Drug Gene Type Source AM580 ABCG2 Text_Mining(increases(expression)) CTD AM580 ABCG2 Text_Mining(increases(reaction)) CTD AM580 ADA Text_Mining(increases(expression)) CTD AM580 AGPAT4 Text_Mining(increases(expression)) CTD AM580 AGRN Text_Mining(decreases(expression)) CTD AM580 AJAP1 Text_Mining(increases(expression)) CTD AM580 APLP2 Text_Mining(increases(expression)) CTD AM580 ATP2B1 Text_Mining(decreases(expression)) CTD AM580 BAG2 Text_Mining(increases(expression)) CTD AM580 C16ORF46 Text_Mining(decreases(expression)) CTD AM580 C4ORF32 Text_Mining(decreases(expression)) CTD AM580 CALCRL Text_Mining(decreases(expression)) CTD AM580 CD1A Text_Mining(decreases(expression)) CTD AM580 CD1D Text_Mining(increases(expression)) CTD AM580 CD1D Text_Mining(decreases(reaction)) CTD AM580 CD300A Text_Mining(increases(expression)) CTD AM580 CD300LB Text_Mining(increases(expression)) CTD AM580 CD300LF Text_Mining(increases(expression)) CTD AM580 CD38 Text_Mining(decreases(reaction)) CTD AM580 CD38 Text_Mining(increases(expression)) CTD AM580 CD38 Text_Mining(affects(cotreatment)) CTD AM580 CDKN1B Text_Mining(affects(localization)) CTD AM580 CDR2L Text_Mining(decreases(expression)) CTD AM580 CGB Text_Mining(increases(expression)) CTD AM580 COL5A3 Text_Mining(increases(expression)) CTD AM580 CTTNBP2 Text_Mining(decreases(expression)) CTD AM580 CYP19A1 Text_Mining(increases(expression)) CTD AM580 DCSTAMP Text_Mining(increases(expression)) CTD AM580 DHRS3 Text_Mining(increases(expression)) CTD AM580 DMPK Text_Mining(decreases(expression)) CTD AM580 DMWD Text_Mining(decreases(expression)) CTD AM580 DNAJC5B Text_Mining(increases(expression)) CTD AM580 ETS2 Text_Mining(increases(expression)) CTD AM580 FAM101B Text_Mining(increases(expression)) CTD AM580 FAM109A Text_Mining(decreases(expression)) CTD AM580 FN1 Text_Mining(increases(expression)) CTD AM580 FUT7 Text_Mining(decreases(expression)) CTD AM580 GALM Text_Mining(increases(expression)) CTD AM580 GDF15 Text_Mining(increases(expression)) CTD AM580 GOLGA8A Text_Mining(decreases(expression)) CTD AM580 GPD1L Text_Mining(decreases(expression)) CTD AM580 GUSB Text_Mining(increases(expression)) CTD AM580 HIPK2 Text_Mining(increases(expression)) CTD AM580 HIST1H2BD Text_Mining(decreases(expression)) CTD AM580 HLX Text_Mining(decreases(expression)) CTD AM580 IFNGR1 Text_Mining(increases(expression)) CTD AM580 IFNGR1 Text_Mining(decreases(reaction)) CTD AM580 IL1R1 Text_Mining(decreases(expression)) CTD AM580 IL1RAP Text_Mining(decreases(expression)) CTD AM580 INPP5F Text_Mining(increases(expression)) CTD AM580 IPCEF1 Text_Mining(decreases(expression)) CTD AM580 IRF1 Text_Mining(affects(localization)) CTD AM580 IRF1 Text_Mining(increases(expression)) CTD AM580 IRF1 Text_Mining(increases(activity)) CTD AM580 IRF1 Text_Mining(decreases(reaction)) CTD AM580 IRF1 Text_Mining(increases(reaction)) CTD AM580 ITGAE Text_Mining(increases(expression)) CTD AM580 KIAA0040 Text_Mining(decreases(expression)) CTD AM580 KIAA1161 Text_Mining(decreases(expression)) CTD AM580 KIFC2 Text_Mining(decreases(expression)) CTD AM580 LAIR1 Text_Mining(increases(expression)) CTD AM580 LELP1 Text_Mining(decreases(expression)) CTD AM580 LILRA1 Text_Mining(increases(expression)) CTD AM580 LRP11 Text_Mining(decreases(expression)) CTD AM580 MAN1C1 Text_Mining(decreases(expression)) CTD AM580 MAP3K6 Text_Mining(decreases(expression)) CTD AM580 MAP4K1 Text_Mining(decreases(expression)) CTD AM580 MAPK1 Text_Mining(affects(cotreatment)) CTD AM580 MAPK1 Text_Mining(increases(activity)) CTD AM580 MAPK1 