Drug Gene Type Source zafirlukast ABCB11 Text_Mining(decreases(activity)) CTD zafirlukast ABCC1 Text_Mining(decreases(reaction)) CTD zafirlukast ABCC1 Text_Mining(decreases(response to substance)) CTD zafirlukast CXCL8 Text_Mining(decreases(reaction)) CTD zafirlukast CXCL8 Text_Mining(increases(activity)) CTD zafirlukast CXCL8 Text_Mining(increases(expression)) CTD zafirlukast CYP1A2 Text_Mining(decreases(reaction)) CTD zafirlukast CYP1A2 Text_Mining(increases(metabolic processing)) CTD zafirlukast CYP2C19 Text_Mining(decreases(reaction)) CTD zafirlukast CYP2C19 Text_Mining(increases(metabolic processing)) CTD zafirlukast CYP2C19 Text_Mining(decreases(activity)) CTD zafirlukast CYP2C8 Text_Mining(decreases(activity)) CTD zafirlukast CYP2C9 Text_Mining(affects(metabolic processing)) CTD zafirlukast CYP2C9 Text_Mining(decreases(reaction)) CTD zafirlukast CYP2C9 Text_Mining(increases(metabolic processing)) CTD zafirlukast CYP2C9 Text_Mining(decreases(activity)) CTD zafirlukast CYP3A4 Text_Mining(increases(metabolic processing)) CTD zafirlukast CYP3A4 Text_Mining(decreases(reaction)) CTD zafirlukast CYP3A4 Text_Mining(decreases(activity)) CTD zafirlukast CYSLTR1 Text_Mining(affects(binding)) CTD zafirlukast CYSLTR1 Text_Mining(decreases(activity)) CTD zafirlukast CYSLTR1 Text_Mining(decreases(reaction)) CTD zafirlukast CYSLTR1 Text_Mining(affects(abundance)) CTD zafirlukast CYSLTR1 Text_Mining(increases(abundance)) CTD zafirlukast CYSLTR1 Text_Mining(increases(reaction)) CTD zafirlukast CYSLTR1 Text_Mining(increases(response to substance)) CTD zafirlukast CYSLTR1 Text_Mining(increases(activity)) CTD zafirlukast CYSLTR1 Text_Mining(increases(expression)) CTD zafirlukast CYSLTR2 Text_Mining(affects(binding)) CTD zafirlukast CYSLTR2 Text_Mining(decreases(activity)) CTD zafirlukast CYSLTR2 Text_Mining(decreases(reaction)) CTD zafirlukast EDN1 Text_Mining(decreases(reaction)) CTD zafirlukast EDN1 Text_Mining(increases(expression)) CTD zafirlukast EDN1 Text_Mining(decreases(expression)) CTD zafirlukast IFNG Text_Mining(affects(cotreatment)) CTD zafirlukast IFNG Text_Mining(decreases(reaction)) CTD zafirlukast IFNG Text_Mining(increases(secretion)) CTD zafirlukast IL6 Text_Mining(decreases(reaction)) CTD zafirlukast IL6 Text_Mining(increases(activity)) CTD zafirlukast IL6 Text_Mining(increases(expression)) CTD zafirlukast RNASE3 Text_Mining(decreases(expression)) CTD zafirlukast SLC22A2 Text_Mining(decreases(reaction)) CTD zafirlukast SLC22A2 Text_Mining(increases(uptake)) CTD zafirlukast SLC47A1 Text_Mining(decreases(reaction)) CTD zafirlukast SLC47A1 Text_Mining(increases(uptake)) CTD zafirlukast SLC47A2 Text_Mining(decreases(reaction)) CTD zafirlukast SLC47A2 Text_Mining(increases(uptake)) CTD zafirlukast TNF Text_Mining(decreases(reaction)) CTD zafirlukast TNF Text_Mining(increases(activity)) CTD zafirlukast TNF Text_Mining(increases(expression)) CTD zafirlukast AHR AhR Potency (uM)=22.3838(uM) D4 PubChem zafirlukast AHR Potency-Replicate_1=26.6032(uM) D4 PubChem zafirlukast AR Potency-Replicate_1=23.9145(uM) D4 PubChem zafirlukast BAZ2B Potency=50.1187(uM) D4 PubChem zafirlukast BAZ2B Potency=50118.7(nM) D4 ChEMBL zafirlukast BCL2L1 None=None(uM) D4 PubChem zafirlukast CACNA1B IC50=None(uM) D4 PubChem zafirlukast CACNA1H None=None(uM) D4 PubChem zafirlukast CYP1A2 Inhibition=None(Unspecified) D4 ChEMBL zafirlukast CYP2C19 Inhibition=None(Unspecified) D4 ChEMBL zafirlukast CYP2C9 Inhibition=None(Unspecified) D4 ChEMBL zafirlukast CYP2D6 Inhibition=None(Unspecified) D4 ChEMBL zafirlukast EIF4H IC50=None(uM) D4 PubChem zafirlukast GFER None=None(uM) D4 PubChem zafirlukast GMNN Potency=21.136(uM) D4 PubChem zafirlukast KAT2A Potency=7.0795(uM) D4 PubChem zafirlukast KAT2A Potency=22.3872(uM) D4 PubChem zafirlukast KAT2A Potency=22387.2(nM) D4 ChEMBL zafirlukast KAT2A Potency=7079.5(nM) D4 ChEMBL zafirlukast KCNQ1 None=None(uM) D4 PubChem zafirlukast MAPK1 Potency=28.1838(uM) D4 PubChem zafirlukast MAPK1 Potency=28183.8(nM) D4 ChEMBL zafirlukast NFE2L2 Potency-Replicate_1=29.847(uM) D4 PubChem zafirlukast NFE2L2 Ratio Potency (uM)=29.847(uM) D4 PubChem zafirlukast NOD1 EC50=None(uM) D4 PubChem zafirlukast NR3C1 Potency-Replicate_1=11.9856(uM) D4 PubChem zafirlukast NRP2 None=None(uM) D4 PubChem zafirlukast POLB Potency=56.2341(uM) D4 PubChem zafirlukast POLB Potency=56234.1(nM) D4 ChEMBL zafirlukast PPARG Potency-Replicate_1=0.1693(uM) D4 PubChem zafirlukast PPARG Ratio Potency (uM)=0.197391(uM) D4 PubChem zafirlukast PPP1CA None=None(uM) D4 PubChem zafirlukast SAE1 IC50=None(uM) D4 PubChem zafirlukast UBA2 IC50=None(uM) D4 PubChem zafirlukast UBE2I IC50=None(uM) D4 PubChem zafirlukast USP1 Potency=35.4813(uM) D4 PubChem zafirlukast VDR Potency=50.1187(uM) D4 PubChem