Drug Gene Type Source o6-benzylguanine AGT Text_Mining(decreases(response to substance)) CTD o6-benzylguanine AGT Text_Mining(increases(response to substance)) CTD o6-benzylguanine AGT Text_Mining(decreases(activity)) CTD o6-benzylguanine AOX1 Text_Mining(affects(metabolic processing)) CTD o6-benzylguanine CDKN1A Text_Mining(affects(cotreatment)) CTD o6-benzylguanine CDKN1A Text_Mining(increases(expression)) CTD o6-benzylguanine CDKN1A Text_Mining(affects(localization)) CTD o6-benzylguanine CDKN1B Text_Mining(affects(cotreatment)) CTD o6-benzylguanine CDKN1B Text_Mining(decreases(expression)) CTD o6-benzylguanine CHEK1 Text_Mining(increases(activity)) CTD o6-benzylguanine CHEK1 Text_Mining(increases(phosphorylation)) CTD o6-benzylguanine CHEK1 Text_Mining(increases(reaction)) CTD o6-benzylguanine CYP1A1 Text_Mining(affects(oxidation)) CTD o6-benzylguanine CYP1A1 Text_Mining(increases(metabolic processing)) CTD o6-benzylguanine CYP1A1 Text_Mining(decreases(reaction)) CTD o6-benzylguanine CYP1A1 Text_Mining(decreases(activity)) CTD o6-benzylguanine CYP1A2 Text_Mining(affects(metabolic processing)) CTD o6-benzylguanine CYP1A2 Text_Mining(decreases(reaction)) CTD o6-benzylguanine CYP1A2 Text_Mining(increases(metabolic processing)) CTD o6-benzylguanine CYP1A2 Text_Mining(decreases(activity)) CTD o6-benzylguanine FECH Text_Mining(affects(cotreatment)) CTD o6-benzylguanine FECH Text_Mining(decreases(response to substance)) CTD o6-benzylguanine MGMT Text_Mining(affects(cotreatment)) CTD o6-benzylguanine MGMT Text_Mining(decreases(response to substance)) CTD o6-benzylguanine MGMT Text_Mining(affects(metabolic processing)) CTD o6-benzylguanine MGMT Text_Mining(decreases(activity)) CTD o6-benzylguanine MGMT Text_Mining(decreases(reaction)) CTD o6-benzylguanine MGMT Text_Mining(increases(response to substance)) CTD o6-benzylguanine MGMT Text_Mining(increases(alkylation)) CTD o6-benzylguanine MGMT Text_Mining(affects(folding)) CTD o6-benzylguanine MLH1 Text_Mining(affects(cotreatment)) CTD o6-benzylguanine MLH1 Text_Mining(affects(expression)) CTD o6-benzylguanine MSH2 Text_Mining(affects(cotreatment)) CTD o6-benzylguanine MSH2 Text_Mining(affects(expression)) CTD o6-benzylguanine PMS1 Text_Mining(affects(cotreatment)) CTD o6-benzylguanine PMS1 Text_Mining(affects(expression)) CTD o6-benzylguanine PMS2 Text_Mining(affects(cotreatment)) CTD o6-benzylguanine PMS2 Text_Mining(affects(expression)) CTD o6-benzylguanine TP53 Text_Mining(affects(cotreatment)) CTD o6-benzylguanine TP53 Text_Mining(increases(expression)) CTD o6-benzylguanine TP53 Text_Mining(increases(response to substance)) CTD o6-benzylguanine CYP1A2 None=None(uM) D4 PubChem o6-benzylguanine CYP1A2 AC50=1000.0(nM) D4 ChEMBL o6-benzylguanine CYP2C19 Potency=6.3096(uM) D4 PubChem o6-benzylguanine CYP2C19 None=None(uM) D4 PubChem o6-benzylguanine CYP2C19 Potency=6309.6(nM) D4 ChEMBL o6-benzylguanine CYP2C19 AC50=6309.57(nM) D4 ChEMBL o6-benzylguanine CYP3A4 Potency=7.9433(uM) D4 PubChem o6-benzylguanine CYP3A4 None=None(uM) D4 PubChem o6-benzylguanine CYP3A4 AC50=7943.28(nM) D4 ChEMBL o6-benzylguanine CYP3A4 Potency=7943.3(nM) D4 ChEMBL o6-benzylguanine DRD3 None=None(uM) D4 PubChem o6-benzylguanine MGMT Activity=None(Unspecified) D4 ChEMBL o6-benzylguanine MGMT Inhibition=None(Unspecified) D4 ChEMBL