Text_Mining(increases(phosphorylation)) CTD AM580 MAPK3 Text_Mining(affects(cotreatment)) CTD AM580 MAPK3 Text_Mining(increases(activity)) CTD AM580 MAPK3 Text_Mining(increases(phosphorylation)) CTD AM580 METRN Text_Mining(decreases(expression)) CTD AM580 MGAT4C Text_Mining(decreases(expression)) CTD AM580 NDRG2 Text_Mining(decreases(expression)) CTD AM580 NRIP1 Text_Mining(increases(expression)) CTD AM580 NRIP3 Text_Mining(increases(expression)) CTD AM580 NUDT7 Text_Mining(decreases(expression)) CTD AM580 OAS2 Text_Mining(increases(expression)) CTD AM580 OAS2 Text_Mining(decreases(reaction)) CTD AM580 OCLN Text_Mining(increases(expression)) CTD AM580 OLR1 Text_Mining(increases(expression)) CTD AM580 OMA1 Text_Mining(increases(expression)) CTD AM580 PALD1 Text_Mining(decreases(expression)) CTD AM580 PAPSS2 Text_Mining(increases(expression)) CTD AM580 PDLIM2 Text_Mining(decreases(expression)) CTD AM580 PDLIM4 Text_Mining(decreases(expression)) CTD AM580 PHLDA2 Text_Mining(decreases(expression)) CTD AM580 PLBD1 Text_Mining(increases(expression)) CTD AM580 PON2 Text_Mining(decreases(expression)) CTD AM580 PPAP2B Text_Mining(increases(expression)) CTD AM580 PRAM1 Text_Mining(increases(expression)) CTD AM580 QPRT Text_Mining(decreases(expression)) CTD AM580 RAB15 Text_Mining(decreases(expression)) CTD AM580 RAB20 Text_Mining(increases(expression)) CTD AM580 RAP1GAP Text_Mining(decreases(expression)) CTD AM580 RARA Text_Mining(affects(binding)) CTD AM580 RARA Text_Mining(increases(activity)) CTD AM580 RARA Text_Mining(increases(expression)) CTD AM580 RB1 Text_Mining(affects(cotreatment)) CTD AM580 RB1 Text_Mining(decreases(phosphorylation)) CTD AM580 RBP1 Text_Mining(increases(expression)) CTD AM580 REPS2 Text_Mining(decreases(expression)) CTD AM580 RFXAP Text_Mining(decreases(expression)) CTD AM580 RHOBTB3 Text_Mining(increases(expression)) CTD AM580 RXRA Text_Mining(increases(activity)) CTD AM580 SELPLG Text_Mining(decreases(expression)) CTD AM580 SIGLEC17P Text_Mining(increases(expression)) CTD AM580 SLC26A11 Text_Mining(increases(expression)) CTD AM580 SLITRK4 Text_Mining(increases(expression)) CTD AM580 SNAI3 Text_Mining(increases(expression)) CTD AM580 SSMEM1 Text_Mining(decreases(expression)) CTD AM580 STAT1 Text_Mining(increases(activity)) CTD AM580 STAT1 Text_Mining(increases(phosphorylation)) CTD AM580 STAT1 Text_Mining(decreases(reaction)) CTD AM580 STS Text_Mining(increases(activity)) CTD AM580 TACSTD2 Text_Mining(decreases(expression)) CTD AM580 TBC1D2 Text_Mining(increases(expression)) CTD AM580 TBL1X Text_Mining(decreases(expression)) CTD AM580 TBL2 Text_Mining(increases(expression)) CTD AM580 TERT Text_Mining(affects(cotreatment)) CTD AM580 TERT Text_Mining(decreases(expression)) CTD AM580 TGM2 Text_Mining(affects(cotreatment)) CTD AM580 TGM2 Text_Mining(increases(activity)) CTD AM580 TGM2 Text_Mining(increases(expression)) CTD AM580 THBS3 Text_Mining(increases(expression)) CTD AM580 TMEM14A Text_Mining(decreases(expression)) CTD AM580 TNFSF12 Text_Mining(decreases(expression)) CTD AM580 TNS1 Text_Mining(decreases(expression)) CTD AM580 ZBTB7B Text_Mining(decreases(expression)) CTD AM580 AR Potency-Replicate_1=48.9662(uM) D4 PubChem AM580 AR Ratio Potency (uM)=48.9662(uM) D4 PubChem AM580 CYP1A2 None=None(uM) D4 PubChem AM580 ESR1 Potency-Replicate_1=0.0043(uM) D4 PubChem AM580 ESR1 ER Potency (uM)=0.0104614(uM) D4 PubChem AM580 NFE2L2 Potency=61.1306(uM) D4 PubChem AM580 NR1H4 Potency-Replicate_1=43.6412(uM) D4 PubChem AM580 NR1H4 Ratio Potency (uM)=43.6412(uM) D4 PubChem AM580 VDR Potency=79.4328(uM) D4 PubChem