Drug Gene Type Source docetaxel ABCA1 Text_Mining(decreases(response to substance)) CTD docetaxel ABCA1 Text_Mining(increases(expression)) CTD docetaxel ABCA10 Text_Mining(decreases(response to substance)) CTD docetaxel ABCA10 Text_Mining(increases(expression)) CTD docetaxel ABCA11P Text_Mining(decreases(response to substance)) CTD docetaxel ABCA11P Text_Mining(increases(expression)) CTD docetaxel ABCA12 Text_Mining(affects(expression)) CTD docetaxel ABCA12 Text_Mining(decreases(response to substance)) CTD docetaxel ABCA3 Text_Mining(decreases(expression)) CTD docetaxel ABCA3 Text_Mining(decreases(response to substance)) CTD docetaxel ABCA4 Text_Mining(decreases(response to substance)) CTD docetaxel ABCA4 Text_Mining(increases(expression)) CTD docetaxel ABCA5 Text_Mining(decreases(response to substance)) CTD docetaxel ABCA5 Text_Mining(increases(expression)) CTD docetaxel ABCA6 Text_Mining(decreases(response to substance)) CTD docetaxel ABCA6 Text_Mining(increases(expression)) CTD docetaxel ABCA7 Text_Mining(decreases(expression)) CTD docetaxel ABCA7 Text_Mining(decreases(response to substance)) CTD docetaxel ABCA8 Text_Mining(decreases(response to substance)) CTD docetaxel ABCA8 Text_Mining(increases(expression)) CTD docetaxel ABCA9 Text_Mining(decreases(response to substance)) CTD docetaxel ABCA9 Text_Mining(increases(expression)) CTD docetaxel ABCB1 Text_Mining(increases(response to substance)) CTD docetaxel ABCB1 Text_Mining(decreases(response to substance)) CTD docetaxel ABCB1 Text_Mining(decreases(reaction)) CTD docetaxel ABCB1 Text_Mining(decreases(expression)) CTD docetaxel ABCB1 Text_Mining(increases(expression)) CTD docetaxel ABCB1 Text_Mining(increases(activity)) CTD docetaxel ABCB1 Text_Mining(increases(reaction)) CTD docetaxel ABCB1 Text_Mining(affects(reaction)) CTD docetaxel ABCB4 Text_Mining(decreases(response to substance)) CTD docetaxel ABCB4 Text_Mining(increases(expression)) CTD docetaxel ABCB6 Text_Mining(decreases(response to substance)) CTD docetaxel ABCB6 Text_Mining(increases(expression)) CTD docetaxel ABCB8 Text_Mining(decreases(expression)) CTD docetaxel ABCB8 Text_Mining(decreases(response to substance)) CTD docetaxel ABCC1 Text_Mining(decreases(response to substance)) CTD docetaxel ABCC1 Text_Mining(increases(expression)) CTD docetaxel ABCC10 Text_Mining(decreases(expression)) CTD docetaxel ABCC10 Text_Mining(decreases(response to substance)) CTD docetaxel ABCC11 Text_Mining(decreases(response to substance)) CTD docetaxel ABCC11 Text_Mining(increases(expression)) CTD docetaxel ABCC2 Text_Mining(affects(transport)) CTD docetaxel ABCC2 Text_Mining(decreases(expression)) CTD docetaxel ABCC2 Text_Mining(decreases(response to substance)) CTD docetaxel ABCC2 Text_Mining(increases(reaction)) CTD docetaxel ABCC3 Text_Mining(decreases(response to substance)) CTD docetaxel ABCC3 Text_Mining(increases(expression)) CTD docetaxel ABCC4 Text_Mining(decreases(expression)) CTD docetaxel ABCC4 Text_Mining(decreases(response to substance)) CTD docetaxel ABCC5 Text_Mining(decreases(response to substance)) CTD docetaxel ABCC5 Text_Mining(increases(expression)) CTD docetaxel ABCC6 Text_Mining(affects(response to substance)) CTD docetaxel ABCC6 Text_Mining(affects(expression)) CTD docetaxel ABCC6 Text_Mining(decreases(response to substance)) CTD docetaxel ABCC9 Text_Mining(decreases(response to substance)) CTD docetaxel ABCC9 Text_Mining(increases(expression)) CTD docetaxel ABCD2 Text_Mining(decreases(expression)) CTD docetaxel ABCD2 Text_Mining(decreases(response to substance)) CTD docetaxel ABCE1 Text_Mining(decreases(expression)) CTD