Drug Gene Type Source calyculin A AKT1 Text_Mining(decreases(phosphorylation)) CTD calyculin A AKT1 Text_Mining(decreases(reaction)) CTD calyculin A ARHGEF17 Text_Mining(affects(cotreatment)) CTD calyculin A ARHGEF17 Text_Mining(decreases(reaction)) CTD calyculin A ARHGEF17 Text_Mining(increases(activity)) CTD calyculin A BCL2L1 Text_Mining(affects(cotreatment)) CTD calyculin A BCL2L1 Text_Mining(decreases(expression)) CTD calyculin A BCL2L1 Text_Mining(decreases(reaction)) CTD calyculin A BCL2L1 Text_Mining(increases(expression)) CTD calyculin A CASR Text_Mining(increases(phosphorylation)) CTD calyculin A CASR Text_Mining(increases(reaction)) CTD calyculin A CCND1 Text_Mining(decreases(expression)) CTD calyculin A CCND1 Text_Mining(decreases(reaction)) CTD calyculin A CREBBP Text_Mining(increases(phosphorylation)) CTD calyculin A CTNNB1 Text_Mining(increases(phosphorylation)) CTD calyculin A CYP1B1 Text_Mining(increases(expression)) CTD calyculin A CYP1B1 Text_Mining(increases(reaction)) CTD calyculin A EIF4EBP1 Text_Mining(decreases(phosphorylation)) CTD calyculin A EIF4EBP1 Text_Mining(decreases(reaction)) CTD calyculin A FOS Text_Mining(increases(expression)) CTD calyculin A LCP1 Text_Mining(increases(phosphorylation)) CTD calyculin A LCP1 Text_Mining(decreases(reaction)) CTD calyculin A LIF Text_Mining(affects(cotreatment)) CTD calyculin A LIF Text_Mining(increases(phosphorylation)) CTD calyculin A LIF Text_Mining(decreases(expression)) CTD calyculin A MCL1 Text_Mining(affects(cotreatment)) CTD calyculin A MCL1 Text_Mining(decreases(expression)) CTD calyculin A MCL1 Text_Mining(decreases(reaction)) CTD calyculin A MCL1 Text_Mining(increases(expression)) CTD calyculin A PDX1 Text_Mining(affects(localization)) CTD calyculin A PDX1 Text_Mining(decreases(reaction)) CTD calyculin A PRKG1 Text_Mining(affects(cotreatment)) CTD calyculin A PRKG1 Text_Mining(decreases(reaction)) CTD calyculin A PRKG1 Text_Mining(increases(activity)) CTD calyculin A RB1 Text_Mining(decreases(phosphorylation)) CTD calyculin A RB1 Text_Mining(decreases(reaction)) CTD calyculin A RBL1 Text_Mining(decreases(phosphorylation)) CTD calyculin A RBL1 Text_Mining(decreases(reaction)) CTD calyculin A RBL2 Text_Mining(decreases(phosphorylation)) CTD calyculin A RBL2 Text_Mining(decreases(reaction)) CTD calyculin A RELA Text_Mining(decreases(activity)) CTD calyculin A RELA Text_Mining(decreases(reaction)) CTD calyculin A RPS6 Text_Mining(decreases(phosphorylation)) CTD calyculin A RPS6 Text_Mining(decreases(reaction)) CTD calyculin A STAT3 Text_Mining(affects(cotreatment)) CTD calyculin A STAT3 Text_Mining(increases(phosphorylation)) CTD calyculin A HTT Potency=1122.0(nM) D4 ChEMBL