Drug Gene Type Source 5-Methylurapidil ADRA1A Text_Mining(affects(binding)) CTD 5-Methylurapidil ADRA1A Text_Mining(decreases(reaction)) CTD 5-Methylurapidil ADRA1A Text_Mining(increases(abundance)) CTD 5-Methylurapidil ADRA1A Text_Mining(increases(activity)) CTD 5-Methylurapidil ADRA1A Text_Mining(decreases(activity)) CTD 5-Methylurapidil ADRA1D Text_Mining(affects(binding)) CTD 5-Methylurapidil HTR1A Text_Mining(affects(binding)) CTD 5-Methylurapidil HTR1A Text_Mining(increases(activity)) CTD 5-Methylurapidil CYP3A4 Potency=19.9526(uM) D4 PubChem 5-Methylurapidil CYP3A4 None=None(uM) D4 PubChem 5-Methylurapidil DRD3 None=None(uM) D4 PubChem