docetaxel ABCE1 Text_Mining(decreases(response to substance)) CTD docetaxel ABCG1 Text_Mining(affects(response to substance)) CTD docetaxel ABCG2 Text_Mining(decreases(expression)) CTD docetaxel ABCG2 Text_Mining(decreases(response to substance)) CTD docetaxel AKT1 Text_Mining(affects(cotreatment)) CTD docetaxel AKT1 Text_Mining(decreases(phosphorylation)) CTD docetaxel AR Text_Mining(decreases(localization)) CTD docetaxel AR Text_Mining(decreases(expression)) CTD docetaxel AR Text_Mining(increases(degradation)) CTD docetaxel BAD Text_Mining(decreases(phosphorylation)) CTD docetaxel BAD Text_Mining(increases(reaction)) CTD docetaxel BAK1 Text_Mining(decreases(reaction)) CTD docetaxel BAK1 Text_Mining(increases(activity)) CTD docetaxel BAK1 Text_Mining(affects(folding)) CTD docetaxel BAK1 Text_Mining(increases(reaction)) CTD docetaxel BAX Text_Mining(increases(expression)) CTD docetaxel BAX Text_Mining(increases(reaction)) CTD docetaxel BAX Text_Mining(decreases(reaction)) CTD docetaxel BAX Text_Mining(increases(activity)) CTD docetaxel BAX Text_Mining(affects(folding)) CTD docetaxel BAX Text_Mining(affects(localization)) CTD docetaxel BAX Text_Mining(affects(cotreatment)) CTD docetaxel BCL2 Text_Mining(decreases(activity)) CTD docetaxel BCL2 Text_Mining(increases(phosphorylation)) CTD docetaxel BCL2 Text_Mining(increases(reaction)) CTD docetaxel BCL2 Text_Mining(decreases(reaction)) CTD docetaxel BCL2 Text_Mining(affects(folding)) CTD docetaxel BCL2 Text_Mining(increases(activity)) CTD docetaxel BCL2 Text_Mining(increases(cleavage)) CTD docetaxel BCL2 Text_Mining(increases(expression)) CTD docetaxel BCL2 Text_Mining(affects(cotreatment)) CTD docetaxel BCL2 Text_Mining(decreases(expression)) CTD docetaxel BCL2L1 Text_Mining(decreases(response to substance)) CTD docetaxel BCL2L1 Text_Mining(affects(cotreatment)) CTD docetaxel BCL2L1 Text_Mining(decreases(expression)) CTD docetaxel BCL2L11 Text_Mining(decreases(reaction)) CTD docetaxel BCL2L11 Text_Mining(increases(degradation)) CTD docetaxel BIRC5 Text_Mining(decreases(response to substance)) CTD docetaxel BIRC5 Text_Mining(decreases(reaction)) CTD docetaxel BIRC5 Text_Mining(increases(expression)) CTD docetaxel BUB1B Text_Mining(affects(response to substance)) CTD docetaxel CASP2 Text_Mining(increases(activity)) CTD docetaxel CASP2 Text_Mining(increases(cleavage)) CTD docetaxel CASP3 Text_Mining(decreases(reaction)) CTD docetaxel CASP3 Text_Mining(increases(activity)) CTD docetaxel CASP3 Text_Mining(increases(cleavage)) CTD docetaxel CASP3 Text_Mining(increases(expression)) CTD docetaxel CASP3 Text_Mining(increases(reaction)) CTD docetaxel CASP3 Text_Mining(affects(cotreatment)) CTD docetaxel CASP3 Text_Mining(decreases(expression)) CTD docetaxel CASP8 Text_Mining(increases(activity)) CTD docetaxel CASP9 Text_Mining(decreases(reaction)) CTD docetaxel CASP9 Text_Mining(increases(activity)) CTD docetaxel CASP9 Text_Mining(increases(cleavage)) CTD docetaxel CASP9 Text_Mining(increases(reaction)) CTD docetaxel CCNB1 Text_Mining(increases(activity)) CTD docetaxel CCNB1 Text_Mining(increases(expression)) CTD docetaxel CDK1 Text_Mining(decreases(reaction)) CTD docetaxel CDK1 Text_Mining(increases(activity)) CTD docetaxel CDK1 Text_Mining(increases(response to substance)) CTD docetaxel CDK2 Text_Mining(decreases(reaction)) CTD docetaxel CDK2 Text_Mining(increases(activity)) CTD docetaxel CDKN1A Text_Mining(affects(cotreatment)) CTD docetaxel CDKN1A Text_Mining(decreases(response to substance)) CTD docetaxel CDKN1A Text_Mining(increases(expression)) CTD docetaxel CDKN1A