Drug Gene Type Source letrozole CCND1 Text_Mining(affects(cotreatment)) CTD letrozole CCND1 Text_Mining(decreases(expression)) CTD letrozole CCND2 Text_Mining(affects(cotreatment)) CTD letrozole CCND2 Text_Mining(decreases(expression)) CTD letrozole CDKN1A Text_Mining(increases(expression)) CTD letrozole CYCS Text_Mining(affects(cotreatment)) CTD letrozole CYCS Text_Mining(affects(localization)) CTD letrozole CYP19A1 Text_Mining(decreases(reaction)) CTD letrozole CYP19A1 Text_Mining(increases(expression)) CTD letrozole CYP19A1 Text_Mining(decreases(activity)) CTD letrozole CYP19A1 Text_Mining(increases(activity)) CTD letrozole CYP51A1 Text_Mining(decreases(activity)) CTD letrozole DKK1 Text_Mining(increases(expression)) CTD letrozole EIF4EBP1 Text_Mining(affects(cotreatment)) CTD letrozole EIF4EBP1 Text_Mining(decreases(activity)) CTD letrozole EIF4EBP1 Text_Mining(increases(phosphorylation)) CTD letrozole FGF22 Text_Mining(increases(expression)) CTD letrozole FSHB Text_Mining(increases(expression)) CTD letrozole LHB Text_Mining(increases(expression)) CTD letrozole LIF Text_Mining(increases(expression)) CTD letrozole LIFR Text_Mining(increases(expression)) CTD letrozole MKI67 Text_Mining(decreases(expression)) CTD letrozole MMP2 Text_Mining(decreases(reaction)) CTD letrozole MMP2 Text_Mining(increases(activity)) CTD letrozole MMP2 Text_Mining(increases(secretion)) CTD letrozole MMP9 Text_Mining(decreases(reaction)) CTD letrozole MMP9 Text_Mining(increases(activity)) CTD letrozole MMP9 Text_Mining(increases(secretion)) CTD letrozole MTOR Text_Mining(affects(activity)) CTD letrozole MTOR Text_Mining(affects(cotreatment)) CTD letrozole MTOR Text_Mining(decreases(reaction)) CTD letrozole MYC Text_Mining(affects(cotreatment)) CTD letrozole MYC Text_Mining(decreases(expression)) CTD letrozole PGR Text_Mining(decreases(expression)) CTD letrozole RB1 Text_Mining(affects(activity)) CTD letrozole RB1 Text_Mining(affects(cotreatment)) CTD letrozole RB1 Text_Mining(decreases(phosphorylation)) CTD letrozole RB1 Text_Mining(decreases(expression)) CTD letrozole RPS6 Text_Mining(affects(cotreatment)) CTD letrozole RPS6 Text_Mining(decreases(phosphorylation)) CTD letrozole SLC22A2 Text_Mining(decreases(reaction)) CTD letrozole SLC22A2 Text_Mining(increases(uptake)) CTD letrozole TERT Text_Mining(decreases(reaction)) CTD letrozole TERT Text_Mining(increases(activity)) CTD letrozole CYP19A1 Potency-Replicate_1=0.0091(uM) D4 PubChem letrozole CYP19A1 Potency-Replicate_1=0.0143(uM) D4 PubChem letrozole CYP19A1 None=None(uM) D4 PubChem letrozole CYP19A1 Inhibition=None(Unspecified) D4 ChEMBL letrozole CYP3A4 Potency=5.0119(uM) D4 PubChem letrozole CYP3A4 None=None(uM) D4 PubChem letrozole CYP3A4 AC50=5011.87(nM) D4 ChEMBL letrozole CYP3A4 Potency=5011.9(nM) D4 ChEMBL letrozole DRD2 None=None(uM) D4 PubChem