Drug Gene Type Source Bergamottin AHR Text_Mining(increases(activity)) CTD Bergamottin CD74 Text_Mining(decreases(expression)) CTD Bergamottin CYP1B1 Text_Mining(decreases(reaction)) CTD Bergamottin CYP1B1 Text_Mining(increases(oxidation)) CTD Bergamottin CYP1B1 Text_Mining(decreases(activity)) CTD Bergamottin CYP2B6 Text_Mining(decreases(activity)) CTD Bergamottin CYP3A4 Text_Mining(decreases(activity)) CTD Bergamottin NR1I2 Text_Mining(increases(activity)) CTD Bergamottin NR1I3 Text_Mining(increases(activity)) CTD Bergamottin UGT1A1 Text_Mining(increases(glucuronidation)) CTD Bergamottin UGT1A10 Text_Mining(increases(glucuronidation)) CTD Bergamottin UGT1A7 Text_Mining(increases(glucuronidation)) CTD Bergamottin UGT1A8 Text_Mining(increases(glucuronidation)) CTD Bergamottin UGT1A9 Text_Mining(increases(glucuronidation)) CTD Bergamottin BACE1 Inhibition=None(Unspecified) D4 ChEMBL Bergamottin CYP1A2 None=None(uM) D4 PubChem Bergamottin CYP2C19 Potency=0.01(uM) D4 PubChem Bergamottin CYP2C19 Potency=10.0(nM) D4 ChEMBL Bergamottin CYP2C9 Potency=0.0316(uM) D4 PubChem Bergamottin CYP2C9 Potency=31.6(nM) D4 ChEMBL Bergamottin CYP2D6 Potency=0.0631(uM) D4 PubChem Bergamottin CYP2D6 Potency=63.1(nM) D4 ChEMBL Bergamottin DRD1 None=None(uM) D4 PubChem Bergamottin TSHR Potency=12.5893(uM) D4 PubChem Bergamottin TSHR Potency=12589.3(nM) D4 ChEMBL