mining(increases(phosphorylation)) CTD bisindolylmaleimide i MAPK1 Text_Mining(increases(activity)) CTD bisindolylmaleimide i MAPK14 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i MAPK14 Text_Mining(increases(phosphorylation)) CTD bisindolylmaleimide i MAPK3 Text_Mining(affects(cotreatment)) CTD bisindolylmaleimide i MAPK3 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i MAPK3 Text_Mining(increases(phosphorylation)) CTD bisindolylmaleimide i MAPK3 Text_Mining(increases(activity)) CTD bisindolylmaleimide i MMP9 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i MMP9 Text_Mining(increases(expression)) CTD bisindolylmaleimide i MMP9 Text_Mining(increases(activity)) CTD bisindolylmaleimide i MMP9 Text_Mining(increases(secretion)) CTD bisindolylmaleimide i NCF1 Text_Mining(affects(localization)) CTD bisindolylmaleimide i NCF1 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i NFKB1 Text_Mining(affects(binding)) CTD bisindolylmaleimide i NFKB1 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i NFKB1 Text_Mining(increases(activity)) CTD bisindolylmaleimide i NRG1 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i NRG1 Text_Mining(increases(activity)) CTD bisindolylmaleimide i NRG1 Text_Mining(increases(phosphorylation)) CTD bisindolylmaleimide i P2RY1 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i P2RY1 Text_Mining(increases(activity)) CTD bisindolylmaleimide i P2RY1 Text_Mining(increases(phosphorylation)) CTD bisindolylmaleimide i PARP1 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i PARP1 Text_Mining(increases(cleavage)) CTD bisindolylmaleimide i PDGFRB Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i PDGFRB Text_Mining(increases(activity)) CTD bisindolylmaleimide i PDGFRB Text_Mining(increases(phosphorylation)) CTD bisindolylmaleimide i PGR Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i PGR Text_Mining(increases(expression)) CTD bisindolylmaleimide i PPARG Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i PPARG Text_Mining(increases(expression)) CTD bisindolylmaleimide i PRKCD Text_Mining(affects(phosphorylation)) CTD bisindolylmaleimide i PRKCD Text_Mining(affects(reaction)) CTD bisindolylmaleimide i PRKD1 Text_Mining(affects(phosphorylation)) CTD bisindolylmaleimide i PRKD1 Text_Mining(affects(reaction)) CTD bisindolylmaleimide i PTGS2 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i PTGS2 Text_Mining(increases(expression)) CTD bisindolylmaleimide i RAC1 Text_Mining(affects(localization)) CTD bisindolylmaleimide i RAC1 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i RAP1A Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i RAP1A Text_Mining(increases(activity)) CTD bisindolylmaleimide i RB1 Text_Mining(increases(expression)) CTD bisindolylmaleimide i RELA Text_Mining(affects(binding)) CTD bisindolylmaleimide i RELA Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i RELA Text_Mining(increases(activity)) CTD bisindolylmaleimide i RELA Text_Mining(affects(localization)) CTD bisindolylmaleimide i RXRA Text_Mining(affects(cotreatment)) CTD bisindolylmaleimide i RXRA Text_Mining(decreases(phosphorylation)) CTD bisindolylmaleimide i SLC6A3 Text_Mining(affects(cotreatment)) CTD bisindolylmaleimide i SLC6A3 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i SLC6A3 Text_Mining(increases(expression)) CTD bisindolylmaleimide i SOD2 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i SOD2 Text_Mining(increases(expression)) CTD bisindolylmaleimide i SOD2 Text_Mining(increases(reaction)) CTD bisindolylmaleimide i SOD2 Text_Mining(decreases(expression)) CTD bisindolylmaleimide i SP1 Text_Mining(increases(expression)) CTD bisindolylmaleimide i STS Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i STS Text_Mining(increases(activity)) CTD bisindolylmaleimide i TAGLN Text_Mining(decreases(expression)) CTD bisindolylmaleimide i TFF1 Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i TFF1 Text_Mining(increases(expression)) CTD bisindolylmaleimide i TFF1 Text_Mining(increases(reaction)) CTD bisindolylmaleimide i TNF Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i TNF Text_Mining(increases(expression)) CTD bisindolylmaleimide i TP53 Text_Mining(decreases(degradation)) CTD bisindolylmaleimide i TP53 Text_Mining(increases(expression)) CTD bisindolylmaleimide i VEGFA Text_Mining(affects(cotreatment)) CTD bisindolylmaleimide i VEGFA Text_Mining(decreases(reaction)) CTD bisindolylmaleimide i VEGFA Text_Mining(increases(expression)) CTD bisindolylmaleimide i VEGFA Text_Mining(affects(localization)) CTD bisindolylmaleimide i VEGFA Text_Mining(increases(abundance)) CTD bisindolylmaleimide i VEGFA Text_Mining(increases(reaction)) CTD bisindolylmaleimide i CYP1A2 None=None(uM) D4 PubChem bisindolylmaleimide i CYP1A2 AC50=7943.28(nM) D4 ChEMBL bisindolylmaleimide i CYP3A4 Potency=12.5893(uM) D4 PubChem bisindolylmaleimide i CYP3A4 None=None(uM) D4 PubChem bisindolylmaleimide i CYP3A4 AC50=12589.2(nM) D4 ChEMBL bisindolylmaleimide i CYP3A4 Potency=12589.3(nM) D4 ChEMBL bisindolylmaleimide i EHMT2 Potency=14.1254(uM) D4 PubChem bisindolylmaleimide i EHMT2 Potency=17.7828(uM) D4 PubChem bisindolylmaleimide i EHMT2 Potency=17782.8(nM) D4 ChEMBL bisindolylmaleimide i EHMT2 Potency=14125.4(nM) D4 ChEMBL bisindolylmaleimide i MAPK1 Potency=0.7943(uM) D4 PubChem bisindolylmaleimide i MAPK1 Potency=1.2589(uM) D4 PubChem bisindolylmaleimide i MAPK1 Potency=794.3(nM) D4 ChEMBL bisindolylmaleimide i MAPK1 Potency=1258.9(nM) D4 ChEMBL bisindolylmaleimide i MAPT Potency=12.5893(uM) D4 PubChem bisindolylmaleimide i MAPT None=None(uM) D4 PubChem bisindolylmaleimide i MAPT Potency=28183.8(nM) D4 ChEMBL bisindolylmaleimide i MAPT Potency=12589.3(nM) D4 ChEMBL bisindolylmaleimide i MAPT Potency=19952.6(nM) D4 ChEMBL bisindolylmaleimide i RECQL Potency=28183.8(nM) D4 ChEMBL bisindolylmaleimide i TDP1 Potency=23.715(uM) D4 PubChem bisindolylmaleimide i USP1 Potency=50.1187(uM) D4 PubChem