Text_Mining(decreases(reaction)) CTD docetaxel CDKN2A Text_Mining(decreases(expression)) CTD docetaxel CHFR Text_Mining(affects(response to substance)) CTD docetaxel CHFR Text_Mining(decreases(response to substance)) CTD docetaxel CSF2 Text_Mining(increases(secretion)) CTD docetaxel CYP19A1 Text_Mining(decreases(expression)) CTD docetaxel CYP1A2 Text_Mining(affects(response to substance)) CTD docetaxel CYP1B1 Text_Mining(affects(response to substance)) CTD docetaxel CYP2D6 Text_Mining(affects(response to substance)) CTD docetaxel CYP3A4 Text_Mining(increases(response to substance)) CTD docetaxel CYP3A4 Text_Mining(increases(expression)) CTD docetaxel DPYD Text_Mining(affects(cotreatment)) CTD docetaxel DPYD Text_Mining(decreases(expression)) CTD docetaxel DPYD Text_Mining(decreases(reaction)) CTD docetaxel DPYD Text_Mining(increases(activity)) CTD docetaxel DPYD Text_Mining(decreases(activity)) CTD docetaxel DPYD Text_Mining(increases(expression)) CTD docetaxel EGFR Text_Mining(affects(cotreatment)) CTD docetaxel EGFR Text_Mining(increases(response to substance)) CTD docetaxel ERBB2 Text_Mining(affects(cotreatment)) CTD docetaxel ERBB2 Text_Mining(affects(response to substance)) CTD docetaxel ERBB2 Text_Mining(increases(response to substance)) CTD docetaxel F2R Text_Mining(decreases(response to substance)) CTD docetaxel FAS Text_Mining(increases(expression)) CTD docetaxel FGF2 Text_Mining(affects(cotreatment)) CTD docetaxel FGF2 Text_Mining(decreases(expression)) CTD docetaxel FMO2 Text_Mining(affects(response to substance)) CTD docetaxel FMO3 Text_Mining(affects(response to substance)) CTD docetaxel GADD45A Text_Mining(increases(expression)) CTD docetaxel GADD45A Text_Mining(increases(response to substance)) CTD docetaxel GSTP1 Text_Mining(increases(response to substance)) CTD docetaxel H2AFX Text_Mining(decreases(reaction)) CTD docetaxel H2AFX Text_Mining(increases(expression)) CTD docetaxel H2AFX Text_Mining(increases(reaction)) CTD docetaxel HRAS Text_Mining(increases(activity)) CTD docetaxel HRAS Text_Mining(increases(expression)) CTD docetaxel IL6 Text_Mining(increases(expression)) CTD docetaxel JUN Text_Mining(increases(phosphorylation)) CTD docetaxel JUN Text_Mining(increases(reaction)) CTD docetaxel KIF12 Text_Mining(decreases(response to substance)) CTD docetaxel KIF5A Text_Mining(decreases(response to substance)) CTD docetaxel KIFC3 Text_Mining(decreases(response to substance)) CTD docetaxel KLK3 Text_Mining(decreases(expression)) CTD docetaxel KLK3 Text_Mining(decreases(secretion)) CTD docetaxel KRT18 Text_Mining(increases(expression)) CTD docetaxel KRT18 Text_Mining(increases(metabolic processing)) CTD docetaxel MAD2L1 Text_Mining(affects(response to substance)) CTD docetaxel MAPK1 Text_Mining(increases(activity)) CTD docetaxel MAPK1 Text_Mining(increases(phosphorylation)) CTD docetaxel MAPK3 Text_Mining(increases(activity)) CTD docetaxel MAPK3 Text_Mining(increases(phosphorylation)) CTD docetaxel MCAM Text_Mining(decreases(response to substance)) CTD docetaxel MCL1 Text_Mining(increases(expression)) CTD docetaxel MCL1 Text_Mining(decreases(reaction)) CTD docetaxel MCM2 Text_Mining(affects(cotreatment)) CTD docetaxel MCM2 Text_Mining(decreases(expression)) CTD docetaxel MDM2 Text_Mining(increases(expression)) CTD docetaxel MMP9 Text_Mining(affects(cotreatment)) CTD docetaxel MMP9 Text_Mining(decreases(expression)) CTD docetaxel NPPB Text_Mining(increases(expression)) CTD docetaxel NR1I2 Text_Mining(affects(binding)) CTD docetaxel NR1I2 Text_Mining(increases(activity)) CTD docetaxel NR1I2 Text_Mining(increases(expression)) CTD docetaxel NR1I2 Text_Mining(increases(reaction)) CTD docetaxel PARP1 Text_Mining(decreases(reaction)) CTD docetaxel PARP1 Text_Mining(increases(cleavage)) CTD docetaxel PARP1 Text_Mining(increases(expression)) CTD docetaxel PARP1 Text_Mining(increases(reaction)) CTD docetaxel PGR Text_Mining(decreases(expression)) CTD docetaxel POR Text_Mining(increases(response to substance)) CTD docetaxel PSIP1 Text_Mining(increases(cleavage)) CTD docetaxel PTGS2 Text_Mining(increases(expression)) CTD docetaxel PTK2 Text_Mining(increases(cleavage)) CTD docetaxel RAD50 Text_Mining(affects(cotreatment)) CTD docetaxel RAD50 Text_Mining(decreases(expression)) CTD docetaxel RAF1 Text_Mining(increases(expression)) CTD docetaxel RB1 Text_Mining(affects(cotreatment)) CTD docetaxel RB1 Text_Mining(decreases(expression)) CTD docetaxel RB1 Text_Mining(decreases(phosphorylation)) CTD docetaxel RGS10 Text_Mining(increases(response to substance)) CTD docetaxel RGS17 Text_Mining(increases(response to substance)) CTD docetaxel TNF Text_Mining(decreases(expression)) CTD docetaxel TNFRSF10A Text_Mining(decreases(reaction)) CTD docetaxel TNFRSF10A Text_Mining(increases(expression)) CTD docetaxel TNFRSF10B Text_Mining(decreases(reaction)) CTD docetaxel TNFRSF10B Text_Mining(increases(expression)) CTD docetaxel TNFSF10 Text_Mining(increases(cleavage)) CTD docetaxel TNFSF10 Text_Mining(increases(reaction)) CTD docetaxel TP53 Text_Mining(affects(cotreatment)) CTD docetaxel TP53 Text_Mining(increases(expression)) CTD docetaxel TP53 Text_Mining(decreases(expression)) CTD docetaxel TP53 Text_Mining(decreases(ubiquitination)) CTD docetaxel TP53 Text_Mining(increases(ubiquitination)) CTD docetaxel TP53 Text_Mining(decreases(response to substance)) CTD docetaxel TP53 Text_Mining(affects(reaction)) CTD docetaxel TP53 Text_Mining(decreases(reaction)) CTD docetaxel TUBB Text_Mining(increases(expression)) CTD docetaxel TUBB Text_Mining(decreases(reaction)) CTD docetaxel TUBB Text_Mining(increases(response to substance)) CTD docetaxel TUBB Text_Mining(decreases(response to substance)) CTD docetaxel TYMP Text_Mining(affects(cotreatment)) CTD docetaxel TYMP Text_Mining(increases(expression)) CTD docetaxel TYMS Text_Mining(decreases(reaction)) CTD docetaxel TYMS Text_Mining(increases(activity)) CTD docetaxel TYMS Text_Mining(increases(expression)) CTD docetaxel TYMS Text_Mining(decreases(expression)) CTD docetaxel TYMS Text_Mining(increases(reaction)) CTD docetaxel TYMS Text_Mining(affects(cotreatment)) CTD docetaxel TYMS Text_Mining(increases(response to substance)) CTD docetaxel UMPS Text_Mining(affects(cotreatment)) CTD docetaxel UMPS Text_Mining(increases(expression)) CTD docetaxel UMPS Text_Mining(increases(reaction)) CTD docetaxel VEGFA Text_Mining(decreases(expression)) CTD docetaxel VEGFA Text_Mining(increases(reaction)) CTD docetaxel XIAP Text_Mining(decreases(expression)) CTD docetaxel XIAP Text_Mining(decreases(response to substance)) CTD docetaxel XRCC5 Text_Mining(affects(cotreatment)) CTD docetaxel XRCC5 Text_Mining(decreases(expression)) CTD docetaxel XRCC6 Text_Mining(affects(cotreatment)) CTD docetaxel XRCC6 Text_Mining(decreases(expression)) CTD docetaxel AR Ratio Potency (uM)=0.00477156(uM) D4 PubChem docetaxel ESR1 ER Potency (uM)=0.0595572(uM) D4 PubChem docetaxel ESR1 Potency-Replicate_1=0.0596(uM) D4 PubChem docetaxel NR3C1 Potency-Replicate_1=10.6822(uM) D4 PubChem docetaxel NR3C1 None=None(uM) D4 PubChem docetaxel TDP1 Potency=0.0011(uM) D4 PubChem docetaxel TDP1 Potency=0.0012(uM) D4 PubChem docetaxel TDP1 Potency=0.0033(uM) D4 PubChem